Identification of a domain affecting agonist potency of meta-chlorophenylbiguanide in 5-HT3 receptors

European Journal of Pharmacology

Volumn 369, Issue 1, 1999, Pages 125-132

  Mochizuki, Shinobu ^a   Miyake, Akira ^a   Furuichi, Kiyoshi ^a  

^a Inst Drug Discov Res   (Japan)

Author keywords

5 HT3 receptor; Ion channel, ligand gated; Meta chlorophenylbiguanide; Xenopus oocyte

Indexed keywords

1 (3 CHLOROPHENYL)BIGUANIDE; ION CHANNEL; SEROTONIN 3 RECEPTOR;

AMINO ACID SEQUENCE; ANIMAL CELL; ARTICLE; BINDING AFFINITY; CHANNEL GATING; DRUG POTENCY; NONHUMAN; NUCLEOTIDE SEQUENCE; OOCYTE; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN EXPRESSION; RECEPTOR AFFINITY; XENOPUS;

AMINO ACID SEQUENCE; ANIMALS; BIGUANIDES; BINDING SITES; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROPHYSIOLOGY; GENE EXPRESSION; HUMANS; MEMBRANE POTENTIALS; MOLECULAR SEQUENCE DATA; MUTATION; OOCYTES; PATCH-CLAMP TECHNIQUES; RATS; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; RECOMBINANT FUSION PROTEINS; SEQUENCE HOMOLOGY, AMINO ACID; SEROTONIN AGONISTS; XENOPUS;

EID: 0032990485     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00058-8     Document Type: Article

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