5-HT3- and 5-HT(2C)-antagonist properties of cyamemazine: Significance for its clinical anxiolytic activity

Psychopharmacology

Volumn 147, Issue 4, 2000, Pages 412-417

  Alvarez Guerra, Miriam ^a,b,c   D'Alché Birée, Françoise ^a,b,c   Wolf, William A ^a,b,c   Vargas, Felix ^a,b,c   Dib, Michel ^a,b,c   Garay, Ricardo P ^a,b,c  

^a INSERM   (France)

^b VETERANS AFFAIRS MEDICAL CENTER   (United States)

^c UNIVERSITY OF GRANADA   (Spain)

Author keywords

5 HT(2C) receptor; 5 HT3 receptor; Anxiety; Cyamemazine; Serotonin

Indexed keywords

CYAMEMAZINE; PHOSPHOLIPASE C; SEROTONIN 2C ANTAGONIST; SEROTONIN ANTAGONIST; ANXIOLYTIC AGENT; NEUROLEPTIC AGENT; PHENOTHIAZINE DERIVATIVE; SEROTONIN 2C RECEPTOR; SEROTONIN 3 RECEPTOR; SEROTONIN RECEPTOR;

ANIMAL CELL; ANIMAL TISSUE; ANXIETY; ARTICLE; BRADYCARDIA; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG RECEPTOR BINDING; GUINEA PIG; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; SEROTONIN RELEASE; TRANQUILIZING ACTIVITY; ANIMAL; CAUDATE NUCLEUS; DRUG EFFECT; ENZYMOLOGY; HEART RATE; IN VITRO STUDY; MEMBRANE; METABOLISM; MUSCLE CONTRACTION; RADIOASSAY; VASCULAR SMOOTH MUSCLE; WISTAR RAT;

ANIMALS; ANTI-ANXIETY AGENTS; ANTIPSYCHOTIC AGENTS; CAUDATE NUCLEUS; GUINEA PIGS; HEART RATE; MALE; MEMBRANES; MUSCLE CONTRACTION; MUSCLE, SMOOTH, VASCULAR; PHENOTHIAZINES; PHOSPHOLIPASE C; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTOR, SEROTONIN, 5-HT2C; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN ANTAGONISTS;

EID: 0033621678     PISSN: 00333158     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002130050010     Document Type: Article

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