Desensitization of kainate receptors by kainate, glutamate and diastereomers of 4-methylglutamate

Neuropharmacology

Volumn 36, Issue 6, 1997, Pages 853-863

  Jones, K A ^a,c   Wilding, T J ^b   Huettner, J E ^b   Costa, A M ^a  

^a Symphony Pharmaceuticals   (United States)

^b WASHINGTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

^c H LUNDBECK A S   (Denmark)

Author keywords

4 methylglutamate; Kainate; SYM 2081, kainate receptor, glutamate receptor, GIuR5, GluR6, dorsal root ganglia

Indexed keywords

4 METHYLGLUTAMIC ACID; GLUTAMIC ACID DERIVATIVE; KAINIC ACID; KAINIC ACID RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DIASTEREOISOMER; DRUG RECEPTOR BINDING; HUMAN; HUMAN CELL; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; RECEPTOR BLOCKING; RECEPTOR DOWN REGULATION; SPINAL GANGLION;

ANIMALS; CELLS, CULTURED; GANGLIA, SPINAL; GLUTAMATES; GLUTAMIC ACID; KAINIC ACID; OSMOLAR CONCENTRATION; PATCH-CLAMP TECHNIQUES; RATS; RECEPTORS, KAINIC ACID; STEREOISOMERISM;

EID: 0030836752     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(97)00066-X     Document Type: Article

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