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3
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0013620126
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Marketed as Evista® (Raloxifene Hydrochloride 60 mg)
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Marketed as Evista® (Raloxifene Hydrochloride 60 mg).
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4
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0021201213
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Sall, D. J.; Bastian, J. A.; Briggs, S. L.; Buben, J. A.; Chirgadze, N. Y; Clawson, D. K.; Denney, M. L.; Giera, D. D.; Gifford-Moore, D. S.; Harper, R. W.; Hauser, K. L.; Klimkowski, V. J.; Kohn, T. J.; Lin, H.-S.; McCowan, J. R.; Palkowitz, A. D.; Smith, G. F.; Takeuchi, K.; Thrasher, K. J.; Tinsley, J. M.; Utterback, B. G.; Yan, S.-C. B.; Zhang, M. J. Med. Chem. 1997, 40, 3489-3493.
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Denney, M.L.7
Giera, D.D.8
Gifford-Moore, D.S.9
Harper, R.W.10
Hauser, K.L.11
Klimkowski, V.J.12
Kohn, T.J.13
Lin, H.-S.14
McCowan, J.R.15
Palkowitz, A.D.16
Smith, G.F.17
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Thrasher, K.J.19
Tinsley, J.M.20
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more..
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23
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0001560775
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All compounds exhibited satisfactory spectral (IR, PMR, CMR) and analytical (EA or HRMS) data
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Ablenas, F. J.; George, B. E.; Maleki, M.; Jain, R.; Hopkinson, A. C.; Lee-Ruff, E. Can. J. Chem. 1987, 65, 1800-1803. All compounds exhibited satisfactory spectral (IR, PMR, CMR) and analytical (EA or HRMS) data.
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0026028015
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NAr has been used on a highly activated perfluorobenzoyl group to prepare a benzothiophene-based reagent for photoaffinity labeling of the estrogen receptor. See
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NAr has been used on a highly activated perfluorobenzoyl group to prepare a benzothiophene-based reagent for photoaffinity labeling of the estrogen receptor. See
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Schissel, D.N.2
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NAr conditions employing dipolar aprotic solvents on substrates of similar reactivity have recently appeared. See
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NAr conditions employing dipolar aprotic solvents on substrates of similar reactivity have recently appeared. See
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33
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0032558508
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Colleagues at Lilly have recently disclosed application of our methodology to the preparation of thrombin inhibitors. See: (a) Sall, D. J.; Briggs, S. L; Chirgadze, N. Y; Clawson, D. K.; Gifford-Moore, D. S,; Klimkowshi, V. J.; McCowan, J. R.; Smith, G. F.; Wikel, J. H. Bioorg. Med. Chem. Lett. 1998, 8, 2527-2532.
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Klimkowshi, V.J.6
McCowan, J.R.7
Smith, G.F.8
Wikel, J.H.9
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34
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0033535105
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(b) Bastian, J. A.; Chirgadze, N.; Denney, M. L.; Gifford-Moore, D. S.; Sall, D. J.; Smith, G. F.; Wikel, J. H. Bioorg. Med. Chem. Lett. 1999, 9, 363-368.
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Sall, D.J.5
Smith, G.F.6
Wikel, J.H.7
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35
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0033535387
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(c) Takeuchi, K.; Kohn, T. J.; Sall, D. J.; Denney, M. L.; McGowan, J. R.; Smith, G. F.; Gifford-Moore, D. S. Bioorg. Med. Chem. Lett 1999, 9, 759-764.
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Smith, G.F.6
Gifford-Moore, D.S.7
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