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Volumn 40, Issue 28, 1999, Pages 5155-5159

Synergistic methodologies for the synthesis of 3-aroyl-2- arylbenzo[b]thiophene-based selective estrogen receptor modulators. Two concise syntheses of raloxifene

Author keywords

[No Author keywords available]

Indexed keywords

ESTROGEN; ESTROGEN RECEPTOR; RALOXIFENE;

EID: 0033538646     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(99)00955-7     Document Type: Article
Times cited : (39)

References (35)
  • 3
    • 0013620126 scopus 로고    scopus 로고
    • Marketed as Evista® (Raloxifene Hydrochloride 60 mg)
    • Marketed as Evista® (Raloxifene Hydrochloride 60 mg).
  • 8
  • 17
    • 0013574646 scopus 로고    scopus 로고
    • U.S. Patent 5 466 810
    • (a) Godfrey, A. G. U.S. Patent 5 466 810, 1995;
    • Godfrey, A.G.1
  • 18
    • 0040485885 scopus 로고    scopus 로고
    • Chem. Abstr. 1996, 124, 175, 813.
    • (1996) Chem. Abstr. , vol.124 , Issue.175 , pp. 813
  • 19
    • 0013625550 scopus 로고    scopus 로고
    • U.S. Patent 5 420 349
    • (b) Godfrey, A. G. U.S. Patent 5 420 349, 1995;
    • Godfrey, A.G.1
  • 20
    • 0013601864 scopus 로고
    • Chem. Abstr. 1995, 123, 111, 843.
    • (1995) Chem. Abstr. , vol.123 , Issue.111 , pp. 843
  • 23
    • 0001560775 scopus 로고
    • All compounds exhibited satisfactory spectral (IR, PMR, CMR) and analytical (EA or HRMS) data
    • Ablenas, F. J.; George, B. E.; Maleki, M.; Jain, R.; Hopkinson, A. C.; Lee-Ruff, E. Can. J. Chem. 1987, 65, 1800-1803. All compounds exhibited satisfactory spectral (IR, PMR, CMR) and analytical (EA or HRMS) data.
    • (1987) Can. J. Chem. , vol.65 , pp. 1800-1803
    • Ablenas, F.J.1    George, B.E.2    Maleki, M.3    Jain, R.4    Hopkinson, A.C.5    Lee-Ruff, E.6
  • 29
    • 0026028015 scopus 로고
    • NAr has been used on a highly activated perfluorobenzoyl group to prepare a benzothiophene-based reagent for photoaffinity labeling of the estrogen receptor. See
    • NAr has been used on a highly activated perfluorobenzoyl group to prepare a benzothiophene-based reagent for photoaffinity labeling of the estrogen receptor. See
    • (1991) Synthesis , pp. 63-68
    • Yeager, G.W.1    Schissel, D.N.2
  • 30
    • 33751499160 scopus 로고
    • NAr conditions employing dipolar aprotic solvents on substrates of similar reactivity have recently appeared. See
    • NAr conditions employing dipolar aprotic solvents on substrates of similar reactivity have recently appeared. See
    • (1991) J. Org. Chem. , vol.56 , pp. 3125-3133
    • Pinney, K.G.1    Katzenellenbogen, J.A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.