메뉴 건너뛰기




Volumn 71, Issue 5, 1998, Pages 2169-2177

Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor

Author keywords

Adenylyl cyclase; D Lysergic acid diethylamide; Ergopeptines; Serotonin; Serotonin 5 HT6 receptors; Site directed mutagenesis

Indexed keywords

ADENYLATE CYCLASE; LYSERGIDE; SEROTONIN RECEPTOR;

EID: 0031722106     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.1998.71052169.x     Document Type: Article
Times cited : (41)

References (29)
  • 1
    • 0028245619 scopus 로고
    • Molecular biology of 5-HT receptors
    • Boess F. G. and Martin I. L. (1994) Molecular biology of 5-HT receptors. Neuropharmacology 33, 275-317.
    • (1994) Neuropharmacology , vol.33 , pp. 275-317
    • Boess, F.G.1    Martin, I.L.2
  • 6
    • 0024847889 scopus 로고
    • Site-directed mutagenesis of m1 muscarinic acetylcholine receptors: Conserved aspartic acids play important roles in receptor function
    • Fraser C. M., Wang C. D., Robinson D. A., Gocayne J. D., and Venter J. C. (1989) Site-directed mutagenesis of m1 muscarinic acetylcholine receptors: conserved aspartic acids play important roles in receptor function. Mol. Pharmacol. 36, 840-847.
    • (1989) Mol. Pharmacol. , vol.36 , pp. 840-847
    • Fraser, C.M.1    Wang, C.D.2    Robinson, D.A.3    Gocayne, J.D.4    Venter, J.C.5
  • 9
    • 0025881062 scopus 로고
    • Three-dimensional models of neurotransmitter G-binding protein-coupled receptors
    • Hibert M. F., Trumpp-Kallmeyer S., Bruinvels A., and Hoflack J. (1991) Three-dimensional models of neurotransmitter G-binding protein-coupled receptors. Mol. Pharmacol. 40, 8-15.
    • (1991) Mol. Pharmacol. , vol.40 , pp. 8-15
    • Hibert, M.F.1    Trumpp-Kallmeyer, S.2    Bruinvels, A.3    Hoflack, J.4
  • 11
    • 0029117219 scopus 로고
    • 1adrenergic receptor subtype selective agonist binding
    • 1adrenergic receptor subtype selective agonist binding. J. Biol. Chem. 270, 23189-23195.
    • (1995) J. Biol. Chem. , vol.270 , pp. 23189-23195
    • Hwa, J.1    Graham, R.M.2    Perez, D.M.3
  • 12
    • 0028920298 scopus 로고
    • Mapping the binding-site of the dopamine D2 receptor by the substituted-cysteine accessibility method
    • Javitch J. A., Fu D., Chen J., and Karlin A. (1995) Mapping the binding-site of the dopamine D2 receptor by the substituted-cysteine accessibility method. Neuron 14, 825-831.
    • (1995) Neuron , vol.14 , pp. 825-831
    • Javitch, J.A.1    Fu, D.2    Chen, J.3    Karlin, A.4
  • 13
    • 0030068285 scopus 로고    scopus 로고
    • Delineation of the peptide binding site of the human galanin receptor
    • Kask K., Berthold M., Kahl U., Nordvall G., and Bartfai T. (1996) Delineation of the peptide binding site of the human galanin receptor. EMBO J. 15, 236-244.
    • (1996) EMBO J. , vol.15 , pp. 236-244
    • Kask, K.1    Berthold, M.2    Kahl, U.3    Nordvall, G.4    Bartfai, T.5
  • 16
    • 0027481384 scopus 로고
    • Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs
    • Monsma F. J., Shen Y., Ward R. P., Hamblin M. W., and Sibley D. R. (1993) Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs. Mol. Pharmacol. 43, 320-327.
    • (1993) Mol. Pharmacol. , vol.43 , pp. 320-327
    • Monsma, F.J.1    Shen, Y.2    Ward, R.P.3    Hamblin, M.W.4    Sibley, D.R.5
  • 20
    • 0343177634 scopus 로고
    • Glutamic acid-113 serves as the retinylidene Schiff base counterion in bovine rhodopsin
    • Sakmar T. P., Franke R. R., and Khorana H. G. (1989) Glutamic acid-113 serves as the retinylidene Schiff base counterion in bovine rhodopsin. Proc. Natl. Acad. Sci. USA 86, 8309-8313.
    • (1989) Proc. Natl. Acad. Sci. USA , vol.86 , pp. 8309-8313
    • Sakmar, T.P.1    Franke, R.R.2    Khorana, H.G.3
  • 22
    • 0026548156 scopus 로고
    • In vitro mutagenesis and the search for structure-function relationships among G protein-coupled receptors
    • Savarese T. M. and Fraser C. M. (1992) In vitro mutagenesis and the search for structure-function relationships among G protein-coupled receptors. Biochem. J. 283, 1-19.
    • (1992) Biochem. J. , vol.283 , pp. 1-19
    • Savarese, T.M.1    Fraser, C.M.2
  • 25
    • 0028087860 scopus 로고
    • Acetylcholine mustard labels the binding site aspartate in muscarinic acetylcholine receptors
    • Spalding T. A., Birdsall N. J. M., Curtis C. A. M., and Hulme E. C. (1994) Acetylcholine mustard labels the binding site aspartate in muscarinic acetylcholine receptors. J. Biol. Chem. 269, 4092-4097.
    • (1994) J. Biol. Chem. , vol.269 , pp. 4092-4097
    • Spalding, T.A.1    Birdsall, N.J.M.2    Curtis, C.A.M.3    Hulme, E.C.4
  • 26
    • 0023740863 scopus 로고
    • Conserved aspartic acid residues 79 and 113 of the β-adrenergic receptor have different roles in receptor function
    • Strader C. D., Sigal I. S., Candelore M. R., Rands E., Hill W. S., and Dixon R. A. F. (1988) Conserved aspartic acid residues 79 and 113 of the β-adrenergic receptor have different roles in receptor function. J. Biol. Chem. 263, 10267-10271.
    • (1988) J. Biol. Chem. , vol.263 , pp. 10267-10271
    • Strader, C.D.1    Sigal, I.S.2    Candelore, M.R.3    Rands, E.4    Hill, W.S.5    Dixon, R.A.F.6
  • 27
    • 0027175853 scopus 로고
    • Site-directed mutagenesis of the serotonin 5-hydroxytryptamine, receptor: Identification of amino acids necessary for ligand binding and receptor activation
    • Wang C.-D., Gallaher T. K., and Shih J. C. (1993) Site-directed mutagenesis of the serotonin 5-hydroxytryptamine, receptor: identification of amino acids necessary for ligand binding and receptor activation. Mol. Pharmacol. 43, 931-940.
    • (1993) Mol. Pharmacol. , vol.43 , pp. 931-940
    • Wang, C.-D.1    Gallaher, T.K.2    Shih, J.C.3
  • 28
    • 0028180615 scopus 로고
    • 2 dopamine receptors: Mutation of a histidine residue specifically affects the binding of a subgroup of substituted benzamide drugs
    • 2 dopamine receptors: mutation of a histidine residue specifically affects the binding of a subgroup of substituted benzamide drugs. J. Neurochem. 62, 1664-1669.
    • (1994) J. Neurochem. , vol.62 , pp. 1664-1669
    • Woodward, R.1    Daniell, S.J.2    Strange, P.G.3    Naylor, L.H.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.