Functional and radioligand binding characterization of rat 5-HT6 receptors stably expressed in HEK293 cells

Neuropharmacology

Volumn 36, Issue 4-5, 1997, Pages 713-720

  Boess, F G ^a   Monsma Jr , F J ^a   Carolo, C ^a   Meyer, V ^a   Rudler, A ^a   Zwingelstein, C ^a   Sleight, A J ^a  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

Author keywords

5 HT6 receptors; 5 Hydroxytryptamine; Adenylyl cyclase; LSD

Indexed keywords

2 METHYLSEROTONIN; 5 BENZYLOXYTRYPTAMINE; 5 CARBAMOYLTRYPTAMINE; 5 METHOXYTRYPTAMINE; ADENYLATE CYCLASE; AMITRIPTYLINE; BUFOTENINE; CLOZAPINE; CYCLIC AMP; ERGOTAMINE; LISURIDE; LYSERGIDE; MESULERGINE; METERGOLINE; METHYSERGIDE; METITEPINE; MIANSERIN; N METHYLSEROTONIN; N,N,N TRIMETHYLSEROTONIN; PARTIAL AGONIST; RADIOLIGAND; RECEPTOR SUBTYPE; RITANSERIN; SEROTONIN; SEROTONIN 6 RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; SEROTONIN RECEPTOR; TRYPTAMINE; TRYPTAMINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BINDING COMPETITION; CONTROLLED STUDY; DRUG POTENCY; GENE EXPRESSION; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING; RECEPTOR DENSITY;

ADENYLATE CYCLASE; ANIMALS; CELL LINE; DNA, COMPLEMENTARY; KINETICS; LYSERGIC ACID DIETHYLAMIDE; MEMBRANES; MOLECULAR SEQUENCE DATA; RADIOLIGAND ASSAY; RATS; RECEPTORS, SEROTONIN; RNA, MESSENGER; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; TRANSFECTION; TRYPTAMINES;

EID: 0030995586     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(97)00019-1     Document Type: Article

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