Development of a homogeneous MAP kinase reporter gene screen for the identification of agonists and antagonists at the CXCR1 chemokine receptor

Journal of Biomolecular Screening

Volumn 6, Issue 1, 2001, Pages 19-27

  Rees, Stephen ^a   Martin, Duncan P ^a   Scott, Sarah V ^a   Brown, Sue H ^a   Fraser, Neil ^a   O'Shaughnessy, Celestine ^a   Beresford, Isabel J M ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 (2 AMINO 3 METHOXYPHENYL)CHROMONE; 4 (4 FLUOROPHENYL) 2 (4 METHYLSULFINYLPHENYL) 5 (4 PYRIDYL)IMIDAZOLE; CHEMOKINE RECEPTOR CXCR1; G PROTEIN COUPLED RECEPTOR; INTERLEUKIN 8; MITOGEN ACTIVATED PROTEIN KINASE;

ANIMAL CELL; ARTICLE; CHO CELL; CONTROLLED STUDY; DRUG SCREENING; ENZYME ACTIVATION; GENETIC TRANSFECTION; MAMMAL CELL; NONHUMAN; PRIORITY JOURNAL; PROTEIN FAMILY; REPORTER GENE; SIGNAL PROCESSING; SIGNAL TRANSDUCTION;

ANIMALS; CHO CELLS; CRICETINAE; DNA-BINDING PROTEINS; DRUG EVALUATION, PRECLINICAL; ENZYME ACTIVATION; ETS-DOMAIN PROTEIN ELK-4; FLAVONOIDS; GENES, REPORTER; HUMANS; INTERLEUKIN-8; MITOGEN-ACTIVATED PROTEIN KINASES; PERTUSSIS TOXIN; RECEPTORS, INTERLEUKIN-8A; SIGNAL TRANSDUCTION; TRANSFECTION; VIRULENCE FACTORS, BORDETELLA;

ANIMALIA; CRICETINAE; CRICETULUS GRISEUS; MAMMALIA;

EID: 0035113925     PISSN: 10870571     EISSN: None     Source Type: Journal    
DOI: 10.1089/108705701750066999     Document Type: Article

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