메뉴 건너뛰기




Volumn 17, Issue 4, 2000, Pages 410-418

Allometric pharmacokinetic scaling: Towards the prediction of human oral pharmacokinetics

Author keywords

Allometric scaling; Interspecies scaling; Pharmacokinetics

Indexed keywords

AMPHOTERICIN B; CAFFEINE; CEFAZOLIN; CEFODIZIME; CEFOPERAZONE; CEFOTETAN; CEFPIRAMIDE; CEFTIZOXIME; CIPROFLOXACIN; DIAZEPAM; ENPROFYLLINE; LATAMOXEF; MIBEFRADIL; MIDAZOLAM; MOFAROTENE; PHENAZONE; PROPRANOLOL; REMOXIPRIDE; SEMATILIDE; TAMSULOSIN; THEOPHYLLINE; VALPROIC ACID;

EID: 0034120946     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1007520818956     Document Type: Article
Times cited : (68)

References (30)
  • 1
    • 0018967595 scopus 로고
    • Interspecies variation in liver weight, hepatic blood flow, and antipyrine intrinsic clearance: Extrapolation of data to benzodiazepines and phenytoin
    • 1. H. Boxenbaum. Interspecies variation in liver weight, hepatic blood flow, and antipyrine intrinsic clearance: extrapolation of data to benzodiazepines and phenytoin. J. Pharmcokin. Biopharm. 2, 165-176 (1980).
    • (1980) J. Pharmcokin. Biopharm. , vol.2 , pp. 165-176
    • Boxenbaum, H.1
  • 2
    • 0021703938 scopus 로고
    • Interspecies pharmacokinetic scaling and the evolutionary-comparative paradigm
    • 2. H. Boxenbaum. Interspecies pharmacokinetic scaling and the evolutionary-comparative paradigm. Drug Metab. Rev. 15:1071-1121 (1984).
    • (1984) Drug Metab. Rev. , vol.15 , pp. 1071-1121
    • Boxenbaum, H.1
  • 3
    • 0022975813 scopus 로고
    • Time concepts in physics, biology, and pharmacokinetics
    • 3. H. Boxenbaum, Time concepts in physics, biology, and pharmacokinetics. J. Pharm. Sci. 75:1053-1062 (1986).
    • (1986) J. Pharm. Sci. , vol.75 , pp. 1053-1062
    • Boxenbaum, H.1
  • 4
    • 0028792083 scopus 로고
    • First-time-in-human dose selection: Allometric thoughts and perspectives
    • 4. H. Boxenbaum and C. Dilea. First-time-in-human dose selection: allometric thoughts and perspectives. J. Clin. Pharmacol. 35: 957-966 (1995).
    • (1995) J. Clin. Pharmacol. , vol.35 , pp. 957-966
    • Boxenbaum, H.1    Dilea, C.2
  • 5
    • 0031725042 scopus 로고    scopus 로고
    • Disposition of the antipsychotic CI-1007 in rat, monkey, dog, and human CYP2D6 extensive metabolizers: Species comparison and allometric scaling
    • 5. M. Rose Feng, J. Loo, and J. Wright. Disposition of the antipsychotic CI-1007 in rat, monkey, dog, and human CYP2D6 extensive metabolizers: species comparison and allometric scaling. Drug Metab. Dispos. 10:982-988 (1998).
    • (1998) Drug Metab. Dispos. , vol.10 , pp. 982-988
    • Feng, M.R.1    Loo, J.2    Wright, J.3
  • 7
    • 0031719267 scopus 로고    scopus 로고
    • Elucidation of human amphotericin b pharmacokinetics: Identification of a new potential factor affecting interspecies pharmacokinetic scaling
    • 7. G. Robbie and W. L. Chiou. Elucidation of human amphotericin B pharmacokinetics: identification of a new potential factor affecting interspecies pharmacokinetic scaling. Pharm. Res. 10: 1630-1636 (1998).
    • (1998) Pharm. Res. , vol.10 , pp. 1630-1636
    • Robbie, G.1    Chiou, W.L.2
  • 8
    • 0029828960 scopus 로고    scopus 로고
    • Interspecies scaling: Predicting clearance of drugs in humans. Three different approaches
    • 8. I. Mahmood, and J. Balian. Interspecies scaling: predicting clearance of drugs in humans. Three different approaches. Xenobiotica 26:887-895 (1996)
    • (1996) Xenobiotica , vol.26 , pp. 887-895
    • Mahmood, I.1    Balian, J.2
  • 9
    • 0030448841 scopus 로고    scopus 로고
    • Interspecies scaling: Predicting clearance of anticancer drugs in humans
    • 9. I. Mahmood. Interspecies scaling: predicting clearance of anticancer drugs in humans. Eur. J. Drug Metab. Pharmacokin. 3: 275-278 (1996).
    • (1996) Eur. J. Drug Metab. Pharmacokin. , vol.3 , pp. 275-278
    • Mahmood, I.1
  • 10
    • 0031719267 scopus 로고    scopus 로고
    • Elucidation of human amphotericin B pharmacokinetics: Identification of a new potential factor affecting interspecies pharmacokinetic scaling
    • 10. G. Robbie and W. L. Chiou. Elucidation of human amphotericin B pharmacokinetics: Identification of a new potential factor affecting interspecies pharmacokinetic scaling. Pharm. Res. 10: 1630-1636 (1998).
    • (1998) Pharm. Res. , vol.10 , pp. 1630-1636
    • Robbie, G.1    Chiou, W.L.2
  • 11
    • 0031723045 scopus 로고    scopus 로고
    • Correlation of plasma clearance of 54 extensively metabolized drugs between human and rats: Mean allometric coefficient of 0.66
    • 11. W. L. Chiou, G. Robbie, S. Chung, T. Wu, and C. Ma. Correlation of plasma clearance of 54 extensively metabolized drugs between human and rats: mean allometric coefficient of 0.66. Pharm. Res. 9:1474-1479 (1998).
    • (1998) Pharm. Res. , vol.9 , pp. 1474-1479
    • Chiou, W.L.1    Robbie, G.2    Chung, S.3    Wu, T.4    Ma, C.5
  • 13
    • 0031949326 scopus 로고    scopus 로고
    • Animal pharmacokinetics and interspecies scaling of Ro 25-6833 and related (Lactamylvinyl)cephalosporins
    • 13. W. G. Richter, P. Heizmann, J. Meyer, V. Starke, and T. Lave. Animal Pharmacokinetics and interspecies scaling of Ro 25-6833 and related (Lactamylvinyl)cephalosporins. J. Pharm. Sci. 4: 496-500 (1998).
    • (1998) J. Pharm. Sci. , vol.4 , pp. 496-500
    • Richter, W.G.1    Heizmann, P.2    Meyer, J.3    Starke, V.4    Lave, T.5
  • 14
    • 0025036920 scopus 로고
    • Prediction of the pharmacokinetics of cefodizime and cefotetan in humans from pharmacokinetic parameters in animals
    • 14. H. Mataushita, H. Suzuki, Y. Sugiyama, etc. Prediction of the pharmacokinetics of cefodizime and cefotetan in humans from pharmacokinetic parameters in animals. J. Pharmacobio-Dyn. 13:602-611 (1990).
    • (1990) J. Pharmacobio-Dyn. , vol.13 , pp. 602-611
    • Mataushita, H.1    Suzuki, H.2    Sugiyama, Y.3
  • 15
    • 0021972617 scopus 로고
    • Pharmacokinetic scale-up: Accurate prediction of human pharmacokinetic profiles from animal data
    • 15. J. Mordenti. Pharmacokinetic scale-up: accurate prediction of human pharmacokinetic profiles from animal data. J. Pharm. Sci. 10:1097-1099 (1985).
    • (1985) J. Pharm. Sci. , vol.10 , pp. 1097-1099
    • Mordenti, J.1
  • 16
    • 0031045628 scopus 로고    scopus 로고
    • Comparative pharmacokinetics and interspecies scaling of amphotericin B in several mammalian species
    • 16. A. Hutchaleelaha, H. Chow, and M. Mayerson. Comparative pharmacokinetics and interspecies scaling of amphotericin B in several mammalian species. J. Pharm. Pharrmacol. 49:178-183 (1997).
    • (1997) J. Pharm. Pharrmacol. , vol.49 , pp. 178-183
    • Hutchaleelaha, A.1    Chow, H.2    Mayerson, M.3
  • 17
    • 0030918716 scopus 로고    scopus 로고
    • Integration of in vitro data into allometric scaling to predict hepatic metabolic clearance in man: Application to 10 extensively metabolized drugs
    • 17. T. Lave, S. Duoin, C. Schmitt, R. C. Chou, D. Jaeck, and P. Coassolo. Integration of in vitro data into allometric scaling to predict hepatic metabolic clearance in man: application to 10 extensively metabolized drugs. J. Pharm. Sci. 5:584-585 (1997).
    • (1997) J. Pharm. Sci. , vol.5 , pp. 584-585
    • Lave, T.1    Duoin, S.2    Schmitt, C.3    Chou, R.C.4    Jaeck, D.5    Coassolo, P.6
  • 18
    • 0026625624 scopus 로고
    • Y. Tsunekawa, t. Hasegawa, m. Nadai, k. Takagi, and t. Nabeshima. Interspecies differences and scaling for the pharmacokinetics of xanthine derivatives
    • 18. Y. Tsunekawa, T. Hasegawa, M. Nadai, K. Takagi, and T. Nabeshima. Interspecies differences and scaling for the pharmacokinetics of xanthine derivatives. J. Pharm. Pharmacol. 44:594-599 (1992).
    • (1992) J. Pharm. Pharmacol. , vol.44 , pp. 594-599
  • 22
    • 0024043031 scopus 로고
    • Pharmacokinetics, renal clearance and metabolism of ciprofloxacin following intravenous and oral administration to calves and pigs
    • 22. J. Nouws, D. Mevius, T. Vree, A. Baars, and J. Larenses. Pharmacokinetics, renal clearance and metabolism of ciprofloxacin following intravenous and oral administration to calves and pigs. Vet. Quart. 3:156-163 (1988).
    • (1988) Vet. Quart. , vol.3 , pp. 156-163
    • Nouws, J.1    Mevius, D.2    Vree, T.3    Baars, A.4    Larenses, J.5
  • 25
    • 0032921527 scopus 로고    scopus 로고
    • Prediction of hepatic metabolic clearance based on interspecies allometric scaling techniques and in vitro - In vivo correlation
    • 25. T. Lave, S. P. Coassolo, and B. Reigner. Prediction of hepatic metabolic clearance based on interspecies allometric scaling techniques and in vitro - in vivo correlation Clin. Pharmacokin. 3:211-231 (1999).
    • (1999) Clin. Pharmacokin. , vol.3 , pp. 211-231
    • Lave, T.1    Coassolo, S.P.2    Reigner, B.3
  • 26
    • 18844481587 scopus 로고    scopus 로고
    • Pharmacokinetics of Susalimod, a highly biliary-excreted sulphasalazine analogue, in various species. Nonpredictable human clearance by allometric scaling
    • 26. Pahlman, M. Edholm, S. Kankaanranta and M.-L. Odell. Pharmacokinetics of Susalimod, a highly biliary-excreted sulphasalazine analogue, in various species. Nonpredictable human clearance by allometric scaling. Pharm. Pharmacol. Commun. 4:493-498 (1998).
    • (1998) Pharm. Pharmacol. Commun. , vol.4 , pp. 493-498
    • Pahlman, P.1    Edholm, M.2    Kankaanranta, S.3    Odell, M.-L.4
  • 27
    • 0028818229 scopus 로고
    • Species similarities and differences in pharmacokinetics
    • 27. J. H. Lin. Species similarities and differences in pharmacokinetics. Drug Metab. Dispos. 10:1008-1020 (1995).
    • (1995) Drug Metab. Dispos. , vol.10 , pp. 1008-1020
    • Lin, J.H.1
  • 28
    • 0031786518 scopus 로고    scopus 로고
    • Linear correlation of the fraction of oral dose absorbed of 64 drugs between human and rats
    • 28. W. L. Chiou and A. Barve. Linear correlation of the fraction of oral dose absorbed of 64 drugs between human and rats. Pharm. Res. 11:1792-1795 (1998).
    • (1998) Pharm. Res. , vol.11 , pp. 1792-1795
    • Chiou, W.L.1    Barve, A.2
  • 29
    • 0030990079 scopus 로고    scopus 로고
    • In vitro permeability across Caco-2 cells (colonic) can predict in vivo (small intestinal) absorption in man - Fact or myth
    • 29. S. Yee. In vitro permeability across Caco-2 cells (colonic) can predict in vivo (small intestinal) absorption in man - fact or myth. Pharm. Res. 14:763-766 (1997).
    • (1997) Pharm. Res. , vol.14 , pp. 763-766
    • Yee, S.1
  • 30
    • 0032733974 scopus 로고    scopus 로고
    • Prediction of human clearance of twenty-nine drugs from hepatic micosomal intrinsic clearance data: An examination of in vitro half-life approach and nonspecific binding to microsomes
    • 30. R. S. Obach. Prediction of human clearance of twenty-nine drugs from hepatic micosomal intrinsic clearance data: an examination of in vitro half-life approach and nonspecific binding to microsomes. Drug Metab. Dispos. 11:1350-1359 (1999).
    • (1999) Drug Metab. Dispos. , vol.11 , pp. 1350-1359
    • Obach, R.S.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.