A continuous fluorescence assay for the study of p-glycoprotein-mediated drug efflux using inside-out membrane vesicles

Analytical Biochemistry

Volumn 268, Issue 2, 1999, Pages 270-277

  Bebawy, Mary ^a   Morris, Michael B ^a   Roufogalis, Basil D ^a  

^a UNIVERSITY OF SYDNEY   (Australia)

Author keywords

Fluorescein colchicine; Inside out membrane vesicle; Methylene blue; Multidrug resistance; P glycoprotein substrates

Indexed keywords

ALKALOIDS; AROMATIC COMPOUNDS; DYES; FLUORESCENCE; PROBES; SUBSTRATES;

FLUORESCEIN-COLCHICINE; MEMBRANE VESICLES; METHYLENE BLUE; MULTIDRUG RESISTANCE; P-GLYCOPROTEIN;

GLYCOPROTEINS;

ADENOSINE TRIPHOSPHATASE (POTASSIUM SODIUM); COLCHICINE; FLUORESCEIN; GLYCOPROTEIN P; METHOTREXATE; VANADIC ACID; VERAPAMIL; VINBLASTINE;

ARTICLE; DRUG TRANSPORT; ENZYME ACTIVITY; FLUORESCENCE ANALYSIS; FLUOROMETRY; HUMAN; HUMAN CELL; LEUKEMIA CELL; MEMBRANE MODEL; MEMBRANE TRANSPORT; PRIORITY JOURNAL;

EID: 0033559160     PISSN: 00032697     EISSN: None     Source Type: Journal    
DOI: 10.1006/abio.1998.3087     Document Type: Article

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