Studies of the human, rat, and guinea pig Y4 receptors using neuropeptide Y analogues and two distinct radioligands

Peptides

Volumn 22, Issue 3, 2001, Pages 351-356

  Berglund, Magnus M ^a   Lundell, Ingrid ^a   Eriksson, Henrik ^a   Söll, Richard ^b   Beck Sickinger, Annette G ^b   Larhammar, Dan ^a  

^a UPPSALA UNIVERSITY   (Sweden)

^b ETH ZURICH   (Switzerland)

Author keywords

Alanine scan; Binding; G protein coupled receptor; Neuropeptide Y (NPY); Pancreatic polypeptide (PP); Peptide YY (PYY); Structure activity relations; Two site model; Y4

Indexed keywords

ALANINE; AMINOCAPROIC ACID; NEUROPEPTIDE Y DERIVATIVE; NEUROPEPTIDE Y4 RECEPTOR; PANCREAS POLYPEPTIDE; PEPTIDE YY; PROLINE; RADIOLIGAND; RECEPTOR SUBTYPE;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING SITE; CONCENTRATION RESPONSE; CONTROLLED STUDY; GUINEA PIG; HUMAN; HUMAN CELL; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING; SPECIES DIFFERENCE; STRUCTURE ACTIVITY RELATION; TISSUE DISTRIBUTION;

AMINO ACIDS; ANIMALS; BINDING SITES; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; GUINEA PIGS; HUMANS; MUTAGENESIS, SITE-DIRECTED; NEUROPEPTIDE Y; PROTEIN BINDING; RADIOLIGAND ASSAY; RATS; RECEPTORS, NEUROPEPTIDE Y; SPECIES SPECIFICITY;

CAVIA PORCELLUS; SUIDAE; SUS SCROFA;

EID: 0035091359     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0196-9781(01)00337-0     Document Type: Article

References (21)

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7. The guinea-pig is not a rodent
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