Cloning and pharmacological characterization of a fourth histamine receptor (H4) expressed in bone marrow

Molecular Pharmacology

Volumn 59, Issue 3, 2001, Pages 420-426

  Liu, Changlu ^a   Ma, Xiao Jun ^a   Jiang, Xiaoxia ^a   Wilson, Sandy J ^a   Hofstra, Claudia L ^a   Blevitt, Jonathan ^a   Pyati, Jayashree ^a   Li, Xiaobing ^a   Chai, Wenying ^a   Carruthers, Nicholas ^a   Lovenberg, Timothy W ^a  

^a R W JOHNSON PHARMACEUTICAL RES I   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CIMETIDINE; DIMAPRIT; DIPHENHYDRAMINE; HISTAMINE H4 RECEPTOR; HISTAMINE RECEPTOR; LORATADINE; RANITIDINE; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ARTICLE; BONE MARROW CELL; CALCIUM MOBILIZATION; DRUG POTENCY; DRUG RECEPTOR BINDING; ENTEROCHROMAFFIN CELL; HUMAN; HUMAN CELL; MOLECULAR CLONING; NEUROTRANSMITTER RELEASE; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR GENE; SMOOTH MUSCLE CONTRACTION; STOMACH ACID SECRETION;

EID: 0035126496     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.59.3.420     Document Type: Article

References (26)

1. Basic local alignment search tool
2. Autoinhibition of brain histamine release mediated by a novel class (H3) of histamine receptor
3. Receptors mediating some actions of histamine
4. Chemical structure and sympathomimetic action of amines
5. Histamine H3 receptors in the guinea pig ileum: Evidence for a postjunctional location
6. Histamine inhibits tumor necrosis factor alpha release by mast cells through H2 and H3 receptors
7. Definition and antagonism of histamine H2-receptors
8. Relation between the inhibition constant K1 and the concentration of inhibitor which causes fifty per cent inhibition (I50) of an enzymic reaction
9. The histamine H3 receptor pharmacotherapy targets in gastrointestinal disorders
10. Graded increase in probability of eosinophilic differentiation of HL-60 promyelocytic leukemia cells induced by culture under alkaline conditions
11. Histamine-induced adherence and migration of equine eosinophils
12. Synthesis of potent non-imidazole histamine H3-receptor antagonists
13. Molecular cloning of a gene encoding the histamine H2 receptor
14. International Union of Pharmacology. XIII. Classification of histamine receptors
15. Histamine can induce leukocyte rolling in rat mesenteric venules
16. Cloning and functional expression of the human histamine H3 receptor
17. Molecular cloning and characterization of novel type of histamine receptor preferentially expressed in leukocytes
18. Pharmacologic characterization of a novel histamine receptor on human eosinophils
19. Characterization of histamine H3 receptors inhibiting 5-HT release from porcine enterochromaffin cells: Further evidence for H3 receptor heterogeneity
20. Regulation of histamine release from human basophil leukocytes: Role of H1, H2 and H3 receptors
21. CC chemokine receptors 1 and 3 are differentially regulated by IL-5 during maturation of eosinophilic HL-60 cells
22. Hyperglycosylation of eosinophil ribonucleases in a promyelocytic leukemia cell line and in differentiated peripheral blood progenitor cells
23. New analogs of burimamide as potent and selective histamine H3 receptor antagonists: The effect of chain length variation of the alkyl spacer and modifications of the N-thiourea substituent
24. Expression cloning of a cDNA encoding the bovine histamine H1 receptor