Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 17, 2000, Pages 1953-1957

  Baraldi, Pier Giovanni ^a   Zaid, Abdel Naser ^a   Lampronti, Ilaria ^a   Fruttarolo, Francesca ^a   Pavani, Maria Giovanna ^a   Tabrizi, Mojgan Aghazadhe ^a   Shryock, John C ^b   Leung, Edward ^c   Romagnoli, Romeo ^a  

^a UNIVERSITY OF FERRARA   (Italy)

^b UNIVERSITY OF FLORIDA COLLEGE OF MEDICINE   (United States)

^c Medco Research Inc   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE A1 RECEPTOR; ADENOSINE A1 RECEPTOR AGONIST; ADENOSINE A1 RECEPTOR ANTAGONIST; THIOPHENE DERIVATIVE;

ANIMAL CELL; ARTICLE; CHO CELL; DRUG ACTIVITY; DRUG EFFECT; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ALLOSTERIC REGULATION; ANIMALS; CHO CELLS; CRICETINAE; CYCLIC AMP; HUMANS; RECEPTORS, PURINERGIC P1; STRUCTURE-ACTIVITY RELATIONSHIP; THIOPHENES;

ANIMALIA; STAPHYLOCOCCUS PHAGE 3A;

EID: 0034605224     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(00)00379-6     Document Type: Article

References (11)