Constitutive activity of histamine H3 receptors stably expressed in SK-N-MC cells: Display of agonism and inverse agonism by H3 antagonists

Journal of Pharmacology and Experimental Therapeutics

Volumn 299, Issue 3, 2001, Pages 908-914

  Wieland, Kerstin ^a   Bongers, Gerold ^a   Yamamoto, Yumiko ^b   Hashimoto, Takeshi ^b   Yamatodani, Atsushi ^b   Menge, Wiro M B P ^a   Timmerman, Henk ^a   Lovenberg, Timothy W ^c   Leurs, Rob ^a  

^a VU UNIVERSITY AMSTERDAM   (Netherlands)

^b OSAKA UNIVERSITY   (Japan)

^c R W JOHNSON PHARMACEUTICAL RES I   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA METHYLHISTAMINE; BURIMAMIDE; CLOBENPROPIT; CYCLIC AMP; FORSKOLIN; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR AGONIST; HISTAMINE H3 RECEPTOR ANTAGONIST; IMPENTAMINE; IODOPHENPROPIT; THIOPERAMIDE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG ACTIVITY; DRUG MECHANISM; HUMAN; HUMAN CELL; MALE; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; RAT; RECEPTOR BINDING; RECEPTOR DENSITY;

ANIMALS; BURIMAMIDE; CYCLIC AMP; HISTAMINE ANTAGONISTS; HUMANS; IMIDAZOLES; MALE; RATS; RATS, WISTAR; RECEPTORS, HISTAMINE H3; RECOMBINANT PROTEINS; THIOUREA; TUMOR CELLS, CULTURED;

EID: 0035200715     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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