메뉴 건너뛰기




Volumn 390, Issue 1-2, 2000, Pages 67-73

Inactivation of 5-HT(1A) receptors in hippocampal and cortical homogenates

Author keywords

5 HT(1A) receptor; 35S GTP S binding assay; Cortex; EEDQ; Hippocampus; Receptor reserve; Spare receptor

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 2 ETHOXY 1(2H) QUINOLINECARBOXYLIC ACID ETHYL ESTER; ALKYLATING AGENT; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; RECEPTOR RESERVE; SEROTONIN; SEROTONIN 1A RECEPTOR; SULFUR 35;

EID: 0034712019     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(00)00032-7     Document Type: Article
Times cited : (11)

References (32)
  • 2
    • 0022414001 scopus 로고
    • 2-adrenoceptor binding and function after irreversible inactivation by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ)
    • 2-adrenoceptor binding and function after irreversible inactivation by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ). Eur. J. Pharmacol. 116:1985;175-178.
    • (1985) Eur. J. Pharmacol. , vol.116 , pp. 175-178
    • Adler, C.H.1    Meller, E.2    Goldstein, M.3
  • 3
    • 0032545813 scopus 로고    scopus 로고
    • 35S]GTPγS binding in rat hippocampal membranes
    • 35S]GTPγS binding in rat hippocampal membranes. Eur. J. Pharmacol. 343:1998;303-312.
    • (1998) Eur. J. Pharmacol. , vol.343 , pp. 303-312
    • Alper, R.H.1    Nelson, D.L.2
  • 5
    • 0026557512 scopus 로고
    • 1A autoreceptor-mediated inhibition of neurotransmitter synthesis: Relationship to receptor reserve
    • 1A autoreceptor-mediated inhibition of neurotransmitter synthesis: relationship to receptor reserve. Neuropharmacology. 31:1992;451-459.
    • (1992) Neuropharmacology , vol.31 , pp. 451-459
    • Bohmaker, K.1    Bordi, F.2    Meller, E.3
  • 7
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
    • Bradford M.M. A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal. Biochem. 72:1976;248-254.
    • (1976) Anal. Biochem. , vol.72 , pp. 248-254
    • Bradford, M.M.1
  • 9
    • 0022555590 scopus 로고
    • 1A receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in guinea pig and rat hippocampal membranes
    • 1A receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in guinea pig and rat hippocampal membranes. J. Pharmacol. Exp. Ther. 238:1986;248-253.
    • (1986) J. Pharmacol. Exp. Ther. , vol.238 , pp. 248-253
    • De Vivo, M.1    Maayani, S.2
  • 10
    • 0023837915 scopus 로고
    • 1A receptors which inhibit cAMP production in hippocampal and cortical neurons in primary culture
    • 1A receptors which inhibit cAMP production in hippocampal and cortical neurons in primary culture. Mol. Pharmacol. 33:1988;178-186.
    • (1988) Mol. Pharmacol. , vol.33 , pp. 178-186
    • Dumuis, A.1    Sebben, M.2    Bockaert, J.3
  • 11
    • 0021941757 scopus 로고
    • Irreversible blockade of central 5-HT binding sites by 8-methoxy-2′-chloro-PAT
    • Emerit M.B., Gozlan H., Hall M.D., Hamon M., Marquet A. Irreversible blockade of central 5-HT binding sites by 8-methoxy-2′-chloro-PAT. Biochem. Pharmacol. 34:1985;883-892.
    • (1985) Biochem. Pharmacol. , vol.34 , pp. 883-892
    • Emerit, M.B.1    Gozlan, H.2    Hall, M.D.3    Hamon, M.4    Marquet, A.5
  • 13
    • 84981848149 scopus 로고
    • Comparison of dissociation constants and of relative efficacies of selected agonists acting on parasympathetic receptors
    • Furchgott R.F., Bursztyn P. Comparison of dissociation constants and of relative efficacies of selected agonists acting on parasympathetic receptors. Ann. NY Acad. Sci. 144:1967;882-888.
    • (1967) Ann. NY Acad. Sci. , vol.144 , pp. 882-888
    • Furchgott, R.F.1    Bursztyn, P.2
  • 14
    • 0028290841 scopus 로고
    • Differential effects of n-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on various 5-HT receptor binding sites in the rat brain
    • Gozlan H., Laporte A.-M., Thibault S., Schechter L.E., Bolaños-Jiménez F., Hamon M. Differential effects of n-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on various 5-HT receptor binding sites in the rat brain. Neuropharmacology. 33:1994;423-431.
    • (1994) Neuropharmacology , vol.33 , pp. 423-431
    • Gozlan, H.1    Laporte, A.-M.2    Thibault, S.3    Schechter, L.E.4    Bolaños-Jiménez, F.5    Hamon, M.6
  • 15
    • 0021220905 scopus 로고
    • Effect of aging on recovery of striatal dopamine receptors following N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) blockade
    • Henry J.M., Roth G.S. Effect of aging on recovery of striatal dopamine receptors following N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) blockade. Life Sci. 35:1984;899-904.
    • (1984) Life Sci. , vol.35 , pp. 899-904
    • Henry, J.M.1    Roth, G.S.2
  • 16
    • 0027283546 scopus 로고
    • Partial agonists, full agonists, antagonists: Dilemmas of definition
    • Hoyer D., Boddeke H.W.G.M. Partial agonists, full agonists, antagonists: dilemmas of definition. Trends Pharmacol. Sci. 14:1993;270-275.
    • (1993) Trends Pharmacol. Sci. , vol.14 , pp. 270-275
    • Hoyer, D.1    Boddeke, H.W.G.M.2
  • 17
    • 0030598069 scopus 로고    scopus 로고
    • 1A receptors following irreversible inactivation by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ)
    • 1A receptors following irreversible inactivation by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ). Brain Res. 728:1996;130-134.
    • (1996) Brain Res. , vol.728 , pp. 130-134
    • Keck, B.J.1    Lakoski, J.M.2
  • 18
    • 0029658721 scopus 로고    scopus 로고
    • 1A receptor turnover following irreversible blockade with EEDQ
    • 1A receptor turnover following irreversible blockade with EEDQ. NeuroReport. 7:1996;2717-2721.
    • (1996) NeuroReport , vol.7 , pp. 2717-2721
    • Keck, B.J.1    Lakoski, J.M.2
  • 19
    • 0028027657 scopus 로고
    • 1A receptor-mediated regulation of plasma neuroendocrine hormones
    • 1A receptor-mediated regulation of plasma neuroendocrine hormones. J. Pharmacol. Exp. Ther. 271:1994;1246-1252.
    • (1994) J. Pharmacol. Exp. Ther. , vol.271 , pp. 1246-1252
    • Meller, E.1    Bohmaker, K.2
  • 20
    • 0026615198 scopus 로고
    • 1A receptor-mediated hypothermia in mice: Absence of spare receptors and rapid induction of tolerance
    • 1A receptor-mediated hypothermia in mice: absence of spare receptors and rapid induction of tolerance. Pharmacol. Biochem. Behav. 43:1992;405-411.
    • (1992) Pharmacol. Biochem. Behav. , vol.43 , pp. 405-411
    • Meller, E.1    Chalfin, M.2    Bohmaker, K.3
  • 22
    • 0026099819 scopus 로고
    • A receptor binding and function by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vitro and in vivo: Effects of aging
    • A receptor binding and function by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vitro and in vivo: effects of aging. J. Neurochem. 56:1991;1241-1247.
    • (1991) J. Neurochem. , vol.56 , pp. 1241-1247
    • Miller, L.G.1    Lumpkin, M.2    Galpern, W.R.3    Greenblatt, D.J.4    Shader, R.I.5
  • 23
    • 0018231884 scopus 로고
    • Characteristics of central 5-HT receptors and their adaptive changes following intracerebral 5,7-dihydroxytryptamine administration in the rat
    • Nelson D.L., Herbet A., Bourgoin S., Glowinski J., Hamon M. Characteristics of central 5-HT receptors and their adaptive changes following intracerebral 5,7-dihydroxytryptamine administration in the rat. Mol. Pharmacol. 14:1978;983-995.
    • (1978) Mol. Pharmacol. , vol.14 , pp. 983-995
    • Nelson, D.L.1    Herbet, A.2    Bourgoin, S.3    Glowinski, J.4    Hamon, M.5
  • 25
    • 0024513755 scopus 로고
    • Irreversible and quaternary muscarinic antagonists discriminate multiple muscarinic receptor binding sites in rat brain
    • Norman A.B., Eubanks J.H., Creese I. Irreversible and quaternary muscarinic antagonists discriminate multiple muscarinic receptor binding sites in rat brain. J. Pharmacol. Exp. Ther. 248:1989;1116-1122.
    • (1989) J. Pharmacol. Exp. Ther. , vol.248 , pp. 1116-1122
    • Norman, A.B.1    Eubanks, J.H.2    Creese, I.3
  • 28
    • 0020391631 scopus 로고
    • Important concepts of receptor theory
    • Ruffolo R.R. Important concepts of receptor theory. J. Auton. Pharmacol. 2:1982;277-295.
    • (1982) J. Auton. Pharmacol. , vol.2 , pp. 277-295
    • Ruffolo, R.R.1
  • 29
    • 0023727660 scopus 로고
    • 1A binding sites inhibit forskolin-stimulated adenylate cyclase activity in calf hippocampus
    • 1A binding sites inhibit forskolin-stimulated adenylate cyclase activity in calf hippocampus. Br. J. Pharmacol. 95:1988;975-985.
    • (1988) Br. J. Pharmacol. , vol.95 , pp. 975-985
    • Schoeffter, P.1    Hoyer, D.2
  • 31
    • 0028314995 scopus 로고
    • Measurement of receptor-stimulated guanosine 5′-O-(γ-thio)triphosphate binding by G proteins
    • Weiland T., Jakobs K.H. Measurement of receptor-stimulated guanosine 5′-O-(γ-thio)triphosphate binding by G proteins. Meth. Enzymol. 237:1994;3-13.
    • (1994) Meth. Enzymol. , vol.237 , pp. 3-13
    • Weiland, T.1    Jakobs, K.H.2
  • 32
    • 0027048880 scopus 로고
    • 1A receptors negatively coupled to adenylyl cyclase activity in rat hippocampal membranes
    • 1A receptors negatively coupled to adenylyl cyclase activity in rat hippocampal membranes. Mol. Pharmacol. 41:1992;1066-1072.
    • (1992) Mol. Pharmacol. , vol.41 , pp. 1066-1072
    • Yocca, F.D.1    Iben, L.2    Meller, E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.