Preparation of 'carba' dipeptides bearing a basic side-chain at the C-terminus: Synthesis of enantiopure Boc-D-Phe-Ψ[CH2CH2]-L-Arg(NO2)-OH and Boc-D-Phe-Ψ[CH2CH2]-D-Arg(NO2)OH

Tetrahedron Letters

Volumn 42, Issue 35, 2001, Pages 6015-6018

  Kende, Andrew S ^a   Dong, Han Qing ^a   Mazur, Adam W ^b   Ebetino, Frank H ^b  

^a UNIVERSITY OF ROCHESTER   (United States)

^b PROCTER AND GAMBLE PHARMACEUTICALS   (United States)

Author keywords

'Carba' dipeptide; Arginine; Guanidination

Indexed keywords

DIPEPTIDE DERIVATIVE; TERT BUTYLOXYCARBONYL DEXTRO PHENYLALANYL PSI DIMETHYL DEXTRO NITROARGININE; TERT BUTYLOXYCARBONYL DEXTRO PHENYLALANYL PSI DIMETHYLNITROARGININE; UNCLASSIFIED DRUG;

ARTICLE; CARBOXY TERMINAL SEQUENCE; CHEMICAL REACTION; DRUG STRUCTURE; DRUG SYNTHESIS; REACTION ANALYSIS;

EID: 0035959513     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(01)01183-2     Document Type: Article

References (20)