메뉴 건너뛰기




Volumn 67, Issue 25, 2000, Pages 3103-3112

Resveratrol, a red wine constituent, is a mechanism-based inactivator of cytochrome P450 3A4

Author keywords

Cytochrome P450 3A4; Mechanism based inhibition; Red wine; Resveratrol

Indexed keywords

CYP3A PROTEIN, HUMAN; CYP3A4 PROTEIN, HUMAN; CYTOCHROME P450; ENZYME INHIBITOR; MIXED FUNCTION OXIDASE; RESVERATROL; STILBENE DERIVATIVE;

EID: 0034634252     PISSN: 00243205     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0024-3205(00)00888-2     Document Type: Article
Times cited : (152)

References (29)
  • 1
    • 0030963473 scopus 로고    scopus 로고
    • Resveratrol: A molecule whose time has come? And gone?
    • Soleas GJ, Diamandis EP, Goldberg DM. Resveratrol: a molecule whose time has come? And gone? Clin. Biochem. 1997; 30(2): 91-113.
    • (1997) Clin. Biochem. , vol.30 , Issue.2 , pp. 91-113
    • Soleas, G.J.1    Diamandis, E.P.2    Goldberg, D.M.3
  • 2
    • 0034645693 scopus 로고    scopus 로고
    • Biological effects of resveratrol
    • Fremont L. Biological effects of resveratrol. Life Sci. 2000; 66 (8): 663-73.
    • (2000) Life Sci. , vol.66 , Issue.8 , pp. 663-673
    • Fremont, L.1
  • 4
    • 0031444281 scopus 로고    scopus 로고
    • Resveratrol, a polyphenolic compound found in grapes and wine, is an agonist for the estrogen receptor
    • Gehm BD, McAndrews JM, Chien PY, Jameson JL. Resveratrol, a polyphenolic compound found in grapes and wine, is an agonist for the estrogen receptor. Proc. Natl. Acad. Sci. USA 1997; 94 (25): 14138-43.
    • (1997) Proc. Natl. Acad. Sci. USA , vol.94 , Issue.25 , pp. 14138-14143
    • Gehm, B.D.1    McAndrews, J.M.2    Chien, P.Y.3    Jameson, J.L.4
  • 5
    • 0029065391 scopus 로고
    • The red wine phenolics trans-resveratrol and quercetin block human platelet aggregation and eicosanoid synthesis: Implications for protection against coronary heart disease
    • Pace-Asciak CR, Hahn S, Diamandis EP, Soleas G, Goldberg DM. The red wine phenolics trans-resveratrol and quercetin block human platelet aggregation and eicosanoid synthesis: implications for protection against coronary heart disease. Clin. Chim. Acta 1995; 235 (2): 207-19.
    • (1995) Clin. Chim. Acta , vol.235 , Issue.2 , pp. 207-219
    • Pace-Asciak, C.R.1    Hahn, S.2    Diamandis, E.P.3    Soleas, G.4    Goldberg, D.M.5
  • 6
    • 0029027416 scopus 로고
    • Beyond alcohol: Beverage consumption and cardiovascular mortality. Clin
    • Goldberg DM, Hahn SE, Parkes JG. Beyond alcohol: beverage consumption and cardiovascular mortality. Clin. Chim. Acta 1995; 237 (1-2): 155-87.
    • (1995) Chim. Acta , vol.237 , Issue.1-2 , pp. 155-187
    • Goldberg, D.M.1    Hahn, S.E.2    Parkes, J.G.3
  • 9
    • 0033584453 scopus 로고    scopus 로고
    • Resveratrol is a selective human cytochrome P450 1A1 inhibitor
    • Chun YJ, Kim MY, Guengerich FP. Resveratrol is a selective human cytochrome P450 1A1 inhibitor. Biochem. Biophys. Res. Commun. 1999; 262 (1): 20-4.
    • (1999) Biochem. Biophys. Res. Commun. , vol.262 , Issue.1 , pp. 20-24
    • Chun, Y.J.1    Kim, M.Y.2    Guengerich, F.P.3
  • 10
    • 0032535055 scopus 로고    scopus 로고
    • Resveratrol inhibits transcription of CYP1A1 in vitro by preventing activation of the aryl hydrocarbon receptor
    • Ciolino HP, Daschner PJ, Yeh GC. Resveratrol inhibits transcription of CYP1A1 in vitro by preventing activation of the aryl hydrocarbon receptor. Cancer Res. 1998; 58 (24): 5707-12.
    • (1998) Cancer Res. , vol.58 , Issue.24 , pp. 5707-5712
    • Ciolino, H.P.1    Daschner, P.J.2    Yeh, G.C.3
  • 11
    • 0032416143 scopus 로고    scopus 로고
    • Modulation by phytochemicals of cytochrome P450-linked enzyme activity
    • Teel RW, Huynh H. Modulation by phytochemicals of cytochrome P450-linked enzyme activity. Cancer Lett. 1998; 133(2): 135-41.
    • (1998) Cancer Lett. , vol.133 , Issue.2 , pp. 135-141
    • Teel, R.W.1    Huynh, H.2
  • 12
    • 0032861582 scopus 로고    scopus 로고
    • Resveratrol has antagonist activity on the aryl hydrocarbon receptor: Implications for prevention of dioxin toxicity
    • Casper RF, Quesne M, Rogers IM, Shirota T, Jolivet A, Milgrom E, Savouret JF. Resveratrol has antagonist activity on the aryl hydrocarbon receptor: implications for prevention of dioxin toxicity. Mol. Pharmacol. 1999; 56 (4): 784-90.
    • (1999) Mol. Pharmacol. , vol.56 , Issue.4 , pp. 784-790
    • Casper, R.F.1    Quesne, M.2    Rogers, I.M.3    Shirota, T.4    Jolivet, A.5    Milgrom, E.6    Savouret, J.F.7
  • 13
    • 0000023835 scopus 로고    scopus 로고
    • Mechanism-based inactivation of human cytochrome P450 3A4 by grapefruit juice and red wine
    • Chan WK, Nguyen LT, Miller VP, Harris RZ. Mechanism-based inactivation of human cytochrome P450 3A4 by grapefruit juice and red wine. Life Sci. 1998; 62 (10): L135-42.
    • (1998) Life Sci. , vol.62 , Issue.10
    • Chan, W.K.1    Nguyen, L.T.2    Miller, V.P.3    Harris, R.Z.4
  • 15
    • 0029741202 scopus 로고    scopus 로고
    • In vitro studies on the metabolic activation of the furanopyridine L-754,394, a highly potent and selective mechanism-based inhibitor of cytochrome P450 3A4
    • Sahali-Sahly Y, Balani SK, Lin JH, Baillie TA. In vitro studies on the metabolic activation of the furanopyridine L-754,394, a highly potent and selective mechanism-based inhibitor of cytochrome P450 3A4. Chem. Res. Toxicol. 1996; 9(6): 1007-12.
    • (1996) Chem. Res. Toxicol. , vol.9 , Issue.6 , pp. 1007-1012
    • Sahali-Sahly, Y.1    Balani, S.K.2    Lin, J.H.3    Baillie, T.A.4
  • 16
    • 0029012009 scopus 로고
    • CYP3A4 ex pressed by insect cells infected with a recombinant baculovirus containing both CYP3A4 and human NADPH-cytochrome P450 reductase is catalytically similar to human liver microsomal CYP3A4
    • Lee CA, Kadwell SH, Kost TA, Serabjit-Singh CJ. CYP3A4 ex pressed by insect cells infected with a recombinant baculovirus containing both CYP3A4 and human NADPH-cytochrome P450 reductase is catalytically similar to human liver microsomal CYP3A4. Arch. Biochem. Biophys. 1995; 319 (1): 157-67.
    • (1995) Arch. Biochem. Biophys. , vol.319 , Issue.1 , pp. 157-167
    • Lee, C.A.1    Kadwell, S.H.2    Kost, T.A.3    Serabjit-Singh, C.J.4
  • 17
    • 73649151319 scopus 로고
    • Esters of methanesulfonic acid as irreversible inhibitors of acetylcholinesterase
    • Kitz R, Wilson IB. Esters of methanesulfonic acid as irreversible inhibitors of acetylcholinesterase. J. Biol. Chem. 1962; 237: 3245-9.
    • (1962) J. Biol. Chem. , vol.237 , pp. 3245-3249
    • Kitz, R.1    Wilson, I.B.2
  • 19
    • 0020079949 scopus 로고
    • Formation of an inactive cytochrome P-450 Fe(II)-metabolite complex after administration of troleandomycin in humans
    • Pessayre D, Larrey D, Vitaux J, Breil P, Belghiti J, Benhamou JP. Formation of an inactive cytochrome P-450 Fe(II)-metabolite complex after administration of troleandomycin in humans. Biochem. Pharmacol. 1982; 31 (9): 1699-704.
    • (1982) Biochem. Pharmacol. , vol.31 , Issue.9 , pp. 1699-1704
    • Pessayre, D.1    Larrey, D.2    Vitaux, J.3    Breil, P.4    Belghiti, J.5    Benhamou, J.P.6
  • 20
    • 0026464616 scopus 로고
    • Identification of rifampin-inducible P450IIIA4 (CYP3A4) in human small bowel enterocytes
    • Kolars JC, Schmiedlin-Ren P, Schuetz JD, Fang C, Watkins PB. Identification of rifampin-inducible P450IIIA4 (CYP3A4) in human small bowel enterocytes. J. Clin. Invest. 1992; 90 (5): 1871-8.
    • (1992) J. Clin. Invest. , vol.90 , Issue.5 , pp. 1871-1878
    • Kolars, J.C.1    Schmiedlin-Ren, P.2    Schuetz, J.D.3    Fang, C.4    Watkins, P.B.5
  • 22
    • 0033584453 scopus 로고    scopus 로고
    • Resveratrol is a selective human cytochrome P450 1A1 inhibitor
    • Chun YJ, Kim MY, Guengerich FP. Resveratrol is a selective human cytochrome P450 1A1 inhibitor. Biochem. Biophys. Res. Commun. 1999; 262 (1): 20-24.
    • (1999) Biochem. Biophys. Res. Commun. , vol.262 , Issue.1 , pp. 20-24
    • Chun, Y.J.1    Kim, M.Y.2    Guengerich, F.P.3
  • 24
    • 0033564235 scopus 로고    scopus 로고
    • Sigmoidal kinetic mode for two co-operative substrate-binding sites in a cytochrome P450 3A4 active site: An example of the metabolism of diazepam and its derivatives
    • Shou M, Mei Q, Ettore MW, Jr., Dai R, Baillie TA, Rushmore TH. Sigmoidal kinetic mode for two co-operative substrate-binding sites in a cytochrome P450 3A4 active site: an example of the metabolism of diazepam and its derivatives. Biochem. J. 1999; 340 (Pt 3): 845-53.
    • (1999) Biochem. J. , vol.340 , Issue.3 PART , pp. 845-853
    • Shou, M.1    Mei, Q.2    Ettore Jr., M.W.3    Dai, R.4    Baillie, T.A.5    Rushmore, T.H.6
  • 25
    • 0000574406 scopus 로고    scopus 로고
    • Evaluation of atypical cytochrome P450 kinetics with two-substrate models: Evidence that multiple substrates can simultaneously bind to cytochrome P450 active sites
    • Korzekwa KR, Krishnamachary N, Shou M, Ogai A, Parise RA, Rettie AE, Gonzalez FJ, Tracy TS. Evaluation of atypical cytochrome P450 kinetics with two-substrate models: evidence that multiple substrates can simultaneously bind to cytochrome P450 active sites. Biochemistry 1998; 37 (12): 4137-47.
    • (1998) Biochemistry , vol.37 , Issue.12 , pp. 4137-4147
    • Korzekwa, K.R.1    Krishnamachary, N.2    Shou, M.3    Ogai, A.4    Parise, R.A.5    Rettie, A.E.6    Gonzalez, F.J.7    Tracy, T.S.8
  • 26
    • 0031670167 scopus 로고    scopus 로고
    • Erythromycin and verapamil considerably increase serum simvastatin and simvastatin acid concentrations
    • Kantola T, Kivisto KT, Neuvonen PJ. Erythromycin and verapamil considerably increase serum simvastatin and simvastatin acid concentrations [see comments]. Clin. Pharmacol. Ther. 1998; 64 (2): 177-82.
    • (1998) Clin. Pharmacol. Ther. , vol.64 , Issue.2 , pp. 177-182
    • Kantola, T.1    Kivisto, K.T.2    Neuvonen, P.J.3
  • 27
    • 0029782647 scopus 로고    scopus 로고
    • Erythromycin-felodipine interaction: Magnitude, mechanism, and comparison with grapefruit juice
    • Bailey DG, Bend JR, Arnold JM, Tran LT, Spence JD. Erythromycin-felodipine interaction: magnitude, mechanism, and comparison with grapefruit juice. Clin. Pharmacol. Ther. 1996; 60 (1): 25-33.
    • (1996) Clin. Pharmacol. Ther. , vol.60 , Issue.1 , pp. 25-33
    • Bailey, D.G.1    Bend, J.R.2    Arnold, J.M.3    Tran, L.T.4    Spence, J.D.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.