Acetyl chloride-methanol as a convenient reagent for: A) quantitative formation of amine hydrochlorides; B) carboxylate ester formation; C) mild removal of N-t-Boc-protective group

Synthetic Communications

Volumn 28, Issue 3, 1998, Pages 471-474

  Nudelman, Ayelet ^a   Bechor, Yosi ^a   Falb, Eliezer ^a   Fischer, Bilha ^a   Wexler, Barry A ^b   Nudelman, Abraham ^a  

^a BAR ILAN UNIVERSITY   (Israel)

^b DUPONT COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINE; AMINO ACID DERIVATIVE; CARBOXYLIC ACID; CHLORIDE; ESTER; HYDROCHLORIC ACID; METHANOL; PHOSPHORAMIDIC ACID;

ARTICLE; ESTERIFICATION; SYNTHESIS;

EID: 0031906453     PISSN: 00397911     EISSN: None     Source Type: Journal    
DOI: 10.1080/00397919808005101     Document Type: Article

References (3)

1. Bois-Choussy, M., Neuville, L., Beugelmans, R. and Zhu, J. J. Org. Chem., 1996, 61, 9309-9322.
2. Cavelier, F. and Enjalbal, C., Tetrahedron Lett., 1996, 37, 5131-5134.
3. Kocienski, P. J., Protective Groups, Georg Thieme Verlag, Stuttgart, 1994, pp. 192-193, and references therein.