P2-achiral, P'-extended α-ketoamide inhibitors of calpain I

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 16, 1999, Pages 2371-2374

  Chatterjee, Sankar ^a   Dunn, Derek ^a   Tao, Ming ^a   Wells, Gregory ^a   Gu, Zi Qiang ^a   Bihovsky, Ron ^a   Ator, Mark A ^a   Siman, Robert ^a   Mallamo, John P ^a  

^a CEPHALON INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA KETOAMIDE INHIBITOR; CALPAIN; PROTEINASE INHIBITOR; UNCLASSIFIED DRUG; AMIDE; RECOMBINANT PROTEIN;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; CHEMISTRY; DRUG ANTAGONISM; HUMAN; STEREOISOMERISM;

AMIDES; CALPAIN; HUMANS; PROTEASE INHIBITORS; RECOMBINANT PROTEINS; STEREOISOMERISM;

EID: 0033575514     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00392-3     Document Type: Article

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