SCOPUS 정보 검색 플랫폼

Volumn 60, Issue 23, 2000, Pages 6577-6580

Activity of a novel camptothecin analogue, homocamptothecin, in camptothecin-resistant cell lines with topoisomerase I alterations

(3) Urasaki, Y a Takebayashi, Y a Pommier, Y a

a NATIONAL CANCER INSTITUTE (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CAMPTOTHECIN; CAMPTOTHECIN DERIVATIVE; CARBENE; DNA; DNA TOPOISOMERASE; ENZYME; HOMOCAMPTOTHECIN; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING SITE; DRUG ACTIVITY; DRUG RESISTANCE; DRUG SENSITIVITY; HAMSTER; HUMAN; HUMAN CELL; MOUSE; NONHUMAN; POINT MUTATION; PRIORITY JOURNAL;

ANIMALS; ANTINEOPLASTIC AGENTS; CAMPTOTHECIN; CRICETINAE; DNA TOPOISOMERASES, TYPE I; DNA, NEOPLASM; DRUG RESISTANCE, NEOPLASM; DRUG SCREENING ASSAYS, ANTITUMOR; ENZYME INHIBITORS; ENZYME STABILITY; HUMANS; INHIBITORY CONCENTRATION 50; LEUKEMIA P388; MALE; MICE; POINT MUTATION; PROSTATIC NEOPLASMS; TUMOR CELLS, CULTURED;

EID: 0034548379 PISSN: 00085472 EISSN: None Source Type: Journal
DOI: None Document Type: Article

Times cited : (39)

References (18)

1
- 0033208192
- Topoisomerase 1 inhibitors: Selectivity and cellular resistance
- (1999) Drug Resistance Update , vol.2 , pp. 307-318
- Pommier, Y.¹ Pourquier, P.² Urasaki, Y.³ Wu, J.⁴ Laco, G.S.⁵

2
- 0032585548
- Homocamptothecins: Synthesis and antitumor activity of novel E-ring-modified camptothecin analogues
- (1998) J. Med. Chem. , vol.41 , pp. 5410-5419
- Lavergne, O.¹ Lesueur-Ginot, L.² Pla Rodas, F.³ Kasprzyk, P.G.⁴ Pommier, J.⁵ Demarquay, D.⁶ Prevost, G.⁷ Ulibarri, G.⁸ Rolland, A.⁹ Schiano-Liberatore, A.M.¹⁰ Harnett, J.¹¹ Pons, D.¹² Camara, J.¹³ Bigg, D.C.H.¹⁴

3
- 0033564494
- Homocamptothecin, an E-ring modified camptothecin with enhanced lactone stability, retains topoisomerase I-targeted activity and antitumor properties
- (1999) Cancer Res. , vol.59 , pp. 2939-2943
- Lesueur-Ginot, L.¹ Demarquay, D.² Kiss, R.³ Kasprzyk, P.G.⁴ Dassonneville, L.⁵ Bailly, C.⁶ Camara, J.⁷ Lavergne, O.⁸ Bigg, D.C.⁹

4
- 0033549870
- Novel A, B, E-ring-modified camptothecins displaying high lipophilicity and markedly improved human blood stabilities
- (1999) J. Med. Chem. , vol.42 , pp. 3018-3022
- Bom, D.¹ Curran, D.P.² Chavan, A.J.³ Kruszewski, S.⁴ Zimmer, S.G.⁵ Fraley, K.A.⁶ Burke, T.G.⁷

5
- 0034049602
- Homocamptothecin, an E-ring-modified camptothecin, exerts more potent antiproliferative activity than other topoisomerase I inhibitors in human colon cancers obtained from surgery and maintained in vitro under histotypical culture conditions
- (2000) Clin. Cancer Res. , vol.6 , pp. 1557-1562
- Philippart, P.¹ Harper, L.² Chaboteaux, C.³ Decaestecker, C.⁴ Bronckart, Y.⁵ Gordover, L.⁶ Lesueur-Ginot, L.⁷ Malonne, H.⁸ Lavergne, O.⁹ Bigg, D.C.¹⁰ Da Costa, P.M.¹¹ Kiss, R.¹²

6
- 0028957974
- Mutation at the catalytic site of topoisomerase I in CEM/C2, a human leukemia cell line resistant to camptothecin
- (1995) Cancer Res. , vol.55 , pp. 1339-1346
- Fujimori, A.¹ Harker, W.G.² Kohlhagen, G.³ Hoki, Y.⁴ Pommier, Y.⁵

7
- 0029825344
- Silencing and selective methylation of the normal topoisomerase I gene in camptothecin-resistant CEM/C2 human leukemia cells
- (1996) Oncol. Res. , vol.8 , pp. 295-301
- Fujimori, A.¹ Hoki, Y.² Popescu, N.C.³ Pommier, Y.⁴

8
- 0026328062
- Synergic cell killing by ionizing radiation and topoisomerase I inhibitor topotecan (SK and F 10864)
- (1991) Cancer Res. , vol.51 , pp. 5813-5816
- Mattern, M.R.¹ Hofmann, G.A.² McCabe, F.L.³ Johnson, R.K.⁴

9
- 0027813132
- In vitro and in vivo effects of clinically important camptothecin analogues on multidrug-resistant cells
- (1993) Oncol. Res. , vol.5 , pp. 467-474
- Mattern, M.R.¹ Hofmaan, G.A.² Polsky, R.M.³ Funk, L.R.⁴ McCabe, F.L.⁵ Johnson, R.K.⁶

10
- 0027368901
- Cloning of Chinese hamster DNA topoisomerase I cDNA and identification of a single point mutation responsible for camptothecin resistance
- (1993) J. Biol. Chem. , vol.268 , pp. 25463-25468
- Tanizawa, A.¹ Bertrand, R.² Kohlhagen, G.³ Tabuchi, A.⁴ Jenkins, J.⁵ Pommier, Y.⁶

11
- 0028485758
- Overexpression of human DNA topoisomerase I in insect cells using a baculovirus vector
- (1994) Protein Expr. Purif. , vol.5 , pp. 364-370
- Zhelkovsky, A.M.¹ Moore, C.L.² Rattner, J.B.³ Hendzel, M.J.⁴ Furbee, C.S.⁵ Muller, M.T.⁶ Bazett-Jones, D.P.⁷

12
- 0033047992
- Synthesis of cytotoxic indenoisoquinoline topoisomerase I poisons
- (1999) J. Med. Chem. , vol.42 , pp. 446-457
- Strumberg, D.¹ Pommier, Y.² Paull, K.³ Jayaraman, M.⁴ Nagafuji, P.⁵ Cushman, M.⁶

13
- 0034652117
- Induction of topoisomerase I cleavage complexes by 1-β-D- arabinofuranosylcytosine (ara-C) in vitro and in ara-C-treated cells
- (2000) Proc. Natl. Acad. Sci. USA , vol.97 , pp. 1885-1890
- Poarquier, P.¹ Takebayashi, Y.² Urasaki, Y.³ Gioffre, C.⁴ Kohlhagen, G.⁵ Pommier, Y.⁶

14
- 0033598698
- Homocamptothecin, an E-ring-modified camptothecin analogue, generates new topoisomerase I-mediated DNA breaks
- (1999) Biochemistry , vol.38 , pp. 15556-15563
- Bailly, C.¹ Lansiaux, A.² Dassonneville, L.³ Demarquay, D.⁴ Coulomb, H.⁵ Huchet, M.⁶ Lavergne, O.⁷ Bigg, D.C.⁸

15
- 0028012774
- The structural basis of camptothecin interactions with human serum albumin: Impact on drug stability
- (1994) J. Med. Chem. , vol.37 , pp. 40-46
- Burke, T.G.¹ Mi, Z.M.²

16
- 0032489634
- Crystal structures of human topoisomerase I in covalent and noncovalent complexes with DNA
- (1998) Science (Washington DC) , vol.279 , pp. 1504-1513
- Redinbo, M.R.¹ Stewart, L.² Kuhn, P.³ Champoux, J.J.⁴ Hol, W.G.⁵

17
- 0025719903
- Effect of local DNA sequence on topoisomerase I cleavage in the presence or absence of camptothecin
- (1991) J. Biol. Chem. , vol.266 , pp. 20418-20423
- Jaxel, C.¹ Capranico, G.² Kerrigan, D.³ Kohn, K.W.⁴ Pommier, Y.⁵

18
- 0032543518
- Molecular modeling studies of the DNA-topoisomerase I ternary cleavable complex with camptothecin
- (1998) J. Med. Chem. , vol.41 , pp. 2216-2226
- Fan, Y.¹ Weinstein, J.N.² Kohn, K.W.³ Shi, L.M.⁴ Pommier, Y.⁵

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