Applications of solid-phase synthesis to drug discovery

Current Medicinal Chemistry

Volumn 4, Issue 3, 1997, Pages 211-227

  Cowley, Phillip M ^a   Rees, David C ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 THIAZOLIDINONE DERIVATIVE; ALPHA 1 ADRENERGIC RECEPTOR; BENZODIAZEPINE DERIVATIVE; CAPTOPRIL; CARBONATE DEHYDRATASE INHIBITOR; CHIR 2279; CHIR 4531; CHOLECYSTOKININ A RECEPTOR; CIPROFLOXACIN; CIPROFLOXACIN DERIVATIVE; CYCLOOXYGENASE 1 INHIBITOR; DIAZEPAM; DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; FLUNITRAZEPAM; GLYCINE DERIVATIVE; HORMONE RECEPTOR; MEMBRANE PROTEIN; MU OPIATE RECEPTOR; NITRAZEPAM; NORDAZEPAM; PHENYTOIN; PHENYTOIN DERIVATIVE; PIPERIDINE DERIVATIVE; PRAZOSIN; PROSTAGLANDIN SYNTHASE INHIBITOR; PYRROLIDINE DERIVATIVE; RADIOLIGAND; SULFONAMIDE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

BINDING AFFINITY; DRUG ACTIVITY; DRUG RECEPTOR BINDING; DRUG RESEARCH; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; LIBRARY; LIGAND BINDING; NONHUMAN; REVIEW; SOLID PHASE SYNTHESIS; TECHNIQUE;

EID: 0030861795     PISSN: 09298673     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

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