Comparative molecular field analysis of colchicine inhibition and tubulin polymerization for combretastatins binding to the colchicine binding site on β-tubulin

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 6, 2000, Pages 1433-1441

  Brown, Milton L ^a   Rieger, Jayson M ^a   Macdonald, Timothy L ^a  

^a UNIVERSITY OF VIRGINIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BETA TUBULIN; COLCHICINE; COMBRETASTATIN; COMBRETASTATIN A4;

ARTICLE; BINDING SITE; CONFORMATION; MICROTUBULE ASSEMBLY; MOLECULAR MODEL; PHYSICAL CHEMISTRY; REGRESSION ANALYSIS; STRUCTURE ACTIVITY RELATION;

BIBENZYLS; BINDING SITES; BIOPOLYMERS; COLCHICINE; MOLECULAR CONFORMATION; STILBENES; TUBULIN;

EID: 0034097923     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00068-7     Document Type: Article

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