Arylpiperazine derivatives of 3-propyl-β-Tetralonohydantoin as new 5-HT1A and 5-HT2A receptor ligands

Polish Journal of Pharmacology

Volumn 53, Issue 4, 2001, Pages 395-401

  Byrtus, H ^a   Pawlowski, M ^a   Duszynska B ^a   Wesolowska, A ^a   Chojnacka Wojcik E ^a   Bojarski, A J ^a  

^a INSTITUTE OF PHARMACOLOGY   (Poland)

Author keywords

1 arylpiperazine derivatives; 3 propyl tetralonohydantoins; 5 HT1A and 5 HT2A receptor affinity; Structure activity relationship

Indexed keywords

HYDANTOIN DERIVATIVE; PIPERAZINE DERIVATIVE; POSTSYNAPTIC RECEPTOR; PRESYNAPTIC RECEPTOR; PSYCHOTROPIC AGENT; SEROTONIN 1A AGONIST; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 2A ANTAGONIST; SEROTONIN 2A RECEPTOR;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BODY TEMPERATURE; BRAIN CORTEX; CONTROLLED STUDY; DRUG STRUCTURE; HEAD TWITCH; HIPPOCAMPUS; IN VIVO STUDY; LIGAND BINDING; MALE; MOUSE; NONHUMAN; RAT; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; BODY TEMPERATURE; CEREBRAL CORTEX; HEAD MOVEMENTS; HIPPOCAMPUS; HYDANTOINS; LIGANDS; LIP; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MICE; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN AGENTS; SPIRO COMPOUNDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0034748583     PISSN: 12306002     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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