The role of the agonist binding site in Ca2+ inhibition of the recombinant 5-HT3A receptor

European Journal of Pharmacology

Volumn 428, Issue 2, 2001, Pages 153-161

  Niemeyer, María I ^a,b   Lummis, Sarah C R ^c,d  

^a UNIVERSITY OF CHILE   (Chile)

^b CENTRO DE ESTUDIOS CIENTÍFICOS CECS   (Chile)

^c MRC LABORATORY OF MOLECULAR BIOLOGY   (United Kingdom)

^d UNIVERSITY OF CAMBRIDGE   (United Kingdom)

Author keywords

5 HT3 receptor; Ca2+; Cation permeability; Divalent cation modulation; Ion channel; Neurotransmitter gated

Indexed keywords

1 (3 CHLOROPHENYL)BIGUANIDE; CALCIUM ION; GRANISETRON; MAGNESIUM ION; RADIOLIGAND; RECEPTOR SUBUNIT; RECOMBINANT RECEPTOR; SEROTONIN 3 RECEPTOR; SEROTONIN 3A RECEPTOR; TRITIUM; UNCLASSIFIED DRUG;

AGONIST; ARTICLE; BINDING SITE; CALCIUM BINDING; CONCENTRATION RESPONSE; CONTROLLED STUDY; HUMAN; HUMAN CELL; IMAGING; ION PERMEABILITY; LIGAND BINDING; PRIORITY JOURNAL; RECEPTOR BINDING; VOLTAGE CLAMP;

BINDING SITES; BINDING, COMPETITIVE; CALCIUM; CATIONS, DIVALENT; CELL LINE; DNA, RECOMBINANT; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; MAGNESIUM; MEMBRANE POTENTIALS; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN; SEROTONIN AGONISTS; TUMOR CELLS, CULTURED;

EID: 0035812646     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(01)01251-1     Document Type: Article

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