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Volumn 19, Issue 1-4, 1999, Pages 547-557

Reactive affinity probes for the mapping of the glycine-binding site of the NMDA receptor NR1 subunit

Author keywords

[No Author keywords available]

Indexed keywords

7 CHLORO 4 HYDROXY 3 (3 PHENOXYPHENYL) 2 QUINOLONE; CYSTEINE; DIZOCILPINE; KYNURENIC ACID DERIVATIVE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR STIMULATING AGENT; PHENCYCLIDINE; RECEPTOR SUBUNIT;

EID: 0033054454     PISSN: 10799893     EISSN: None     Source Type: Journal    
DOI: 10.3109/10799899909036671     Document Type: Conference Paper
Times cited : (2)

References (32)
  • 1
    • 0027466062 scopus 로고
    • The Role of NMDA Receptors in Information Processing
    • Daw, N. W.; Stein, P. S. G.; and Fox, K. The Role of NMDA Receptors in Information Processing. Annu. Rev. Neurosci. 16, 207-222, 1993.
    • (1993) Annu. Rev. Neurosci. , vol.16 , pp. 207-222
    • Daw, N.W.1    Stein, P.S.G.2    Fox, K.3
  • 2
    • 0028179069 scopus 로고
    • N-methyl-D-aspartic acid receptor structure and function
    • McBain, C. J.; and Mayer, M. L. N-methyl-D-aspartic acid receptor structure and function. Physiol. Rev. 74, 723-760, 1994.
    • (1994) Physiol. Rev. , vol.74 , pp. 723-760
    • McBain, C.J.1    Mayer, M.L.2
  • 3
    • 0027487896 scopus 로고
    • The NMDA receptor complex
    • Scatton, B. The NMDA receptor complex. Fundam. Clin. Pharmacol. 7, 389-400, 1993.
    • (1993) Fundam. Clin. Pharmacol. , vol.7 , pp. 389-400
    • Scatton, B.1
  • 4
    • 0002083159 scopus 로고
    • The pharmacology of excitatory amino acids: A TIPS special report
    • Lodge, D.; and Collingridge, G. The pharmacology of excitatory amino acids: a TIPS special report. Trends Pharmacol. Sci. (special issue), 1-89, 1991.
    • (1991) Trends Pharmacol. Sci. , Issue.SPEC. ISSUE , pp. 1-89
    • Lodge, D.1    Collingridge, G.2
  • 5
    • 33845189959 scopus 로고    scopus 로고
    • NMDA antagonists: Their role in neuroprotection
    • Small, D. L.; and Buchan, A. L. NMDA antagonists: their role in neuroprotection. Int. Rev. Neurobiol. 40, 137-171, 1997.
    • (1997) Int. Rev. Neurobiol. , vol.40 , pp. 137-171
    • Small, D.L.1    Buchan, A.L.2
  • 6
    • 0003062412 scopus 로고
    • edited by G. L. Collingridge, and J. C. Watkins, Oxford University Press, Oxford
    • Lodge, D.; Jones, M.; and Fletcher, E. In The NMDA receptor, edited by G. L. Collingridge, and J. C. Watkins, p. 105-131, Oxford University Press, Oxford, 1994.
    • (1994) The NMDA Receptor , pp. 105-131
    • Lodge, D.1    Jones, M.2    Fletcher, E.3
  • 7
    • 0003131895 scopus 로고
    • edited by G. L. Collingridge, and J. C. Watkins, Oxford University Press, Oxford
    • Jane, D. E.; Olverman, H. J.; and Watkins, J. C. In The NMDA receptor, edited by G. L. Collingridge, and J. C. Watkins, p. 31-104, Oxford University Press, Oxford, 1994.
    • (1994) The NMDA Receptor , pp. 31-104
    • Jane, D.E.1    Olverman, H.J.2    Watkins, J.C.3
  • 8
    • 0032576701 scopus 로고    scopus 로고
    • Quantitative analysis of the structural requirements for blockade of the N-methyl-D-aspartate receptor at the phencyclidine binding site
    • Kroemer, R. T.; Koutsilieri, E.; Hecht, P.; Liedl, K. R.; Riederer, P.; and Kornhuber, J. Quantitative analysis of the structural requirements for blockade of the N-methyl-D-aspartate receptor at the phencyclidine binding site. J. Med. Chem. 41, 393-400, 1998.
    • (1998) J. Med. Chem. , vol.41 , pp. 393-400
    • Kroemer, R.T.1    Koutsilieri, E.2    Hecht, P.3    Liedl, K.R.4    Riederer, P.5    Kornhuber, J.6
  • 9
    • 0025740632 scopus 로고
    • Kynurenic acid derivatives. Structure-activity relationships for excitatory amino acid antagonism and identification of potent and selective antagonists at the glycine site on the N-methyl-D-aspartate receptor
    • Leeson, P. D.; Baker, R.; Carling, R. W.; Curtis, N. R.; Moore, K. W.; Williams, B. J.; Foster, A. C.; Donald, A. E.; Kemp, J. A.; and Marshall, G. R. Kynurenic acid derivatives. Structure-activity relationships for excitatory amino acid antagonism and identification of potent and selective antagonists at the glycine site on the N-methyl-D-aspartate receptor. J. Med. Chem. 34, 1343-1352, 1991.
    • (1991) J. Med. Chem. , vol.34 , pp. 1343-1352
    • Leeson, P.D.1    Baker, R.2    Carling, R.W.3    Curtis, N.R.4    Moore, K.W.5    Williams, B.J.6    Foster, A.C.7    Donald, A.E.8    Kemp, J.A.9    Marshall, G.R.10
  • 10
    • 0027988561 scopus 로고
    • The glycine site on the NMDA receptor: Structure activity relationships and therapeutic potentials
    • Leeson, P. D.; and Iversen, L. L. The glycine site on the NMDA receptor: Structure activity relationships and therapeutic potentials. J. Med. Chem. 37, 4053-4067, 1994.
    • (1994) J. Med. Chem. , vol.37 , pp. 4053-4067
    • Leeson, P.D.1    Iversen, L.L.2
  • 11
    • 0028979826 scopus 로고
    • Molecular design of the N-methyl-D-aspartate receptor binding site for phencyclidine and dizolcipine
    • Ferrer-Montiel, A. V.; Sun, W.; and Montai, M. Molecular design of the N-methyl-D-aspartate receptor binding site for phencyclidine and dizolcipine. Proc. Natl. Acad. Sci. USA 92, 8021-8025, 1995.
    • (1995) Proc. Natl. Acad. Sci. USA , vol.92 , pp. 8021-8025
    • Ferrer-Montiel, A.V.1    Sun, W.2    Montai, M.3
  • 12
    • 0028284469 scopus 로고
    • Mutational analysis of the glycine-binding site of the NMDA receptor: Structural similarity with bacterial amino acid-binding proteins
    • Kuryatov, A.; Laube, B.; Betz, H.; and Kuhse, J. Mutational analysis of the glycine-binding site of the NMDA receptor: Structural similarity with bacterial amino acid-binding proteins. Neuron 12, 1291-1300, 1994.
    • (1994) Neuron , vol.12 , pp. 1291-1300
    • Kuryatov, A.1    Laube, B.2    Betz, H.3    Kuhse, J.4
  • 13
    • 0028921951 scopus 로고
    • Identification of amino acids in the N-methyl-D-aspartate receptor NR1 subunit that contribute to the glycine-binding site
    • Wafford, K. A.; Kathoria, M.; Bain, C. J.; Marshall, G.; Lebourdelles, B.; Kemp, J. A.; and Whiting, P. J. Identification of amino acids in the N-methyl-D-aspartate receptor NR1 subunit that contribute to the glycine-binding site. Mol. Pharmacol. 47, 374-380, 1995.
    • (1995) Mol. Pharmacol. , vol.47 , pp. 374-380
    • Wafford, K.A.1    Kathoria, M.2    Bain, C.J.3    Marshall, G.4    Lebourdelles, B.5    Kemp, J.A.6    Whiting, P.J.7
  • 14
    • 0029921964 scopus 로고    scopus 로고
    • Activation of N-methyl-D-aspartate receptors by glycine: Role of an aspartate residue in the M3-M4 loop of the NR1 subunit
    • Williams, K.; Chao, J.; Kashiwagi, K.; Masuko, T.; and Igarashi, K. Activation of N-methyl-D-aspartate receptors by glycine: Role of an aspartate residue in the M3-M4 loop of the NR1 subunit. Mol. Pharmacol. 50, 701-708, 1996.
    • (1996) Mol. Pharmacol. , vol.50 , pp. 701-708
    • Williams, K.1    Chao, J.2    Kashiwagi, K.3    Masuko, T.4    Igarashi, K.5
  • 15
    • 0031023519 scopus 로고    scopus 로고
    • An alanine residue in the M3-M4 linker lines the glycine binding pocket of the N-methyl-D-aspartate receptor
    • Wood, M. W.; VanDongen, H. M. A.; and VanDongen, A. M. J. An alanine residue in the M3-M4 linker lines the glycine binding pocket of the N-methyl-D-aspartate receptor. J. Biol. Chem. 272, 3532-3537, 1997.
    • (1997) J. Biol. Chem. , vol.272 , pp. 3532-3537
    • Wood, M.W.1    VanDongen, H.M.A.2    VanDongen, A.M.J.3
  • 16
    • 0030887429 scopus 로고    scopus 로고
    • Analysis of the glycine binding domain of the NMDA receptor channel zeta 1 subunit
    • Uchino, S.; NakajimaLijima, S.; Okuda, K.; Mishina, M.; and Kawamoto, S. Analysis of the glycine binding domain of the NMDA receptor channel zeta 1 subunit. Neuroreport 8, 445-449, 1997.
    • (1997) Neuroreport , vol.8 , pp. 445-449
    • Uchino, S.1    NakajimaLijima, S.2    Okuda, K.3    Mishina, M.4    Kawamoto, S.5
  • 17
    • 0029893942 scopus 로고    scopus 로고
    • The glycine binding site of the N-methyl-D-aspartate receptor subunit NR1: Identification of novel determinants of co-agonist potentiation in the extracellular M3-M4 loop region
    • Hirai, H.; Kirsch, J.; Laube, B.; Betz, H.; and Kuhse, J. The glycine binding site of the N-methyl-D-aspartate receptor subunit NR1: Identification of novel determinants of co-agonist potentiation in the extracellular M3-M4 loop region. Proc. Natl. Acad. Sci. USA 93, 6031-6036, 1996.
    • (1996) Proc. Natl. Acad. Sci. USA , vol.93 , pp. 6031-6036
    • Hirai, H.1    Kirsch, J.2    Laube, B.3    Betz, H.4    Kuhse, J.5
  • 18
    • 0030991790 scopus 로고    scopus 로고
    • Molecular determinants of agonist discrimination by NMDA receptor subunits: Analysis of the glutamate binding site on the NR2B subunit
    • Laube, B.; Hirai, H.; Sturgess, M.; Betz, H.; and Kuhse, J. Molecular determinants of agonist discrimination by NMDA receptor subunits: Analysis of the glutamate binding site on the NR2B subunit. Neuron 18, 493-503, 1997.
    • (1997) Neuron , vol.18 , pp. 493-503
    • Laube, B.1    Hirai, H.2    Sturgess, M.3    Betz, H.4    Kuhse, J.5
  • 19
  • 20
    • 13044308629 scopus 로고
    • Über Derivate der Nitrophtalsäuren
    • Seidel, H.; and Bittner, J. C. Über Derivate der Nitrophtalsäuren. Monatshefte Chem. 23, 415-425, 1902.
    • (1902) Monatshefte Chem. , vol.23 , pp. 415-425
    • Seidel, H.1    Bittner, J.C.2
  • 21
    • 0345508076 scopus 로고    scopus 로고
    • A convenient synthesis of nitriles from primary amides under mild conditions
    • Campagna, F.; Carotti, A.; and Casini, G. A convenient synthesis of nitriles from primary amides under mild conditions. Tetrahedron Lett. 21, 1813-1816, 1997.
    • (1997) Tetrahedron Lett. , vol.21 , pp. 1813-1816
    • Campagna, F.1    Carotti, A.2    Casini, G.3
  • 22
    • 0002075852 scopus 로고
    • Reduction of aromatic nitro compounds by titanium(III) chloride
    • Ho, T.-L.; and Wong, C. M. Reduction of aromatic nitro compounds by titanium(III) chloride. J. Org. Chem. 39, 45, 1974.
    • (1974) J. Org. Chem. , vol.39 , pp. 45
    • Ho, T.-L.1    Wong, C.M.2
  • 23
    • 0024843391 scopus 로고
    • Different modes of action of 3-amino-1-hydroxy-2-pyrrolidone (HA-966) and 7-chlorokynurenic acid in the modulation of N-methyl-D-aspartate-sensitive glutamate receptor
    • Danysz, W.; Fadda, E.; Wroblewski, J. T.; and Costa, E. Different modes of action of 3-amino-1-hydroxy-2-pyrrolidone (HA-966) and 7-chlorokynurenic acid in the modulation of N-methyl-D-aspartate-sensitive glutamate receptor. Mol. Pharmacol. 36, 912-916, 1989.
    • (1989) Mol. Pharmacol. , vol.36 , pp. 912-916
    • Danysz, W.1    Fadda, E.2    Wroblewski, J.T.3    Costa, E.4
  • 25
    • 0028845059 scopus 로고
    • Nonlinear regression using spreadsheets
    • Bowen, W. P.; and Jerman, J. C. Nonlinear regression using spreadsheets. Trends Pharmacol. Sci. 16, 413-417, 1995.
    • (1995) Trends Pharmacol. Sci. , vol.16 , pp. 413-417
    • Bowen, W.P.1    Jerman, J.C.2
  • 28
    • 0000039703 scopus 로고    scopus 로고
    • Synthesis and structure-activity relationships of 1,2,3,4-tetrahydroquinoline-2,3,4-trione 3-oximes: Novel and highly potent antagonists for NMDA receptor glycine site
    • Cai, S. X.; Zhou, Z. L.; Huang, J. C.; Whittemore, E. R.; Egbuwoku, Z. O.; Lu, Y. X.; Hawkinson, J. E.; Woodward, R. M.; Weber, E.; and Keana, J. F. W. Synthesis and structure-activity relationships of 1,2,3,4-tetrahydroquinoline-2,3,4-trione 3-oximes: Novel and highly potent antagonists for NMDA receptor glycine site. J. Med. Chem. 39, 3248-3255, 1996.
    • (1996) J. Med. Chem. , vol.39 , pp. 3248-3255
    • Cai, S.X.1    Zhou, Z.L.2    Huang, J.C.3    Whittemore, E.R.4    Egbuwoku, Z.O.5    Lu, Y.X.6    Hawkinson, J.E.7    Woodward, R.M.8    Weber, E.9    Keana, J.F.W.10
  • 29
    • 0026686821 scopus 로고
    • Cloning of an apparent splice variant of the rat N-methyl-D-aspartate receptor NMDAR1 with altered sensitivity to polyamines and activators of protein kinase-C
    • Durand, G. M.; Gregor, P.; Zheng, X.; Bennett, M. V. L.; Uhl, G. R.; and Zukin, R. S. Cloning of an apparent splice variant of the rat N-methyl-D-aspartate receptor NMDAR1 with altered sensitivity to polyamines and activators of protein kinase-C. Proc. Natl. Acad. Sci. USA 89, 9359-9363, 1992.
    • (1992) Proc. Natl. Acad. Sci. USA , vol.89 , pp. 9359-9363
    • Durand, G.M.1    Gregor, P.2    Zheng, X.3    Bennett, M.V.L.4    Uhl, G.R.5    Zukin, R.S.6
  • 30
    • 0028169661 scopus 로고
    • Ligand affinities at recombinant N-methyl-D-aspartate receptors depend on subunit composition
    • Laurie, D. J.; and Seeburg, P. H. Ligand affinities at recombinant N-methyl-D-aspartate receptors depend on subunit composition. Eur. J. Pharmacol.-Molec. Pharm. 268, 335-345, 1994.
    • (1994) Eur. J. Pharmacol.-Molec. Pharm. , vol.268 , pp. 335-345
    • Laurie, D.J.1    Seeburg, P.H.2


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