A cluster of Ser/Thr residues at the C-terminus of μ-opioid receptor is required for G protein-coupled receptor kinase 2-mediated desensitization

Neuropharmacology

Volumn 39, Issue 3, 2000, Pages 353-363

  Wang, H L ^a  

^a CHANG GUNG UNIVERSITY COLLEGE OF MEDICINE   (Taiwan)

Author keywords

opioid receptor; DAMGO; Desensitization; GRK2

Indexed keywords

COMPLEMENTARY DNA; CYCLIC AMP; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; FORSKOLIN; G PROTEIN COUPLED RECEPTOR; MU OPIATE RECEPTOR; PHOSPHOTRANSFERASE; POLYPEPTIDE; SERINE; THREONINE;

ARTICLE; CONTROLLED STUDY; DELETION MUTANT; EMBRYO; EMBRYO CELL; ENZYME ACTIVATION; GENE EXPRESSION; HUMAN; HUMAN CELL; LIGAND BINDING; MOLECULAR CLONING; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION;

ANALGESICS, OPIOID; ANIMALS; BETA-ADRENERGIC RECEPTOR KINASE; CELL LINE; CYCLIC AMP-DEPENDENT PROTEIN KINASES; DRUG TOLERANCE; ENKEPHALIN, ALA(2)-MEPHE(4)-GLY(5)-; HUMANS; NALOXONE; NARCOTIC ANTAGONISTS; RATS; RECEPTORS, OPIOID, MU; SERINE; THREONINE; TRANSFECTION;

EID: 0033978672     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(99)00174-4     Document Type: Article

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