Putative conventional protein kinase C inhibitor Gödecke 6976 [12-(2-cyanoethyl)-6,7,12,13-tetrahydro-13-methyl-5-oxo-5H- indolo(2,3-a)pyrrolo(3,4-c)-carbazole] Stimulates transglutaminase activity in primary mouse epidermal keratinocytes

Journal of Pharmacology and Experimental Therapeutics

Volumn 302, Issue 1, 2002, Pages 352-358

  Shapiro, Brian A ^a   Ray, Sagarika ^a   Jung, Eunmi ^a   Allred, William T ^a   Bollag, Wendy B ^a  

^a MEDICAL COLLEGE OF GEORGIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

12 (2 CYANOETHYL) 6,7,12,13 TETRAHYDRO 13 METHYL 5 OXOINDOLO[2,3 A]PYRROLO[3,4 C]CARBAZOLE; 2 [1 (3 AMIDINOTHIOPROPYL) 1H INDOL 3 YL] 3 (1 METHYL 1H INDOL 3 YL)MALEIMIDE; 3 [1 (3 AMINOPROPYL) 3 INDOLYL] 4 (1 METHYL 3 INDOLYL) 1H PYRROLE 2,5 DIONE; BISINDOLYLMALEIMIDE; BISINDOLYLMALEIMIDE I; CALCITRIOL; CELL DNA; KERATIN; PHORBOL ESTER DERIVATIVE; PROTEIN GLUTAMINE GAMMA GLUTAMYLTRANSFERASE; PROTEIN KINASE; PROTEIN KINASE C ALPHA; PROTEIN KINASE C INHIBITOR; PROTEIN KINASE D; STAUROSPORINE; THYMIDINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL DIFFERENTIATION; CELL PROLIFERATION; CONTROLLED STUDY; DNA DETERMINATION; DNA SYNTHESIS; DRUG SELECTIVITY; ENZYME ACTIVATION; ENZYME ACTIVITY; EPIDERMIS CELL; KERATINOCYTE; MOUSE; NONHUMAN; PRIORITY JOURNAL;

ANIMALS; BLOTTING, WESTERN; CARBAZOLES; CELL DIFFERENTIATION; CELL DIVISION; DNA; ENZYME INHIBITORS; EPIDERMIS; KERATINOCYTES; MICE; MICE, INBRED ICR; NERVE GROWTH FACTORS; NUCLEIC ACID SYNTHESIS INHIBITORS; PROTEIN KINASE C; RECEPTORS, DOPAMINE D2; RECEPTORS, DOPAMINE D3; STIMULATION, CHEMICAL; TRANSGLUTAMINASES;

EID: 0036082364     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.302.1.352     Document Type: Article

References (32)

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