Interaction of KATP channel modulators with sulfonylurea receptor SUR2B: Implication for tetramer formation and allosteric coupling of subunits

Molecular Pharmacology

Volumn 61, Issue 2, 2002, Pages 407-414

  Löffler Walz, Cornelia ^a   Hambrock, Annette ^a   Quast, Ulrich ^a  

^a UNIVERSITY OF TÜBINGEN   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

2 CYANO 1 (1,1 DIMETHYLPROPYL) 3 (3 PYRIDYL)GUANIDINE; ADENOSINE TRIPHOSPHATE; ADENOSINE TRIPHOSPHATE MAGNESIUM; GLIBENCLAMIDE; PINACIDIL; POTASSIUM; POTASSIUM CHANNEL; RECEPTOR SUBTYPE; RECEPTOR SUBUNIT; SULFONYLUREA RECEPTOR; TETRAMER; TRITIUM;

ALLOSTERISM; ARTICLE; BINDING AFFINITY; BINDING SITE; DRUG BINDING; DRUG BINDING SITE; DRUG EFFECT; DRUG RECEPTOR BINDING; EMBRYO; HUMAN; HUMAN CELL; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; SMOOTH MUSCLE;

ADENOSINE TRIPHOSPHATE; ALLOSTERIC REGULATION; AMINO ACID SUBSTITUTION; ANIMALS; ANTI-ARRHYTHMIA AGENTS; ATP-BINDING CASSETTE TRANSPORTERS; BINDING SITES; CELLS, CULTURED; DRUG INTERACTIONS; GLYBURIDE; GUANIDINES; HUMANS; MEMBRANE PROTEINS; MICE; MODELS, BIOLOGICAL; MUTAGENESIS, SITE-DIRECTED; POLYMERS; POTASSIUM CHANNELS; POTASSIUM CHANNELS, INWARDLY RECTIFYING; PYRIDINES; RECEPTORS, DRUG; TRANSFECTION; TRITIUM; VASODILATOR AGENTS;

EID: 0036151632     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.61.2.407     Document Type: Article

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