Interaction of tryptamine and ergoline compounds with threonine 196 in the ligand binding site of the 5-hydroxytryptamine6 receptor

Molecular Pharmacology

Volumn 52, Issue 3, 1997, Pages 515-523

  Boess, Frank G ^a,b   Monsma Jr , Frederick J ^a   Meyer, Valerie ^a   Zwingelstein, Catherine ^a   Sleight, Andrew J ^a  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

^b F HOFFMANN LA ROCHE LTD   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

4 (3 BUTOXY 4 METHOXYBENZYL) 2 IMIDAZOLIDINONE; AMITRIPTYLINE; CLOZAPINE; ERGOLINE DERIVATIVE; MESULERGINE; METERGOLINE; METHYSERGIDE; METITEPINE; MIANSERIN; RITANSERIN; SEROTONIN RECEPTOR; TRYPTAMINE;

AMINO ACID SEQUENCE; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING SITE; GENE MUTATION; HUMAN; HUMAN CELL; HYDROGEN BOND; LIGAND BINDING; MAMMAL; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; SITE DIRECTED MUTAGENESIS;

EID: 0030880426     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.52.3.515     Document Type: Article

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