The effects of cyclopentane and cyclopentene analogues of GABA at recombinant GABAC receptors

European Journal of Pharmacology

Volumn 430, Issue 2-3, 2001, Pages 185-192

  Chebib, Mary ^a   Duke, Rujee K ^a   Allan, Robin D ^a   Johnston, Graham A R ^a  

^a University of Sydney   (Australia)

Author keywords

Aminobutyric acid (GABA); Cyclopentane and cyclopentene analogues of GABA; GABAC receptor; Structure activity relationship; Xenopus oocyte

Indexed keywords

3 AMINOCYCLOPENTANECARBOXYLIC ACID DERIVATIVE; 4 AMINOBUTYRIC ACID C RECEPTOR; 4 AMINOBUTYRIC ACID DERIVATIVE; 4 AMINOCYCLOPENT 1 ENE 1 CARBOXYLIC ACID DERIVATIVE; AMINE; CARBOXYLIC ACID; CYCLOPENTANE DERIVATIVE; CYCLOPENTENE DERIVATIVE; PARTIAL AGONIST; RECOMBINANT RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG EFFECT; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; ELECTRODE; ENANTIOMER; NONHUMAN; OOCYTE; PRIORITY JOURNAL; STEREOCHEMISTRY; VOLTAGE CLAMP; XENOPUS;

ANIMALS; CYCLOPENTANES; DOSE-RESPONSE RELATIONSHIP, DRUG; FEMALE; GAMMA-AMINOBUTYRIC ACID; HUMANS; MEMBRANE POTENTIALS; OOCYTES; RECEPTORS, GABA; RECOMBINANT PROTEINS; STEREOISOMERISM; XENOPUS LAEVIS;

EID: 0035798363     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(01)01390-5     Document Type: Article

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