Methaqualone derivatives are potent noncompetitive AMPA receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 11, 2000, Pages 1203-1205

  Chenard, B L ^a   Menniti, F S ^a   Pagnozzi, M J ^a   Shenk, K D ^a   Ewing, F E ^a   Welch, W M ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMPA RECEPTOR; METHAQUALONE; METHAQUALONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL MODIFICATION; DRUG ACTIVITY; DRUG POTENCY; DRUG STRUCTURE; NONHUMAN; PARTIAL DRUG SYNTHESIS; RAT; RECEPTOR BLOCKING; STRUCTURE ACTIVITY RELATION;

ANIMALS; CELLS, CULTURED; CEREBELLUM; CYTOPLASMIC GRANULES; EXCITATORY AMINO ACID ANTAGONISTS; METHAQUALONE; RATS; RECEPTORS, AMPA;

EID: 0034608633     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(00)00216-X     Document Type: Article

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