-
1
-
-
0029865228
-
Prospects for β3-adrenoceptor agonists in the treatment of obesity and diabetes
-
Arch JR and Wilson S (1996) Prospects for β3-adrenoceptor agonists in the treatment of obesity and diabetes. Int J Obes Relat Metab Disord 20:191-199.
-
(1996)
Int J Obes Relat Metab Disord
, vol.20
, pp. 191-199
-
-
Arch, J.R.1
Wilson, S.2
-
2
-
-
0009644628
-
Some quantitative uses of drug antagonists
-
Arunlakshana O and Schild HO (1959) Some quantitative uses of drug antagonists. Br J Pharmacol 14:48-58.
-
(1959)
Br J Pharmacol
, vol.14
, pp. 48-58
-
-
Arunlakshana, O.1
Schild, H.O.2
-
3
-
-
0028959882
-
Control of lipolysis in intra-abdominal fat cells of nonhuman primates: Comparison with humans
-
Bousquet-Mélou A, Galitzky J, Lafontan M and Berlan M (1995) Control of lipolysis in intra-abdominal fat cells of nonhuman primates: Comparison with humans. J Lipid Res 36:451-461.
-
(1995)
J Lipid Res
, vol.36
, pp. 451-461
-
-
Bousquet-Mélou, A.1
Galitzky, J.2
Lafontan, M.3
Berlan, M.4
-
4
-
-
0025953997
-
Developmental changes in adenylyl cyclase and GTP binding proteins in brown fat
-
Chaudhry A and Granneman JG (1991) Developmental changes in adenylyl cyclase and GTP binding proteins in brown fat. Am J Physiol 261:R403-R411.
-
(1991)
Am J Physiol
, vol.261
-
-
Chaudhry, A.1
Granneman, J.G.2
-
5
-
-
0028061556
-
Influence of cell type upon the desensitization of the β3-adrenergic receptor
-
Chaudhry A and Granneman JG (1994) Influence of cell type upon the desensitization of the β3-adrenergic receptor. J Pharmacol Exp Ther 271:1253-1258.
-
(1994)
J Pharmacol Exp Ther
, vol.271
, pp. 1253-1258
-
-
Chaudhry, A.1
Granneman, J.G.2
-
7
-
-
0029761541
-
3-adrenoceptors in human brown and white adipose tissues
-
3-adrenoceptors in human brown and white adipose tissues. Br J Pharmacol 118:929-934.
-
(1996)
Br J Pharmacol
, vol.118
, pp. 929-934
-
-
Deng, C.1
Paoloni-Giacobino, A.2
Kuehne, F.3
Boss, O.4
Revelli, J.-P.5
Moinat, M.6
Cawthorne, M.A.7
Muzzin, P.8
Giacobino, J.-P.9
-
9
-
-
0002177268
-
The quantitative effects of antagonist drugs
-
Gaddum JH (1937) The quantitative effects of antagonist drugs. J Physiol (Lond) 89:7P-9P.
-
(1937)
J Physiol (Lond)
, vol.89
-
-
Gaddum, J.H.1
-
11
-
-
0032541084
-
G protein-coupled receptors. II. Mechanism of agonist activation
-
Gether U and Kobilka BK (1998) G protein-coupled receptors. II. Mechanism of agonist activation. J Biol Chem 273;17979-17982.
-
(1998)
J Biol Chem
, vol.273
, pp. 17979-17982
-
-
Gether, U.1
Kobilka, B.K.2
-
12
-
-
0025166751
-
Norepinephrine and BRL 37344 stimulate adenylate cyclase by different receptors in rat brown adipose tissue
-
Granneman JG (1990) Norepinephrine and BRL 37344 stimulate adenylate cyclase by different receptors in rat brown adipose tissue. J Pharmacol Exp Ther 254: 508-513.
-
(1990)
J Pharmacol Exp Ther
, vol.254
, pp. 508-513
-
-
Granneman, J.G.1
-
16
-
-
0031750286
-
Agonist interactions with chimeric and mutant β1- and β3-adrenergic receptors: Involvement of the seventh transmembrane region in conferring subtype selectivity
-
Granneman JG, Lahners KN and Zhai Y (1998) Agonist interactions with chimeric and mutant β1- and β3-adrenergic receptors: Involvement of the seventh transmembrane region in conferring subtype selectivity. Mol Pharmacol 53:856-861.
-
(1998)
Mol Pharmacol
, vol.53
, pp. 856-861
-
-
Granneman, J.G.1
Lahners, K.N.2
Zhai, Y.3
-
17
-
-
0026090708
-
CGP 12177A modulates brown fat adenylate cyclase activity by interacting with two distinct receptor sites
-
Granneman JG and Whitty C (1991) CGP 12177A modulates brown fat adenylate cyclase activity by interacting with two distinct receptor sites. J Pharmacol Exp Ther 256:421-425.
-
(1991)
J Pharmacol Exp Ther
, vol.256
, pp. 421-425
-
-
Granneman, J.G.1
Whitty, C.2
-
19
-
-
0031711336
-
Mice expressing human but not murine beta3-adrenergic receptors under the control of human gene regulatory elements
-
Ito M, Grujic D, Abel ED, Vidal-Puig A, Susulic VS, Lawitts J, Harper ME, Himms-Hagen J, Strosberg AD and Lowell BB (1998) Mice expressing human but not murine beta3-adrenergic receptors under the control of human gene regulatory elements. Diabetes 47:1464-1471.
-
(1998)
Diabetes
, vol.47
, pp. 1464-1471
-
-
Ito, M.1
Grujic, D.2
Abel, E.D.3
Vidal-Puig, A.4
Susulic, V.S.5
Lawitts, J.6
Harper, M.E.7
Himms-Hagen, J.8
Strosberg, A.D.9
Lowell, B.B.10
-
21
-
-
0030776329
-
Modulation of human cardiac function through 4 β-adrenoceptor populations
-
Kaumann AJ and Molenaar P (1997) Modulation of human cardiac function through 4 β-adrenoceptor populations. Naunyn Schmiedebergs Arch Pharmacol 355:667-681.
-
(1997)
Naunyn Schmiedebergs Arch Pharmacol
, vol.355
, pp. 667-681
-
-
Kaumann, A.J.1
Molenaar, P.2
-
22
-
-
0031980254
-
(-)-CGP 12177 causes cardiostimulation and binds to cardiac putative β4-adrenoceptors in both wild-type and β3-adrenoceptor knockout mice
-
Kaumann AJ, Preitner F, Sarsero D, Molenaar P, Revelli JP and Giacobino JP (1998) (-)-CGP 12177 causes cardiostimulation and binds to cardiac putative β4-adrenoceptors in both wild-type and β3-adrenoceptor knockout mice. Mol Pharmacol 53:670-675.
-
(1998)
Mol Pharmacol
, vol.53
, pp. 670-675
-
-
Kaumann, A.J.1
Preitner, F.2
Sarsero, D.3
Molenaar, P.4
Revelli, J.P.5
Giacobino, J.P.6
-
23
-
-
0020053249
-
The Schild regression in the process of receptor classification
-
Kenakin TP (1982) The Schild regression in the process of receptor classification. Can J Physiol Pharmacol 60:249-265.
-
(1982)
Can J Physiol Pharmacol
, vol.60
, pp. 249-265
-
-
Kenakin, T.P.1
-
26
-
-
0024405758
-
3H]CGP-12177, generally classified as an antagonist, is a thermogenic agonist in brown adipose tissue
-
3H]CGP-12177, generally classified as an antagonist, is a thermogenic agonist in brown adipose tissue. Biochem J 261:401-405.
-
(1989)
Biochem J
, vol.261
, pp. 401-405
-
-
Mohell, N.1
Dicker, A.2
-
29
-
-
0031869348
-
Metabolic response to various beta-adrenoceptor agonists in beta3-adrenoceptor knockout mice: Evidence for a new beta-adrenergic receptor in brown adipose tissue
-
Preitner F, Muzzin P, Revelli JP, Seydoux J, Galitzky J, Berlan M, Lafontan M and Giacobino JP (1998) Metabolic response to various beta-adrenoceptor agonists in beta3-adrenoceptor knockout mice: Evidence for a new beta-adrenergic receptor in brown adipose tissue. Br J Pharmacol 124:1684-1688
-
(1998)
Br J Pharmacol
, vol.124
, pp. 1684-1688
-
-
Preitner, F.1
Muzzin, P.2
Revelli, J.P.3
Seydoux, J.4
Galitzky, J.5
Berlan, M.6
Lafontan, M.7
Giacobino, J.P.8
-
30
-
-
0030015497
-
Targeted disruption of the mouse β1-adrenergic receptor gene: Developmental and cardiovascular effects
-
Rohrer DK, Desai KH, Jasper JR, Stevens ME, Regula DP Jr, Barsh GS, Bernstein D and Kobilka BK (1996) Targeted disruption of the mouse β1-adrenergic receptor gene: Developmental and cardiovascular effects. Proc Natl Acad Sci USA 93:7375-7380.
-
(1996)
Proc Natl Acad Sci USA
, vol.93
, pp. 7375-7380
-
-
Rohrer, D.K.1
Desai, K.H.2
Jasper, J.R.3
Stevens, M.E.4
Regula D.P., Jr.5
Barsh, G.S.6
Bernstein, D.7
Kobilka, B.K.8
-
32
-
-
7144254440
-
3-adrenoceptor agonists of differing selectivities
-
3-adrenoceptor agonists of differing selectivities. J Pharmacol Exp Ther 285: 1084-1095.
-
(1998)
J Pharmacol Exp Ther
, vol.285
, pp. 1084-1095
-
-
Sennitt, M.V.1
Kaumann, A.J.2
Molenaar, P.3
Beeley, L.J.4
Young, P.W.5
Kelly, J.6
Chapman, H.7
Henson, S.M.8
Berge, J.M.9
Dean, J.M.10
Kotecha, N.R.11
Morgan, H.K.A.12
Rami, H.K.13
Ward, R.W.14
Thompson, M.15
Wilson, S.16
Smith, S.A.17
Cawthorne, M.A.18
Stock, M.J.19
Arch, J.R.S.20
more..
-
33
-
-
0020523811
-
CGP-12177 a hydrophilic β-adrenergic receptor radioligand reveals high affinity binding of agonists to intact cells
-
Staehelin M, Simons P, Jaeggi K and Wigger N (1983) CGP-12177 a hydrophilic β-adrenergic receptor radioligand reveals high affinity binding of agonists to intact cells. J Biol Chem 258:3496-3502.
-
(1983)
J Biol Chem
, vol.258
, pp. 3496-3502
-
-
Staehelin, M.1
Simons, P.2
Jaeggi, K.3
Wigger, N.4
-
34
-
-
0028838836
-
Targeted disruption of the β3-adrenergic receptor gene
-
Susulic VS, Frederich RC, Lawitts J, Tozzo E, Kahn BB, Harper ME, Himms-Hagen J, Flier JS and Lowell BB (1995) Targeted disruption of the β3-adrenergic receptor gene. J Biol Chem 270:29483-29492.
-
(1995)
J Biol Chem
, vol.270
, pp. 29483-29492
-
-
Susulic, V.S.1
Frederich, R.C.2
Lawitts, J.3
Tozzo, E.4
Kahn, B.B.5
Harper, M.E.6
Himms-Hagen, J.7
Flier, J.S.8
Lowell, B.B.9
-
35
-
-
0029670720
-
Expression of β3-adrenoceptors with low lipolytic action in human subcutaneous white adipocytes
-
Tavernier G, Barbe P, Galitzky J, Berlan M, Caput D, Lafontan M and Langin D (1996) Expression of β3-adrenoceptors with low lipolytic action in human subcutaneous white adipocytes. J Lipid Res 37:87-97.
-
(1996)
J Lipid Res
, vol.37
, pp. 87-97
-
-
Tavernier, G.1
Barbe, P.2
Galitzky, J.3
Berlan, M.4
Caput, D.5
Lafontan, M.6
Langin, D.7
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