Binding properties of a highly potent and selective iodinated aminopeptidase N inhibitor appropriate for radioautography

FEBS Letters

Volumn 467, Issue 1, 2000, Pages 81-86

  Noble, Florence ^a   Luciani, Nathalie ^a   Da Nascimento, Sophie ^a   Laï Kuen, René ^b   Bischoff, Laurent ^a   Chen, Huixiong ^a   Fournié Zaluski, Marie Claude ^a   Roques, Bernard P ^a  

^a Laboratoire de Pharmacochimie   (France)

^b UNIVERSITÉ PARIS DESCARTES   (France)

Author keywords

Aminopeptidase N; Binding; Inhibitor; Rat brain membrane; Recombinant APN

Indexed keywords

2 BENZYL 3 [HYDROXY(1' AMINOETHYL)PHOSPHINYL]PROPANOYL 3 IODOTYROSINE; ENZYME INHIBITOR; MICROSOMAL AMINOPEPTIDASE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BRAIN; ENZYME BINDING; ENZYME INHIBITION; IN VITRO STUDY; IODINATION; ISOTOPE LABELING; NONHUMAN; PRIORITY JOURNAL; RAT;

AMINO ACID SUBSTITUTION; ANIMALS; ANTIGENS, CD13; AUTORADIOGRAPHY; BINDING, COMPETITIVE; BRAIN; CELL MEMBRANE; COS CELLS; HYDROXAMIC ACIDS; INTESTINES; IODINE RADIOISOTOPES; MONOIODOTYROSINE; MUTATION; PHENYLALANINE; PROTEASE INHIBITORS; PROTEIN BINDING; RATS; RECOMBINANT PROTEINS; SULFHYDRYL COMPOUNDS; SWINE; THERMODYNAMICS; TRANSFECTION;

EID: 0033978419     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-5793(99)01645-2     Document Type: Article

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