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Volumn 9, Issue 2, 2001, Pages 431-444

High affinity central benzodiazepine receptor ligands. Part 2: Quantitative structure-activity relationships and comparative molecular field analysis of pyrazolo[4,3-c]quinolin-3-ones

(10) Savini, L b Chiasserini, L b Pellerano, C b Biggio, G c Maciocco, E c Serra, M c Cinone, N a,d Carrieri, A a Altomare, C a Carotti, A a

a UNIVERSITY OF BARI (Italy)

b UNIVERSITY OF SIENA (Italy)

c UNIVERSITY OF CAGLIARI (Italy)

d UNIVERSITY OF CHIETI (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

2 PHENYL 5H PYRAZOLO[4,3 C]QUINOLIN 3 ONE; 2,5 DIHYDROPYRAZOLO[4,3 C]QUINOLIN 3(3H) ONE DERIVATIVE; BENZODIAZEPINE RECEPTOR; KNI 547; LIGAND; N TERT BUTYL 3 [3 (2,3 DIMETHYLSUCCINYL)AMINO 2 HYDROXY 4 PHENYLBUTANOYL] 1,3 THIAZOLIDINE 4 CARBOXAMIDE; QUINOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; COMPARATIVE STUDY; DRUG BINDING SITE; DRUG CONFORMATION; DRUG SYNTHESIS; HYDROGEN BOND; MALE; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RAT; RECEPTOR AFFINITY; STEREOSPECIFICITY;

ANIMALS; BINDING, COMPETITIVE; CEREBRAL CORTEX; ELECTROSTATICS; GABA AGONISTS; GABA ANTAGONISTS; INHIBITORY CONCENTRATION 50; LIGANDS; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MODELS, MOLECULAR; PROTEIN BINDING; PYRAZOLES; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; QUINOLONES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-A;

EID: 0035087606 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(00)00262-5 Document Type: Article

Times cited : (27)

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