Microphysiometric analysis of human α(1a)-adrenoceptor expressed in Chinese hamster ovary cells

British Journal of Pharmacology

Volumn 127, Issue 4, 1999, Pages 962-968

  Taniguchi, Takanobu ^a   Inagaki, Rika ^a   Murata, Satoshi ^a   Akiba, Isamu ^b   Muramatsu, Ikunobu ^a  

^a UNIVERSITY OF FUKUI   (Japan)

^b NIPPON BOEHRINGER INGELHEIM CO LTD   (Japan)

Author keywords

1 adrenoceptor; Microphysiometer; Partial agonist; Spare receptor

Indexed keywords

2 [[2 (2,6 DIMETHOXYPHENOXY)ETHYL]AMINOMETHYL] 1,4 BENZODIOXAN; 8 [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] 8 AZASPIRO[4.5]DECANE 7,9 DIONE; ALPHA 1A ADRENERGIC RECEPTOR; CLONIDINE; METHOXAMINE; NORADRENALIN; OXYMETAZOLINE; PHENYLEPHRINE; PRAZOSIN; RADIOLIGAND;

ACIDIFICATION; ANIMAL CELL; ARTICLE; BINDING AFFINITY; CELL CLONE; CHO CELL; DRUG POTENCY; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR DENSITY;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; CHO CELLS; CRICETINAE; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; HYDROGEN-ION CONCENTRATION; NOREPINEPHRINE; RECEPTORS, ADRENERGIC, ALPHA-1; RECOMBINANT PROTEINS;

EID: 0032983684     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702609     Document Type: Article

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