메뉴 건너뛰기




Volumn 59, Issue 3, 2001, Pages 514-523

Interactions of tryptamine derivatives with serotonin transporter species variants implicate transmembrane domain I in substrate recognition

Author keywords

[No Author keywords available]

Indexed keywords

CITALOPRAM; MAZINDOL; SEROTONIN TRANSPORTER; TRYPTAMINE;

EID: 0035122827     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.59.3.514     Document Type: Article
Times cited : (80)

References (47)
  • 4
    • 0029860223 scopus 로고    scopus 로고
    • Identification of a single amino acid, phenylalanine 586, that is responsible for high affinity interactions of tricyclic antidepressants with the human serotonin transporter
    • (1996) Mol Pharmacol , vol.50 , pp. 957-965
    • Barker, E.L.1    Blakely, R.D.2
  • 14
    • 0028577297 scopus 로고
    • Chimeric dopamine-norepinephrine transporters delineate structural domains influencing selectivity for catecholamines and 1-methyl-4-phenylpyridinium
    • (1994) Proc Natl Acad Sci USA , vol.91 , pp. 12584-12588
    • Buck, K.J.1    Amara, S.G.2
  • 19
    • 0015861774 scopus 로고
    • Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (IC50) of an enzymatic reaction
    • (1973) Biochem Pharmacol , vol.22 , pp. 3099-3108
    • Cheng, Y.1    Prusoff, W.H.2
  • 23
    • 0015860717 scopus 로고
    • Structure activity relations for the inhibition of 5-HT into rat hypothalamic homogenates by serotonin and tryptamine analogues
    • (1973) J Neurochemistry , vol.21 , pp. 883-888
    • Horn, A.S.1
  • 24
    • 0018198123 scopus 로고
    • Structure-activity relationships of serotonin neurotoxins: Effects on serotonin uptake
    • (1978) Ann NY Acad Sci , vol.305 , pp. 128-133
    • Horn, A.S.1
  • 38
    • 0002264450 scopus 로고    scopus 로고
    • The structure and function of norepinephrine, dopamine, and serotonin transporters
    • Neurotransmitter Transporters: Structure, Function, and Regulation (Reith MEA ed), Humana Press, Totowa, NJ
    • (1997) , pp. 1-28
    • Povlock, S.L.1    Amara, S.G.2
  • 41
    • 0026546876 scopus 로고
    • The molecular mechanism of "ecstasy" [3,4-methylenedioxymethamphetamine (MDMA)]: Serotonin transporters are targets for MDMA-induced serotonin release
    • (1992) Proc Natl Acad Sci USA , vol.89 , pp. 1817-1821
    • Rudnick, G.1    Wall, S.C.2
  • 42
    • 0000372083 scopus 로고    scopus 로고
    • 5-hydroxytryptamine (serotonin) receptor agonists and antagonists
    • The Pharmacological Basis of Therapeutics (Hardman JG, Limbird LE, Molinoff PB, Ruddon RW and Gilman AG eds), McGraw-Hill, New York
    • (1996) , pp. 249-263
    • Sanders-Bush, E.1    Mayer, S.E.2
  • 43
    • 0028889607 scopus 로고
    • Heterogeneity of antidepressant binding sites on the recombinant rat serotonin transporter SERT1
    • (1995) Biochemistry , vol.34 , pp. 12590-12595
    • Schloss, P.1    Betz, H.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.