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Volumn 21, Issue 2, 1996, Pages 167-176

Alkylation of [3H]8-OH-DPAT binding sites in rat cerebral cortex and hippocampus

Author keywords

8 hydroxy 2 (di n propylamino)tetralin or 8 OH DPAT; L dithiothreitol; N ethoxycarbonyl 2 ethoxy 1,2 dihydroquinoline or EEDQ; N ethylmaleimide; Serotonin(1A) receptors

Indexed keywords

1 (2 METHOXYPHENYL) 4 (4 PHTHALIMIDOBUTYL)PIPERAZINE; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 2 ETHOXY 1(2H) QUINOLINECARBOXYLIC ACID ETHYL ESTER; BUSPIRONE; N TERT BUTYL 3 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL] 2 PHENYLPROPIONAMIDE; PINDOLOL; PROPRANOLOL; RITANSERIN; SEROTONIN; SEROTONIN ANTAGONIST; SPIPERONE; ALKYLATING AGENT; DIAGNOSTIC AGENT; DISULFIDE; DITHIOTHREITOL; N ETHYLMALEIMIDE; QUINOLINE DERIVATIVE; THIOL REAGENT; TRITIUM;

EID: 0029658083     PISSN: 03643190     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF02529134     Document Type: Article
Times cited : (17)

References (49)
  • 1
    • 0026761109 scopus 로고
    • 5-Hydroxytryptamine receptors
    • Zifa, E., and Fillion, G. 1992. 5-Hydroxytryptamine receptors. Pharmacol. Rev. 44:401-158.
    • (1992) Pharmacol. Rev. , vol.44 , pp. 401-1158
    • Zifa, E.1    Fillion, G.2
  • 2
    • 0027233748 scopus 로고
    • A proposed new nomenclature for 5-HT receptors
    • Humphrey, P. P. A., Hartig, P., and Hoyer, D. 1993. A proposed new nomenclature for 5-HT receptors. TIPS 14:233-235.
    • (1993) TIPS , vol.14 , pp. 233-235
    • Humphrey, P.P.A.1    Hartig, P.2    Hoyer, D.3
  • 3
    • 0027518402 scopus 로고
    • 5-Hydroxytryptamine receptors
    • Peroutka, S. J. 1993. 5-Hydroxytryptamine receptors. J. Neurochem. 60:408-416.
    • (1993) J. Neurochem. , vol.60 , pp. 408-416
    • Peroutka, S.J.1
  • 5
    • 0021892571 scopus 로고
    • 3H]8-hydroxy-2-(Di-n-Propylamino)tetralin binding to pre- and postsynaptic 5-hydroxytryptamine sites in various regions of the rat brain
    • 3H]8-hydroxy-2-(Di-n-Propylamino)tetralin binding to pre- and postsynaptic 5-hydroxytryptamine sites in various regions of the rat brain. J. Neurochem. 44:1685-1695.
    • (1985) J. Neurochem. , vol.44 , pp. 1685-1695
    • Hall, M.1    El Mestikawy, S.2    Emerit, M.B.3    Pichat, L.4    Hamon, M.5    Gozlan, H.6
  • 7
    • 0025962706 scopus 로고
    • Autoradiography of serotonin receptor subtypes in the central nervous system
    • Radja, F., Laporte, A. M., Daval, G., Vergé, D., Gozlan, H., and Hamon, M. 1991. Autoradiography of serotonin receptor subtypes in the central nervous system. Neurochem. Int. 18:1-15.
    • (1991) Neurochem. Int. , vol.18 , pp. 1-15
    • Radja, F.1    Laporte, A.M.2    Daval, G.3    Vergé, D.4    Gozlan, H.5    Hamon, M.6
  • 8
    • 0027340365 scopus 로고
    • 2 receptors in adult rat brain after neonatal destruction of nigrostriatal dopamine neurons: A quantitative autoradiographic study
    • 2 receptors in adult rat brain after neonatal destruction of nigrostriatal dopamine neurons: a quantitative autoradiographic study. Brain Res. 606:273-285.
    • (1993) Brain Res. , vol.606 , pp. 273-285
    • Radja, F.1    Descarries, L.2    Dewar, K.M.3    Reader, T.A.4
  • 11
    • 0027333308 scopus 로고
    • 1A receptor antagonists: Utility as research tools and therapeutic agents
    • 1A receptor antagonists: utility as research tools and therapeutic agents. TIPS 14:441-448.
    • (1993) TIPS , vol.14 , pp. 441-448
    • Fletcher, A.1    Cliffe, I.A.2    Dourish, C.T.3
  • 13
    • 0027048880 scopus 로고
    • 1A receptors negatively coupled to adenylyl cyclase activity in rat hippocampal membranes
    • 1A receptors negatively coupled to adenylyl cyclase activity in rat hippocampal membranes. Molec. Pharmacol. 41:1066-1072.
    • (1992) Molec. Pharmacol. , vol.41 , pp. 1066-1072
    • Yocca, F.D.1    Iben, L.2    Meller, E.3
  • 15
    • 0025267308 scopus 로고
    • Cellular localization of serotonin 1A, 1B and uptake sites in cingulate cortex of the rat
    • Crin, P. B., Vogt, B. A., Volicer, L., and Wiley, R. G. 1990. Cellular localization of serotonin 1A, 1B and uptake sites in cingulate cortex of the rat. J. Pharmacol. Exp. Ther. 252:651-656.
    • (1990) J. Pharmacol. Exp. Ther. , vol.252 , pp. 651-656
    • Crin, P.B.1    Vogt, B.A.2    Volicer, L.3    Wiley, R.G.4
  • 16
    • 0023837915 scopus 로고
    • Pharmacology of 5-hydroxytryptamine-1A receptors which inhibit cAMP production in hippocampal and cortical neurons in primary culture
    • Dumuis, A., Sebben, M., and Bockaert, J. 1988. Pharmacology of 5-hydroxytryptamine-1A receptors which inhibit cAMP production in hippocampal and cortical neurons in primary culture. Mol. Pharmacol. 33:178-186.
    • (1988) Mol. Pharmacol. , vol.33 , pp. 178-186
    • Dumuis, A.1    Sebben, M.2    Bockaert, J.3
  • 18
    • 0022556726 scopus 로고
    • 3H]8-OH-DPAT labels the serotonin transporter in the rat striatum
    • 3H]8-OH-DPAT labels the serotonin transporter in the rat striatum. Eur. J. Pharmacol. 124:371-373.
    • (1986) Eur. J. Pharmacol. , vol.124 , pp. 371-373
    • Schoemaker, H.1    Langer, S.Z.2
  • 20
    • 0004183979 scopus 로고
    • The chemical properties of SH groups; Sulfhydryl reagents
    • Pergamon Press, Metzler D., ed., Oxford, New York, Toronto
    • Torchinsky, Y. M. 1981. The chemical properties of SH groups; Sulfhydryl reagents. In: Sulfur in proteins. Pergamon Press, Metzler D., ed., Oxford, New York, Toronto, pp 3-7.
    • (1981) Sulfur in Proteins , pp. 3-7
    • Torchinsky, Y.M.1
  • 21
    • 33947482089 scopus 로고
    • Dithiothreitol, a new protective reagent for SH groups
    • Cleland, W. W. 1964. Dithiothreitol, a new protective reagent for SH groups. Biochemistry 3:480-482.
    • (1964) Biochemistry , vol.3 , pp. 480-482
    • Cleland, W.W.1
  • 22
  • 23
    • 0025275353 scopus 로고
    • Pretreatment with N-ethoxycarbony-1-2-ethoxy-1,2-dihydroquinoline accelerates the electroshock-induced decrease in the density of β-adrenoceptors but not functional downregulation
    • Pile, A., and Vetulani, J. 1990. Pretreatment with N-ethoxycarbony-1-2-ethoxy-1,2-dihydroquinoline accelerates the electroshock-induced decrease in the density of β-adrenoceptors but not functional downregulation. Neuropharmacology 29:469-473.
    • (1990) Neuropharmacology , vol.29 , pp. 469-473
    • Pile, A.1    Vetulani, J.2
  • 25
    • 0015049463 scopus 로고
    • Pharmacological estimation of drug-receptor dissociation constants. Statistical evaluation. I. Agonists
    • Parker, R. B., and Waud, D. R. 1971. Pharmacological estimation of drug-receptor dissociation constants. Statistical evaluation. I. Agonists. J. Pharmacol. Exp. Ther. 177:1-12.
    • (1971) J. Pharmacol. Exp. Ther. , vol.177 , pp. 1-12
    • Parker, R.B.1    Waud, D.R.2
  • 27
    • 0018001339 scopus 로고
    • Simultaneous analysis of families of sigmoidal curves: Application to bioassay, radioligand assay, and physiologicaldose-response curve
    • De Léan, A., Munson, P. J., and Rodbard, D. 1978. Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiologicaldose-response curve. Am. J. Physiol. 235:E97-E102.
    • (1978) Am. J. Physiol. , vol.235
    • De Léan, A.1    Munson, P.J.2    Rodbard, D.3
  • 28
    • 0019061918 scopus 로고
    • LIGAND: A versatile computerized approach for the characterization of ligand binding systems
    • Munson, P. J., and Rodbard, D. 1980. LIGAND: A versatile computerized approach for the characterization of ligand binding systems. Anal. Biochem. 107:220-239.
    • (1980) Anal. Biochem. , vol.107 , pp. 220-239
    • Munson, P.J.1    Rodbard, D.2
  • 29
    • 0022005744 scopus 로고
    • Analysis of radioligand binding experiments: A collection of computer programs for the IBM PC
    • McPherson, G. A. 1985. Analysis of radioligand binding experiments: A collection of computer programs for the IBM PC. J. Pharmacol. Meth. 14:213-228.
    • (1985) J. Pharmacol. Meth. , vol.14 , pp. 213-228
    • McPherson, G.A.1
  • 30
    • 0027398771 scopus 로고
    • 1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HELA cells
    • 1993
    • 1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HELA cells. Biochem. Pharmacol. 45:375-383, 1993.
    • (1993) Biochem. Pharmacol. , vol.45 , pp. 375-383
    • Pauwels, P.J.1    Van Gompel, P.2    Leysen, J.E.3
  • 35
    • 0027007705 scopus 로고
    • Serotonin (5-HT2) receptor mediated enhancement of cortical unit activity
    • Newman, R. S., and Zebrowska, G. 1992. Serotonin (5-HT2) receptor mediated enhancement of cortical unit activity. Can. J. Physiol. Pharmacol. 70:1604-1609.
    • (1992) Can. J. Physiol. Pharmacol. , vol.70 , pp. 1604-1609
    • Newman, R.S.1    Zebrowska, G.2
  • 36
    • 0026559955 scopus 로고
    • Pharmacological and physico-chemical properties of pre- versus postsynaptic 5-HT1A receptor binding sites in the rat brain
    • Radja, F., Daval, G., Hamon, M., and Vergé, D. 1992. Pharmacological and physico-chemical properties of pre- versus postsynaptic 5-HT1A receptor binding sites in the rat brain. J. Neurochem. 52:1338-1346.
    • (1992) J. Neurochem. , vol.52 , pp. 1338-1346
    • Radja, F.1    Daval, G.2    Hamon, M.3    Vergé, D.4
  • 38
    • 0023637301 scopus 로고
    • 2-adrenoceptors from GTP-binding proteins by N-ethylmaleimide
    • 2-adrenoceptors from GTP-binding proteins by N-ethylmaleimide. J. Neurochem. 49:1894-1901.
    • (1987) J. Neurochem. , vol.49 , pp. 1894-1901
    • Kitamura, Y.1    Nomura, Y.2
  • 42
    • 0000836690 scopus 로고
    • Evidence for possible non-specific reactions between N-ethylmaleimide and proteins
    • Brewer, C. F., and Riehm, J. P. 1967. Evidence for possible non-specific reactions between N-ethylmaleimide and proteins. Anal. Biochem. 18:248-255.
    • (1967) Anal. Biochem. , vol.18 , pp. 248-255
    • Brewer, C.F.1    Riehm, J.P.2
  • 44
    • 84969001783 scopus 로고
    • The attractions of proteins for small molecules and ions
    • Scatchard, G. 1949. The attractions of proteins for small molecules and ions. Ann. N.Y. Acad. Sci. 51:660-672.
    • (1949) Ann. N.Y. Acad. Sci. , vol.51 , pp. 660-672
    • Scatchard, G.1
  • 45
    • 0014511179 scopus 로고
    • The mechanism of irreversible adrenergic blockade by N-carbethoxydihydroquinolines. Model studies with typical serine hydrolases
    • Belleau, B., DiTullio, V., and Godin, D. 1969. The mechanism of irreversible adrenergic blockade by N-carbethoxydihydroquinolines. Model studies with typical serine hydrolases. Biochem. Pharmacol. 18:1039-1044.
    • (1969) Biochem. Pharmacol. , vol.18 , pp. 1039-1044
    • Belleau, B.1    DiTullio, V.2    Godin, D.3
  • 47
    • 0027186438 scopus 로고
    • Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase
    • Plassat, J.-C, Amlaiky, N., and Hen, R. 1993. Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase. Molec. Pharmacol. 44:229-236.
    • (1993) Molec. Pharmacol. , vol.44 , pp. 229-236
    • Plassat, J.-C.1    Amlaiky, N.2    Hen, R.3
  • 48
    • 0028180634 scopus 로고
    • A receptor-activated current in cultured rat suprachiasmatic neurones
    • A receptor-activated current in cultured rat suprachiasmatic neurones. J. Physiol. 478:67-73.
    • (1994) J. Physiol. , vol.478 , pp. 67-73
    • Kawahara, F.1    Saito, H.2    Katsuki, H.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.