Complementarity of δ opioid ligand pharmacophore and receptor models

Biopolymers - Peptide Science Section

Volumn 51, Issue 6, 1999, Pages 426-439

  Mosberg, Henry I ^a  

^a UNIVERSITY OF MICHIGAN   (United States)

Author keywords

Bioactive conformation; Conformationally restricted peptides; G protein coupled receptors; Ligand receptor interactions; Molecular recognition; Opioid peptides

Indexed keywords

BIOLOGICAL MEMBRANES; CONFORMATIONS; MATHEMATICAL MODELS; PHYSIOLOGICAL MODELS; PROTEINS;

LIGANDS; MOLECULAR RECOGNITION; PHARMACOPHORES;

POLYPEPTIDES;

DELTA OPIATE RECEPTOR; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; G PROTEIN COUPLED RECEPTOR; LEUCINE ENKEPHALIN; METENKEPHALIN; TYROSYLCYCLO[DEXTRO CYSTEINYLPHENYLALANYL DEXTRO PENICILLAMINE];

ARTICLE; BINDING AFFINITY; CONFORMATIONAL TRANSITION; DRUG BINDING SITE; DRUG CONFORMATION; DRUG RECEPTOR BINDING; DRUG STRUCTURE; HYDROGEN BOND; MOLECULAR RECOGNITION; PHARMACOPHORE;

AMINO ACID SEQUENCE; BINDING SITES; GTP-BINDING PROTEINS; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; OPIOID PEPTIDES; PROTEIN CONFORMATION; RECEPTORS, OPIOID; STEREOISOMERISM;

EID: 0033511768     PISSN: 00063525     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1097-0282(1999)51:6<426::AID-BIP5>3.0.CO;2-G     Document Type: Article

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