2-(Anilino)imidazolines and 2-(benzyl)imidazoline derivatives as h5-HT 1D serotonin receptor ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 18, 2004, Pages 4697-4699

  Prisinzano, Thomas ^a   Dukat, Małgorzata ^a   Law, Ho ^a   Slassi, Abdelmalik ^b   MacLean, Neil ^b   DeLannoy, Inés ^b   Glennon, Richard A ^a  

^a UNIVERSITY OF RICHMOND   (United States)

^b NPS Pharmaceuticals   (Canada)

Author keywords

Serotonin migraine

Indexed keywords

IMIDAZOLINE DERIVATIVE; SEROTONIN 1D AGONIST; SEROTONIN 1D RECEPTOR;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG BRAIN LEVEL; DRUG RECEPTOR BINDING; NONHUMAN; RABBIT;

ADENYLATE CYCLASE; ANILINE COMPOUNDS; ANIMALS; BENZYL COMPOUNDS; HUMANS; IMIDAZOLINES; LIGANDS; MUSCLE, SMOOTH, VASCULAR; RADIOLIGAND ASSAY; RATS; RECEPTOR, SEROTONIN, 5-HT1D; SAPHENOUS VEIN; SEROTONIN AGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 8544247195     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.06.085     Document Type: Article

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