Solution-phase combinatorial synthesis via the olefin metathesis reaction

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 4, 1997, Pages 463-468

  Boger, Dale L ^a   Chai, Wenying ^a   Ozer, Rachel S ^a   Andersson, Carl Magnus ^a,b  

^a SCRIPPS RESEARCH INSTITUTE   (United States)

^b LUND UNIVERSITY   (Sweden)

Author keywords

[No Author keywords available]

Indexed keywords

PEPTIDE DERIVATIVE;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; PEPTIDE SYNTHESIS; STEREOCHEMISTRY; TECHNIQUE;

EID: 0031576842     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00043-7     Document Type: Article

References (58)

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18. 10. Reviews: Balkenhohl, F.; von dem Bussche-Hünnefeld, C.; Lansky, A.; Zechel, C. Angew. Chem., Int. Ed. Engl. 1996, 35, 2288. Gordon, E. M.; Gallop, M. A.; Patel, D. V. Acc. Chem. Res. 1996, 29, 144. Ellman, J. A. Acc. Chem. Res. 1996, 29, 132. Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron 1995, 51, 8135. Gallop, M. A.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gordon, E. M. J. Med. Chem. 1994, 37, 1233 and 1385. Janda, K. D. Proc. Natl. Acad. Sci. U.S.A. 1994, 91, 10779. Pavia, M. R.; Sawyer, T. K.; Moos, W. H. Bioorg. Med. Chem. Lett. 1993, 3, 387. Books and monographs: Molecular Diversity and Combinatorial Chemistry: Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; ACS: Washington, 1996. Combinatorial Libraries-Synthesis, Screening, and Application Potential, Cortese, R., Ed.; Walter de Gruyter: Berlin, 1996. Combinatorial Libraries: The Theory and Practice of Combinatorial Chemistry, Houghten, R. A., Ed.; ESCOM: Leiden, 1995. Symposium-in-Print: Bioorg. Med. Chem. Lett. 1993, 3, 381-476. Bioorg. Med. Chem. 1996, 4, 631-738.
19. 10. Reviews: Balkenhohl, F.; von dem Bussche-Hünnefeld, C.; Lansky, A.; Zechel, C. Angew. Chem., Int. Ed. Engl. 1996, 35, 2288. Gordon, E. M.; Gallop, M. A.; Patel, D. V. Acc. Chem. Res. 1996, 29, 144. Ellman, J. A. Acc. Chem. Res. 1996, 29, 132. Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron 1995, 51, 8135. Gallop, M. A.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gordon, E. M. J. Med. Chem. 1994, 37, 1233 and 1385. Janda, K. D. Proc. Natl. Acad. Sci. U.S.A. 1994, 91, 10779. Pavia, M. R.; Sawyer, T. K.; Moos, W. H. Bioorg. Med. Chem. Lett. 1993, 3, 387. Books and monographs: Molecular Diversity and Combinatorial Chemistry: Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; ACS: Washington, 1996. Combinatorial Libraries-Synthesis, Screening, and Application Potential, Cortese, R., Ed.; Walter de Gruyter: Berlin, 1996. Combinatorial Libraries: The Theory and Practice of Combinatorial Chemistry, Houghten, R. A., Ed.; ESCOM: Leiden, 1995. Symposium-in-Print: Bioorg. Med. Chem. Lett. 1993, 3, 381-476. Bioorg. Med. Chem. 1996, 4, 631-738.
20. 10. Reviews: Balkenhohl, F.; von dem Bussche-Hünnefeld, C.; Lansky, A.; Zechel, C. Angew. Chem., Int. Ed. Engl. 1996, 35, 2288. Gordon, E. M.; Gallop, M. A.; Patel, D. V. Acc. Chem. Res. 1996, 29, 144. Ellman, J. A. Acc. Chem. Res. 1996, 29, 132. Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron 1995, 51, 8135. Gallop, M. A.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gordon, E. M. J. Med. Chem. 1994, 37, 1233 and 1385. Janda, K. D. Proc. Natl. Acad. Sci. U.S.A. 1994, 91, 10779. Pavia, M. R.; Sawyer, T. K.; Moos, W. H. Bioorg. Med. Chem. Lett. 1993, 3, 387. Books and monographs: Molecular Diversity and Combinatorial Chemistry: Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; ACS: Washington, 1996. Combinatorial Libraries-Synthesis, Screening, and Application Potential, Cortese, R., Ed.; Walter de Gruyter: Berlin, 1996. Combinatorial Libraries: The Theory and Practice of Combinatorial Chemistry, Houghten, R. A., Ed.; ESCOM: Leiden, 1995. Symposium-in-Print: Bioorg. Med. Chem. Lett. 1993, 3, 381-476. Bioorg. Med. Chem. 1996, 4, 631-738.
21. 10. Reviews: Balkenhohl, F.; von dem Bussche-Hünnefeld, C.; Lansky, A.; Zechel, C. Angew. Chem., Int. Ed. Engl. 1996, 35, 2288. Gordon, E. M.; Gallop, M. A.; Patel, D. V. Acc. Chem. Res. 1996, 29, 144. Ellman, J. A. Acc. Chem. Res. 1996, 29, 132. Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron 1995, 51, 8135. Gallop, M. A.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gordon, E. M. J. Med. Chem. 1994, 37, 1233 and 1385. Janda, K. D. Proc. Natl. Acad. Sci. U.S.A. 1994, 91, 10779. Pavia, M. R.; Sawyer, T. K.; Moos, W. H. Bioorg. Med. Chem. Lett. 1993, 3, 387. Books and monographs: Molecular Diversity and Combinatorial Chemistry: Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; ACS: Washington, 1996. Combinatorial Libraries-Synthesis, Screening, and Application Potential, Cortese, R., Ed.; Walter de Gruyter: Berlin, 1996. Combinatorial Libraries: The Theory and Practice of Combinatorial Chemistry, Houghten, R. A., Ed.; ESCOM: Leiden, 1995. Symposium-in-Print: Bioorg. Med. Chem. Lett. 1993, 3, 381-476. Bioorg. Med. Chem. 1996, 4, 631-738.
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