Solution-phase combinatorial chemistry: Synthesis of novel heterocyclic libraries

Chemtracts

Volumn 11, Issue 9, 1998, Pages 639-646

  Barvian, Mark R ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

HETEROCYCLIC COMPOUND; POLYAMINE; PYRIDINOPOLYAMINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; DRUG STRUCTURE; ESCHERICHIA COLI; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; SHORT SURVEY; STREPTOCOCCUS PYOGENES; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

EID: 0031791793     PISSN: 14319268     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Short Survey

References (19)

1. Orthogonal protection refers to the complete and selective removal of one group in the presence of others. For an elegant presentation, see: Eichler, J., Lucka, A.W., Houghten, R.A. Innovation and Perspectives in Solid Phase Synthesis and Combinatorial Chemical Libraries, Collected Papers, 4th International Symposium, Epton, R., ed. Mayflower Scientific: Birmingham, UK, 1996.
2. Recent reviews and treatises: Acc. Chem Res. 1996, 29(3), Thompson, L.A., Ellman, J.A. Chem. Rev. 1996, 96, 555; Wilson, S., Czarnik, A.W. Combinatorial Chemistry: Synthesis and Application. Wiley: New York, 1997; Czarnik, A.W., DeWitt, S.H., eds. A Practical Guide to Combinatorial Chemistry. American Chemical Society: Washington, DC, 1997; Moos, W.H., Pavia, M.R., Kay, B.K., Ellington, A.D., eds. Annual Reports in Combinatorial Chemistry and Molecular Diversity, Vol. 1. ESCOM: Leiden, Netherlands, 1997.
3. Recent reviews and treatises: Acc. Chem Res. 1996, 29(3), Thompson, L.A., Ellman, J.A. Chem. Rev. 1996, 96, 555; Wilson, S., Czarnik, A.W. Combinatorial Chemistry: Synthesis and Application. Wiley: New York, 1997; Czarnik, A.W., DeWitt, S.H., eds. A Practical Guide to Combinatorial Chemistry. American Chemical Society: Washington, DC, 1997; Moos, W.H., Pavia, M.R., Kay, B.K., Ellington, A.D., eds. Annual Reports in Combinatorial Chemistry and Molecular Diversity, Vol. 1. ESCOM: Leiden, Netherlands, 1997.
4. Recent reviews and treatises: Acc. Chem Res. 1996, 29(3), Thompson, L.A., Ellman, J.A. Chem. Rev. 1996, 96, 555; Wilson, S., Czarnik, A.W. Combinatorial Chemistry: Synthesis and Application. Wiley: New York, 1997; Czarnik, A.W., DeWitt, S.H., eds. A Practical Guide to Combinatorial Chemistry. American Chemical Society: Washington, DC, 1997; Moos, W.H., Pavia, M.R., Kay, B.K., Ellington, A.D., eds. Annual Reports in Combinatorial Chemistry and Molecular Diversity, Vol. 1. ESCOM: Leiden, Netherlands, 1997.
5. Recent reviews and treatises: Acc. Chem Res. 1996, 29(3), Thompson, L.A., Ellman, J.A. Chem. Rev. 1996, 96, 555; Wilson, S., Czarnik, A.W. Combinatorial Chemistry: Synthesis and Application. Wiley: New York, 1997; Czarnik, A.W., DeWitt, S.H., eds. A Practical Guide to Combinatorial Chemistry. American Chemical Society: Washington, DC, 1997; Moos, W.H., Pavia, M.R., Kay, B.K., Ellington, A.D., eds. Annual Reports in Combinatorial Chemistry and Molecular Diversity, Vol. 1. ESCOM: Leiden, Netherlands, 1997.
6. Recent reviews and treatises: Acc. Chem Res. 1996, 29(3), Thompson, L.A., Ellman, J.A. Chem. Rev. 1996, 96, 555; Wilson, S., Czarnik, A.W. Combinatorial Chemistry: Synthesis and Application. Wiley: New York, 1997; Czarnik, A.W., DeWitt, S.H., eds. A Practical Guide to Combinatorial Chemistry. American Chemical Society: Washington, DC, 1997; Moos, W.H., Pavia, M.R., Kay, B.K., Ellington, A.D., eds. Annual Reports in Combinatorial Chemistry and Molecular Diversity, Vol. 1. ESCOM: Leiden, Netherlands, 1997.
7. Recent examples: Bailey, N., Cooper, A.W.J., Deal, M.J., Dean, A.W., Gore, A.L.; Hawes, M.C., Judd, D.B., Merritt, A.T., Storer, R., Travers, S., Watson, S.P. Chimia 1997, 51, 832; Darvas, F., Kovacs, L. In High Throughput Screening, Devlin, J.P., ed. Dekker: New York, 1997, pp. 223-242; Boger, D.L., Ozer, R.S., Andersson, C.-M. Bioorg. Med. Chem. Lett. 1997, 7, 1903; Carell, T., Wintner, E.A., BashirHashemi, A., Rebek, J., Jr. Angew Chem. Int. Ed. Eng. 1994, 33, 2059.
8. Recent examples: Bailey, N., Cooper, A.W.J., Deal, M.J., Dean, A.W., Gore, A.L.; Hawes, M.C., Judd, D.B., Merritt, A.T., Storer, R., Travers, S., Watson, S.P. Chimia 1997, 51, 832; Darvas, F., Kovacs, L. In High Throughput Screening, Devlin, J.P., ed. Dekker: New York, 1997, pp. 223-242; Boger, D.L., Ozer, R.S., Andersson, C.-M. Bioorg. Med. Chem. Lett. 1997, 7, 1903; Carell, T., Wintner, E.A., BashirHashemi, A., Rebek, J., Jr. Angew Chem. Int. Ed. Eng. 1994, 33, 2059.
9. Recent examples: Bailey, N., Cooper, A.W.J., Deal, M.J., Dean, A.W., Gore, A.L.; Hawes, M.C., Judd, D.B., Merritt, A.T., Storer, R., Travers, S., Watson, S.P. Chimia 1997, 51, 832; Darvas, F., Kovacs, L. In High Throughput Screening, Devlin, J.P., ed. Dekker: New York, 1997, pp. 223-242; Boger, D.L., Ozer, R.S., Andersson, C.-M. Bioorg. Med. Chem. Lett. 1997, 7, 1903; Carell, T., Wintner, E.A., BashirHashemi, A., Rebek, J., Jr. Angew Chem. Int. Ed. Eng. 1994, 33, 2059.
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