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Volumn 49, Issue 5, 2001, Pages 606-612

Ethenesulfonamide derivatives, a novel class of orally active endothelin-A receptor antagonists

(9) Harada, H a Kazami, J I a Watanuki, S a Tsuzuki, R a Sudoh, K a Fujimori, A a Tanaka, A a Tsukamoto, S I a Yanagisawa, I a

a ASTELLAS PHARMA INC (Japan)

Author keywords

Endothelin antagonist; ETA selective; Ethenesulfonamide

Indexed keywords

BOSENTAN; ENDOTHELIN 1; ENDOTHELIN A RECEPTOR ANTAGONIST; N [6 (2 FLUOROETHOXY) 5 (2 METHOXYPHENOXY) 2 (PYRIMIDIN 2 YL)PYRIMIDIN 4 YL] 2 PHENYLETHENESULFONAMIDE; N [6 (2 HYDROXYETHOXY) 5 (2 METHOXYPHENOXY) 2 (PYRIMIDIN 2 YL)PYRIMIDIN 4 YL] 2 PHENYLETHENESULFONAMIDATE; SULFONAMIDE; UNCLASSIFIED DRUG; YM 62899;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ANTIHYPERTENSIVE ACTIVITY; ARTICLE; BLOOD VESSEL REACTIVITY; CONTROLLED STUDY; DOSE RESPONSE; DRUG ANTAGONISM; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; IC 50; MALE; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

ANIMALS; AORTA, THORACIC; BLOOD PRESSURE; DECEREBRATE STATE; FEMALE; INDICATORS AND REAGENTS; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MUSCLE CONTRACTION; MUSCLE, SMOOTH, VASCULAR; PREGNANCY; RATS; RATS, WISTAR; RECEPTOR, ENDOTHELIN A; RECEPTOR, ENDOTHELIN B; RECEPTORS, ENDOTHELIN; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 0034985845 PISSN: 00092363 EISSN: None Source Type: Journal
DOI: 10.1248/cpb.49.606 Document Type: Article

Times cited : (12)

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