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Volumn 288, Issue 1, 1999, Pages 204-210

Differences in degree of trapping of low-affinity uncompetitive N- methyl-D-aspartic acid receptor antagonists with similar kinetics of block

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINO 5 PHOSPHONOVALERIC ACID; AMANTADINE; AMINOACRIDINE; DIZOCILPINE; KETAMINE; LANICEMINE; MEMANTINE; N METHYL DEXTRO ASPARTIC ACID; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT;

EID: 0032934209     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (90)

References (28)
  • 1
    • 0028915935 scopus 로고
    • Trapping of glutamate and glycine during open channel block of rat hippocampal neuron NMDA receptors by 9-aminoacridine
    • Benveniste M and Mayer M (1995) Trapping of glutamate and glycine during open channel block of rat hippocampal neuron NMDA receptors by 9-aminoacridine. J Physiol 483:367-384.
    • (1995) J Physiol , vol.483 , pp. 367-384
    • Benveniste, M.1    Mayer, M.2
  • 2
    • 0028971863 scopus 로고
    • N-Methyl-D-aspartate- or glutamate-mediated toxicity in cultured rat cortical neurons is antagonized by FPL 15896AR
    • Black MA, Tremblay R, Mealing G, Ray R, Durkin JP, Whitfield JF, Blosser J and Morley P (1995) N-Methyl-D-aspartate- or glutamate-mediated toxicity in cultured rat cortical neurons is antagonized by FPL 15896AR. J Neurochem 65:2170-2177.
    • (1995) J Neurochem , vol.65 , pp. 2170-2177
    • Black, M.A.1    Tremblay, R.2    Mealing, G.3    Ray, R.4    Durkin, J.P.5    Whitfield, J.F.6    Blosser, J.7    Morley, P.8
  • 3
    • 0031020529 scopus 로고    scopus 로고
    • Trapping channel block of NMDA-activated responses by amantadine and memantine
    • Blanpied TA, Boeckman FA, Aizenman E and Johnson JW (1997) Trapping channel block of NMDA-activated responses by amantadine and memantine. J Neurophysiol 77:309-323.
    • (1997) J Neurophysiol , vol.77 , pp. 309-323
    • Blanpied, T.A.1    Boeckman, F.A.2    Aizenman, E.3    Johnson, J.W.4
  • 4
    • 0031034905 scopus 로고    scopus 로고
    • Mechanism of memantine block of NMDA-activated channels in rat retinal ganglion cells: Uncompetitive antagonism
    • Chen HV and Lipton S (1997) Mechanism of memantine block of NMDA-activated channels in rat retinal ganglion cells: uncompetitive antagonism. J Physiol 499: 27-46.
    • (1997) J Physiol , vol.499 , pp. 27-46
    • Chen, H.V.1    Lipton, S.2
  • 5
    • 0026564448 scopus 로고
    • Open-channel block of N-methyl-D-aspartate (NMDA) responses by memantine: Therapeutic advantage against NMDA receptor-mediated toxicity
    • Chen HSV, Pellegrini JW, Aggarwal SK, Lei SZ, Warach S, Jensen FE and Lipton SA (1992) Open-channel block of N-methyl-D-aspartate (NMDA) responses by memantine: Therapeutic advantage against NMDA receptor-mediated toxicity. J Neurosci 12:4427-4435.
    • (1992) J Neurosci , vol.12 , pp. 4427-4435
    • Chen, H.S.V.1    Pellegrini, J.W.2    Aggarwal, S.K.3    Lei, S.Z.4    Warach, S.5    Jensen, F.E.6    Lipton, S.A.7
  • 7
    • 0028240582 scopus 로고
    • Sensitive and rapid behavioural differentiation of N-methyl-D-aspartate receptor antagonists
    • Ginski MJ and Witkin JM (1994) Sensitive and rapid behavioural differentiation of N-methyl-D-aspartate receptor antagonists. Psychopharmacology 114:573-582.
    • (1994) Psychopharmacology , vol.114 , pp. 573-582
    • Ginski, M.J.1    Witkin, J.M.2
  • 8
    • 0021256821 scopus 로고
    • The channel blocking action of methonium compounds on rat submandibular ganglion cells
    • Gurney AM and Rang HP (1984) The channel blocking action of methonium compounds on rat submandibular ganglion cells. Br J Pharmacol 82:623-642.
    • (1984) Br J Pharmacol , vol.82 , pp. 623-642
    • Gurney, A.M.1    Rang, H.P.2
  • 9
    • 0001945122 scopus 로고
    • Subtypes of glutamate receptors: Pharmacological classification
    • (Stone TW ed) CRC Press, New York
    • Harris E (1995) Subtypes of glutamate receptors: Pharmacological classification, in CNS Neurotransmitters and Neuromodulators: Glutamate (Stone TW ed) pp 95-125, CRC Press, New York.
    • (1995) CNS Neurotransmitters and Neuromodulators: Glutamate , pp. 95-125
    • Harris, E.1
  • 10
    • 0001249750 scopus 로고
    • Block of N-methyl-D-aspartate-activated current by the anticonvulsant (+)-MK-801: Selective binding to open channels
    • Huettner JE and Bean BP (1988) Block of N-methyl-D-aspartate-activated current by the anticonvulsant (+)-MK-801: selective binding to open channels. Proc Natl Acad Sci USA 86:1307-1311.
    • (1988) Proc Natl Acad Sci USA , vol.86 , pp. 1307-1311
    • Huettner, J.E.1    Bean, B.P.2
  • 11
    • 0027104318 scopus 로고
    • The anticonvulsant (±)-5-aminocarbonyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine (ADCI) selectively blocks NMDA-activated current in cultured rat hippocampal neurones: Kinetic analysis and comparison with dizocilpine
    • Jones SJ and Rogawski MA (1992) The anticonvulsant (±)-5-aminocarbonyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine (ADCI) selectively blocks NMDA-activated current in cultured rat hippocampal neurones: Kinetic analysis and comparison with dizocilpine. Mol Neuropharmacol 2:303-310.
    • (1992) Mol Neuropharmacol , vol.2 , pp. 303-310
    • Jones, S.J.1    Rogawski, M.A.2
  • 12
    • 0342548523 scopus 로고
    • Non-competetive antagonists of excitatory amino acid receptors
    • Kemp JA, Foster AC and Wong EHF (1987) Non-competetive antagonists of excitatory amino acid receptors. Trends Neurosci 16:527-532.
    • (1987) Trends Neurosci , vol.16 , pp. 527-532
    • Kemp, J.A.1    Foster, A.C.2    Wong, E.H.F.3
  • 14
    • 0020646186 scopus 로고
    • Different types of blockade of crustacean acetylcholine-induced currents
    • Lingle C (1983) Different types of blockade of crustacean acetylcholine-induced currents. J Physiol 339:419-437.
    • (1983) J Physiol , vol.339 , pp. 419-437
    • Lingle, C.1
  • 15
    • 0023232903 scopus 로고
    • Use-dependent block of excitatory amino acid currents in cultured neurons by ketamine
    • MacDonald JF, Miljkovic Z and Pennefether P (1987) Use-dependent block of excitatory amino acid currents in cultured neurons by ketamine. J Neurophysiol 58:251-266.
    • (1987) J Neurophysiol , vol.58 , pp. 251-266
    • MacDonald, J.F.1    Miljkovic, Z.2    Pennefether, P.3
  • 17
    • 0030946384 scopus 로고    scopus 로고
    • NR1 and NR2 Subunit contributions to N-methyl-D-aspartate receptor channel blocker pharmacology
    • Monaghan DT and Larsen H (1997) NR1 and NR2 Subunit contributions to N-methyl-D-aspartate receptor channel blocker pharmacology. J Pharmacol Exp Ther 280:614-620.
    • (1997) J Pharmacol Exp Ther , vol.280 , pp. 614-620
    • Monaghan, D.T.1    Larsen, H.2
  • 18
    • 0029086845 scopus 로고
    • Noncompetitive NMDA receptor antagonists with fast open-channel blocking kinetics and strong voltage-dependency as potential therapeutic agents for Alzheimer's dementia
    • Muller WE, Mutschler E and Riederer P (1995) Noncompetitive NMDA receptor antagonists with fast open-channel blocking kinetics and strong voltage-dependency as potential therapeutic agents for Alzheimer's dementia. Pharmacopsychiatry 28:113-124.
    • (1995) Pharmacopsychiatry , vol.28 , pp. 113-124
    • Muller, W.E.1    Mutschler, E.2    Riederer, P.3
  • 19
    • 0024338054 scopus 로고
    • Pathological changes induced in cerebrocortical neurons by phencyclidine and related drugs
    • Olney JW, Labruyere J and Price MT (1989) Pathological changes induced in cerebrocortical neurons by phencyclidine and related drugs. Science 244:1360-1362.
    • (1989) Science , vol.244 , pp. 1360-1362
    • Olney, J.W.1    Labruyere, J.2    Price, M.T.3
  • 20
    • 0030907708 scopus 로고    scopus 로고
    • Multiple mechanisms of ketamine blockade of N-methyl-D-aspartate receptors
    • Orser BA, Pennefather PS and MacDonald JF (1997) Multiple mechanisms of ketamine blockade of N-methyl-D-aspartate receptors. Anesthesiology 86:903-917.
    • (1997) Anesthesiology , vol.86 , pp. 903-917
    • Orser, B.A.1    Pennefather, P.S.2    MacDonald, J.F.3
  • 21
    • 0030828561 scopus 로고    scopus 로고
    • Low-affinity NMDA receptor antagonists: The neuroprotective potential of ARL 15896AR
    • Palmer GC, Miller JA, Cregan EF, Gendron P and Peeling J (1997) Low-affinity NMDA receptor antagonists: The neuroprotective potential of ARL 15896AR. Ann NY Acad Sci 825:220-231.
    • (1997) Ann NY Acad Sci , vol.825 , pp. 220-231
    • Palmer, G.C.1    Miller, J.A.2    Cregan, E.F.3    Gendron, P.4    Peeling, J.5
  • 22
    • 0344624493 scopus 로고    scopus 로고
    • Neuroprotective potential of the low affinity NMDA receptor antagonist ARL 15896AR
    • (Savage LM ed) IBC Biomedical Library Series, Southborough, MA
    • Palmer GC, Murray RJ and McCarthy DJ (1996) Neuroprotective potential of the low affinity NMDA receptor antagonist ARL 15896AR, in Advances in the Understanding of Therapy of Ischemic Stroke, 2nd ed (Savage LM ed) pp 34-64, IBC Biomedical Library Series, Southborough, MA.
    • (1996) Advances in the Understanding of Therapy of Ischemic Stroke, 2nd Ed , pp. 34-64
    • Palmer, G.C.1    Murray, R.J.2    McCarthy, D.J.3
  • 23
    • 0027731677 scopus 로고
    • Patch clamp studies on the kinetics and selectivity of N-methyl-D-aspartate receptor antagonism by memantme (1-amino-3,5-dimethyladmantan)
    • Parsons CG, Gruner R, Rozental J, Millar J and Lodge D (1993) Patch clamp studies on the kinetics and selectivity of N-methyl-D-aspartate receptor antagonism by memantme (1-amino-3,5-dimethyladmantan). Neuropharmacotogy 32:1337-1350.
    • (1993) Neuropharmacotogy , vol.32 , pp. 1337-1350
    • Parsons, C.G.1    Gruner, R.2    Rozental, J.3    Millar, J.4    Lodge, D.5
  • 24
    • 0029971255 scopus 로고    scopus 로고
    • Comparative patch-clamp studies with freshly dissociated rat hippocampal and striatal neurons on the NMDA receptor antagonistic effects of amantadine and memantine
    • Parsons CG, Panchenko VA, Pinchenko VO, Tsyndrenko AY and Krishtal OA (1996) Comparative patch-clamp studies with freshly dissociated rat hippocampal and striatal neurons on the NMDA receptor antagonistic effects of amantadine and memantine. Eur J Neurosci 8:446-454.
    • (1996) Eur J Neurosci , vol.8 , pp. 446-454
    • Parsons, C.G.1    Panchenko, V.A.2    Pinchenko, V.O.3    Tsyndrenko, A.Y.4    Krishtal, O.A.5
  • 25
    • 0028885626 scopus 로고
    • Comparison of the potency, kinetics and voltage-dependency of a series of uncompetitive NMDA receptor antagonists in vitro with anticonvulsive and motor impairment activity in vivo
    • Parsons CG, Quack G, Bresink I, Baran L, Przegalinski E, Kostowski W, Krzascik P, Hartmann S and Danysz W (1995) Comparison of the potency, kinetics and voltage-dependency of a series of uncompetitive NMDA receptor antagonists in vitro with anticonvulsive and motor impairment activity in vivo. Neuropharmacology 34:1238-1258.
    • (1995) Neuropharmacology , vol.34 , pp. 1238-1258
    • Parsons, C.G.1    Quack, G.2    Bresink, I.3    Baran, L.4    Przegalinski, E.5    Kostowski, W.6    Krzascik, P.7    Hartmann, S.8    Danysz, W.9
  • 26
    • 0027176541 scopus 로고
    • Therapeutic potential of excitatory amino acid antagonists: Channel blockers and 2,3-benzodiazepines
    • Rogawski MA (1993) Therapeutic potential of excitatory amino acid antagonists: channel blockers and 2,3-benzodiazepines. Trends Pharmacol Sci 14:325-331.
    • (1993) Trends Pharmacol Sci , vol.14 , pp. 325-331
    • Rogawski, M.A.1
  • 27
    • 0029043964 scopus 로고
    • Anticonvulsant efficacy of ADCI (5-aminocarbonyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine) after acute and chronic dosing in mice
    • Rogawski MA, Lee DQ, Uyakul D, Pannell L, Subramaniam S, Yamaguchi S and Kokate TG (1995) Anticonvulsant efficacy of ADCI (5-aminocarbonyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine) after acute and chronic dosing in mice. Epilepsia 36:566-571.
    • (1995) Epilepsia , vol.36 , pp. 566-571
    • Rogawski, M.A.1    Lee, D.Q.2    Uyakul, D.3    Pannell, L.4    Subramaniam, S.5    Yamaguchi, S.6    Kokate, T.G.7


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