메뉴 건너뛰기




Volumn 37, Issue 10-11, 1998, Pages 1223-1237

Pharmacological differentiation of kainate receptors on neonatal rat spinal motoneurones and dorsal roots

Author keywords

(RS) 2 Amino 3 (5 t butyl 3 hydroxyisoxazol 4 yl)propanoic acid (ATPA); (RS) 3,4 Dicarboxyphenylglycine (3,4 DCPG); (RS) 3,5 Dicarboxyphenylglycine (3,5 DCPG); GYKI53655; Neonatal rat spinal cord; Willardiine analogues

Indexed keywords

1 (4 AMINOPHENYL) 3,4 DIHYDRO 4 METHYL 3 METHYLCARBAMOYL 7,8 METHYLENEDIOXY 5H 2,3 BENZODIAZEPINE; 2 AMINO 5 PHOSPHONOVALERIC ACID; ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; CYCLOTHIAZIDE; GLYCINE DERIVATIVE; KAINIC ACID; KAINIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID; PROPIONIC ACID DERIVATIVE; WILLARDIINE;

EID: 0032192103     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(98)00124-5     Document Type: Conference Paper
Times cited : (20)

References (29)
  • 1
    • 0022979956 scopus 로고
    • The primary afferent depolarizing action of kainate in the rat
    • Agrawal, S.G., Evans, R.H., 1986. The primary afferent depolarizing action of kainate in the rat. British Journal of Pharmacology 87, 345-355.
    • (1986) British Journal of Pharmacology , vol.87 , pp. 345-355
    • Agrawal, S.G.1    Evans, R.H.2
  • 2
    • 0025259963 scopus 로고
    • Cloning of a novel glutamate receptor subunit, GluR5: Expression in the nervous system during development
    • Bettler, B., Boulter, J., Hermans-Borgmeyer, L, et al., 1990. Cloning of a novel glutamate receptor subunit, GluR5: expression in the nervous system during development. Neuron 5, 583-595.
    • (1990) Neuron , vol.5 , pp. 583-595
    • Bettler, B.1    Boulter, J.2    Hermans-Borgmeyer, L.3
  • 3
    • 0029240274 scopus 로고
    • Neurotransmitter receptors. 2. AMPA and kainate receptors
    • Bettler, B., Mulle, C., 1995. Neurotransmitter receptors. 2. AMPA and kainate receptors. Neuropharmacology 34, 123-139.
    • (1995) Neuropharmacology , vol.34 , pp. 123-139
    • Bettler, B.1    Mulle, C.2
  • 6
    • 0030483692 scopus 로고    scopus 로고
    • Activity of 2,3-benzodiazepines at native rat and recombinant human glutamate receptors in vitro: Stereospecificity and selectivity profiles
    • Bleakman, D., Ballyk, B.A., Schoepp, D.D., et al., 1996a. Activity of 2,3-benzodiazepines at native rat and recombinant human glutamate receptors in vitro: stereospecificity and selectivity profiles. Neuropharmacology 35, 1689-1702.
    • (1996) Neuropharmacology , vol.35 , pp. 1689-1702
    • Bleakman, D.1    Ballyk, B.A.2    Schoepp, D.D.3
  • 7
    • 0029979667 scopus 로고    scopus 로고
    • Pharmacological discrimination of GluR5 and GluR6 kainate receptor subtypes by (3S;4aR,6R,8aR)-6-[2-(1(2H)-tetrazole-5-yl)ethyl]decahydro-isoquinoline-3-carboxylic acid
    • Bleakman, D., Schoepp, D.D., Ballyk, B., et al., 1996b. Pharmacological discrimination of GluR5 and GluR6 kainate receptor subtypes by (3S;4aR,6R,8aR)-6-[2-(1(2H)-tetrazole-5-yl)ethyl]decahydro-isoquinoline-3-carboxylic acid. Molecular Pharmacology 49, 581-585.
    • (1996) Molecular Pharmacology , vol.49 , pp. 581-585
    • Bleakman, D.1    Schoepp, D.D.2    Ballyk, B.3
  • 8
    • 0030863091 scopus 로고    scopus 로고
    • A hippocampal GluR5 kainate receptor regulating inhibitory synaptic transmission
    • Clarke, V.R., Ballyk, B.A., Hoo, K.H., et al., 1997. A hippocampal GluR5 kainate receptor regulating inhibitory synaptic transmission. Nature 389, 599-603.
    • (1997) Nature , vol.389 , pp. 599-603
    • Clarke, V.R.1    Ballyk, B.A.2    Hoo, K.H.3
  • 9
    • 0030995878 scopus 로고    scopus 로고
    • Pharmacology and functions of metabotropic glutamate receptors
    • Conn, P.J., Pin, J.P., 1997. Pharmacology and functions of metabotropic glutamate receptors. Annual Review of Pharmacology and Toxicology 37, 205-237.
    • (1997) Annual Review of Pharmacology and Toxicology , vol.37 , pp. 205-237
    • Conn, P.J.1    Pin, J.P.2
  • 11
    • 0020062045 scopus 로고
    • The effects of a series of ω-phosphonic α-carboxylic amino acids on electrically evoked and amino acid induced responses in isolated spinal cord preparations
    • Evans, R.H., Francis, A.A., Jones, A.W., Smith, D.A.S., Watkins, J.C., 1982. The effects of a series of ω-phosphonic α-carboxylic amino acids on electrically evoked and amino acid induced responses in isolated spinal cord preparations. British Journal of Pharmacology 75, 65-75.
    • (1982) British Journal of Pharmacology , vol.75 , pp. 65-75
    • Evans, R.H.1    Francis, A.A.2    Jones, A.W.3    Smith, D.A.S.4    Watkins, J.C.5
  • 12
    • 0029990678 scopus 로고    scopus 로고
    • New developments in the molecular pharmacology of α-amino-3-hydroxy-5-methyl-4-isoxazole propionate and kainate receptors
    • Fletcher, E.J., Lodge, D., 1996. New developments in the molecular pharmacology of α-amino-3-hydroxy-5-methyl-4-isoxazole propionate and kainate receptors. Pharmacology and Therapeutics 70, 65-89.
    • (1996) Pharmacology and Therapeutics , vol.70 , pp. 65-89
    • Fletcher, E.J.1    Lodge, D.2
  • 14
    • 0003131895 scopus 로고
    • Agonists and competitive antagonists: Structure-activity and molecular modelling studies
    • Collingridge, G.L., Watkins, J.C. (Eds.), Oxford University, Oxford
    • Jane, D.E., Olverman, H.J., Watkins, J.C., 1994. Agonists and competitive antagonists: structure-activity and molecular modelling studies. In: Collingridge, G.L., Watkins, J.C. (Eds.), The NMDA Receptor, 2. Oxford University, Oxford.
    • (1994) The NMDA Receptor , vol.2
    • Jane, D.E.1    Olverman, H.J.2    Watkins, J.C.3
  • 15
    • 0030693165 scopus 로고    scopus 로고
    • Synthesis of willardiine and 6-azawillardiine analogues: Pharmacological characterisation on cloned homomeric human AMPA and kainate receptor subtypes
    • Jane, D.E., Hoo, K., Kamboj, R., Deverill, M., Bleakman, D., Mandlezys, A., 1997. Synthesis of willardiine and 6-azawillardiine analogues: Pharmacological characterisation on cloned homomeric human AMPA and kainate receptor subtypes. Journal of Medicinal Chemistry 40, 3645-3650.
    • (1997) Journal of Medicinal Chemistry , vol.40 , pp. 3645-3650
    • Jane, D.E.1    Hoo, K.2    Kamboj, R.3    Deverill, M.4    Bleakman, D.5    Mandlezys, A.6
  • 16
    • 0030836752 scopus 로고    scopus 로고
    • Desensitisation of kainate receptors by kainate, glutamate and diastereomers of 4-methylglutamate
    • Jones, K.A., Wilding, T.J., Heuttner, J.E., Costa, A.M., 1997. Desensitisation of kainate receptors by kainate, glutamate and diastereomers of 4-methylglutamate. Neuropharmacology 36, 853-863.
    • (1997) Neuropharmacology , vol.36 , pp. 853-863
    • Jones, K.A.1    Wilding, T.J.2    Heuttner, J.E.3    Costa, A.M.4
  • 18
    • 0027715150 scopus 로고
    • Selective modulation of desensitization at AMPA versus kainate receptors by cyclothiazide and concanavalin A
    • Partin, K.M., Patneau, D.K., Winters, C.A., Mayer, M.L., Buonanno, A., 1993. Selective modulation of desensitization at AMPA versus kainate receptors by cyclothiazide and concanavalin A. Neuron 11, 1069-1082.
    • (1993) Neuron , vol.11 , pp. 1069-1082
    • Partin, K.M.1    Patneau, D.K.2    Winters, C.A.3    Mayer, M.L.4    Buonanno, A.5
  • 19
    • 0026556811 scopus 로고
    • Activation and desensitization of AMPA/kainate receptors by novel derivatives of willardiine
    • Patneau, D.K., Mayer, M.L., Jane, D.E., Watkins, J.C., 1992. Activation and desensitization of AMPA/kainate receptors by novel derivatives of willardiine. Journal of Neuroscience 12, 595-606.
    • (1992) Journal of Neuroscience , vol.12 , pp. 595-606
    • Patneau, D.K.1    Mayer, M.L.2    Jane, D.E.3    Watkins, J.C.4
  • 20
    • 0027529881 scopus 로고
    • A comparison of the actions of agonists and antagonists at non-NMDA receptors of C fibres and motoneurones of the immature rat spinal cord in vitro
    • Pook, P.C.K., Brugger, F., Hawkins, N.S., Clark, K.C., Watkins, J.C., Evans, R.H., 1993. A comparison of the actions of agonists and antagonists at non-NMDA receptors of C fibres and motoneurones of the immature rat spinal cord in vitro. British Journal of Pharmacology 108, 179.
    • (1993) British Journal of Pharmacology , vol.108 , pp. 179
    • Pook, P.C.K.1    Brugger, F.2    Hawkins, N.S.3    Clark, K.C.4    Watkins, J.C.5    Evans, R.H.6
  • 21
    • 0030810255 scopus 로고    scopus 로고
    • Rat GluR7 and a carboxy-terminal splice variant, GluR7b, are functional kainate receptor subunits with a low sensitivity to glutamate
    • Schiffer, H.H., Swanson, G.T., Heinemann, S.F., 1997. Rat GluR7 and a carboxy-terminal splice variant, GluR7b, are functional kainate receptor subunits with a low sensitivity to glutamate. Neuron 19, 1141-1146.
    • (1997) Neuron , vol.19 , pp. 1141-1146
    • Schiffer, H.H.1    Swanson, G.T.2    Heinemann, S.F.3
  • 22
    • 0029122303 scopus 로고
    • In-vitro and in-vivo antagonism of AMPA receptor activation by (3S, 4aR, 6R, 8aR)-6-[2-(1(2H)-tetrazole-5-yl)ethyl]decahydro-isoquinoline-3-carboxylic acid
    • Schoepp, D.D., Lodge, D., Bleakman, D., et al., 1995. In-vitro and in-vivo antagonism of AMPA receptor activation by (3S, 4aR, 6R, 8aR)-6-[2-(1(2H)-tetrazole-5-yl)ethyl]decahydro-isoquinoline-3-carboxylic acid. Neuropharmacology 34, 1159-1168.
    • (1995) Neuropharmacology , vol.34 , pp. 1159-1168
    • Schoepp, D.D.1    Lodge, D.2    Bleakman, D.3
  • 23
    • 0030995529 scopus 로고    scopus 로고
    • Excitatory amino-acid receptor agonists. Synthesis and pharmacology of analogues of 2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic acid
    • Sløk, F.A., Ebert, B., Lang, Y., Krogsgaard-Larsen, P., Lenz, S. M., Madsen, U., 1997. Excitatory amino-acid receptor agonists. Synthesis and pharmacology of analogues of 2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic acid. European Journal of Medicinal Chemistry 32, 329-338.
    • (1997) European Journal of Medicinal Chemistry , vol.32 , pp. 329-338
    • Sløk, F.A.1    Ebert, B.2    Lang, Y.3    Krogsgaard-Larsen, P.4    Lenz, S.M.5    Madsen, U.6
  • 24
    • 0030669518 scopus 로고    scopus 로고
    • Dicarboxyphenylglycines as selective antagonists of AMPA-induced depolarisations in neonatal rat motoneurones
    • Thomas, N.K., Clayton, P., Jane, D.E., 1997. Dicarboxyphenylglycines as selective antagonists of AMPA-induced depolarisations in neonatal rat motoneurones. European Journal of Pharmacology 338, 111-116.
    • (1997) European Journal of Pharmacology , vol.338 , pp. 111-116
    • Thomas, N.K.1    Clayton, P.2    Jane, D.E.3
  • 26
    • 0031406507 scopus 로고    scopus 로고
    • The synaptic activation of the GluR5 subtype of kainate receptor in the area CA3 of the rat hippocampus
    • Vignes, M., Bleakman, D., Lodge, D., Collingridge, G.L., 1997. The synaptic activation of the GluR5 subtype of kainate receptor in the area CA3 of the rat hippocampus. Neuropharmacology 36, 1477-1481.
    • (1997) Neuropharmacology , vol.36 , pp. 1477-1481
    • Vignes, M.1    Bleakman, D.2    Lodge, D.3    Collingridge, G.L.4
  • 27
    • 0025191432 scopus 로고
    • Structure-activity relationships in the development of excitatory amino acid receptor agonists and competitive antagonists
    • Watkins, J.C., Krogsgaard-Larsen, P., Honoré, T., 1990. Structure-activity relationships in the development of excitatory amino acid receptor agonists and competitive antagonists. Trends in Pharmacological Science 11, 25-33.
    • (1990) Trends in Pharmacological Science , vol.11 , pp. 25-33
    • Watkins, J.C.1    Krogsgaard-Larsen, P.2    Honoré, T.3
  • 28
    • 0028357664 scopus 로고
    • Willardiines differentiate agonist binding sites for kainate-versus AMPA-preferring glutamate receptors in DRG and hippocampal neurones
    • Wong, L.A., Mayer, M.L., Jane, D.E., Watkins, J.C., 1994. Willardiines differentiate agonist binding sites for kainate-versus AMPA-preferring glutamate receptors in DRG and hippocampal neurones. Journal of Neuroscience 14, 3881-3897.
    • (1994) Journal of Neuroscience , vol.14 , pp. 3881-3897
    • Wong, L.A.1    Mayer, M.L.2    Jane, D.E.3    Watkins, J.C.4
  • 29
    • 0026522095 scopus 로고
    • Pharmacological characterization of non-NMDA subtypes of glutamate receptor in the neonatal rat hemisected spinal-cord in vitro
    • Zeman, S., Lodge, D., 1992. Pharmacological characterization of non-NMDA subtypes of glutamate receptor in the neonatal rat hemisected spinal-cord in vitro. British Journal of Pharmacoogy 106, 367-372.
    • (1992) British Journal of Pharmacoogy , vol.106 , pp. 367-372
    • Zeman, S.1    Lodge, D.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.