Enhanced expression of G protein-coupled receptor kinase 2 selectively increases the sensitivity of A(2A) adenosine receptors to agonist-induced desensitization

British Journal of Pharmacology

Volumn 125, Issue 2, 1998, Pages 347-356

  Mundell, Stuart J ^a   Luty, Jason S ^a   Willets, Jon ^a   Benovic, Jeffrey L ^b   Kelly, Eamonn ^a  

^a UNIVERSITY OF BRISTOL   (United Kingdom)

^b THOMAS JEFFERSON UNIVERSITY   (United States)

Author keywords

A2 adenosine receptor; Desensitization; G protein coupled receptor; G protein coupled receptor kinase; NG108 15 cells

Indexed keywords

ADENOSINE A2A RECEPTOR; ADENOSINE A2B RECEPTOR; ADENOSINE DEAMINASE; ADENYLATE CYCLASE; FLUORIDE SODIUM; FORSKOLIN; ILOPROST; SECRETIN;

ANIMAL CELL; ARTICLE; CELL FREE SYSTEM; CONTROLLED STUDY; GLIOMA CELL; MOUSE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION;

ADENYLATE CYCLASE; ANIMALS; BETA-ADRENERGIC RECEPTOR KINASE; BINDING, COMPETITIVE; CYCLIC AMP; CYCLIC AMP-DEPENDENT PROTEIN KINASES; GENE EXPRESSION; MICE; RATS; RECEPTOR, ADENOSINE A2A; RECEPTORS, CELL SURFACE; RECEPTORS, PURINERGIC P1; TRANSFECTION; TUMOR CELLS, CULTURED;

EID: 0031664668     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702081     Document Type: Article

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