P-glycoprotein- and mrp2-mediated octreotide transport in renal proximal tubule

British Journal of Pharmacology

Volumn 129, Issue 2, 2000, Pages 251-256

  Gutmann, Heike ^a,b   Miller, David S ^a,c   Droulle, Agathe ^a,d   Drewe, Jürgen ^b   Fahr, Alfred ^a,e   Fricker, Gert ^a,f,g  

^a MOUNT DESERT ISLAND BIOLOGICAL LABORATORY   (United States)

^b UNIVERSITY HOSPITAL BASEL   (Switzerland)

^c NATIONAL INSTITUTE OF ENVIRONMENTAL HEALTH SCIENCES   (United States)

^d Lycee Roosevelt   (France)

^e PHILIPPS UNIVERSITY MARBURG   (Germany)

^f UNIVERSITY OF HEIDELBERG   (Germany)

^g Inst for Pharmaceut/Biopharmacy   (Germany)

Author keywords

Active transport; Confocal microscopy; Kidney; Killifish; Multidrug resistance associated protein2 (mrp2); Multidrug resistance protein; Octreotide; P glycoprotein (Pgp); Renal secretion

Indexed keywords

CYCLOSPORIN A DERIVATIVE; FLUORESCEIN; GLYCOPROTEIN P; LEUKOTRIENE C4; METHOTREXATE; MULTIDRUG RESISTANCE PROTEIN; OCTREOTIDE; SODIUM CYANIDE; VALSPODAR; VERAPAMIL;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BRUSH BORDER; CELL METABOLISM; CONCENTRATION RESPONSE; CONFOCAL MICROSCOPY; CONTROLLED STUDY; CYPRINODONTIFORMES; DRUG ACCUMULATION; DRUG METABOLISM; DRUG TOXICITY; DRUG TRANSPORT; FLUORESCENCE; IMAGE ANALYSIS; KIDNEY PROXIMAL TUBULE; NONHUMAN; PRIORITY JOURNAL; STEADY STATE;

EID: 0033984880     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0703003     Document Type: Article

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