Competitive antagonism of the mouse 5-hydroxytryptamine3 receptor by bisindolylmaleimide I, a 'selective' protein kinase C inhibitor

Journal of Pharmacology and Experimental Therapeutics

Volumn 290, Issue 1, 1999, Pages 76-82

  Coultrap, Steven J ^a   Sun, Hongwei ^a   Tenner Jr , Thomas E ^a   Machu, Tina K ^a  

^a TEXAS TECH UNIVERSITY HEALTH SCIENCES CENTER SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 [1 (3 DIMETHYLAMINOPROPYL) 3 INDOLYL] 3 (3 INDOLYL)MALEIMIDE; 3 (5 METHYL 1H IMIDAZOL 4 YL) 1 (1 METHYL 1H INDOL 3 YL) 1 PROPANONE; CALPHOSTIN C; CHELERYTHRINE; SEROTONIN 3 RECEPTOR; STAUROSPORINE;

ANIMAL CELL; ARTICLE; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG BINDING SITE; DRUG POTENCY; DRUG RECEPTOR BINDING; ENZYME INHIBITION; NONHUMAN; PRIORITY JOURNAL;

ALKALOIDS; ANIMALS; BENZOPHENANTHRIDINES; BINDING, COMPETITIVE; CELL MEMBRANE; DNA; ENZYME INHIBITORS; INDOLES; MALEIMIDES; MICE; NAPHTHALENES; OOCYTES; PATCH-CLAMP TECHNIQUES; PHENANTHRIDINES; PROTEIN KINASE C; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; RNA; SEROTONIN ANTAGONISTS; STAUROSPORINE; XENOPUS LAEVIS;

EID: 0032966912     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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