Design, synthesis, and evaluation of novel modular bisubstrate analogue inhibitors of farnesyltransferase

Angewandte Chemie - International Edition

Volumn 38, Issue 13-14, 1999, Pages 2032-2034

  Schlitzer, Martin ^a   Sattler, Isabel ^b  

^a PHILIPPS UNIVERSITY MARBURG   (Germany)

^b HANS KNÖLL INSTITUTE   (Germany)

Author keywords

Enzyme inhibitors; Farnesyltransferase; Peptidomimetics; Signal transduction; Tumour therapy

Indexed keywords

PROTEIN FARNESYLTRANSFERASE INHIBITOR;

ARTICLE; CHEMICAL REACTION; DRUG STRUCTURE; DRUG SYNTHESIS; FLUORESCENCE; KINETICS; REACTION ANALYSIS; SACCHAROMYCES CEREVISIAE; STRUCTURE ANALYSIS;

EID: 0033549534     PISSN: 14337851     EISSN: None     Source Type: Journal    
DOI: 10.1002/(sici)1521-3773(19990712)38:13/14<2032::aid-anie2032>3.0.co;2-d     Document Type: Article

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