Cannabidiol, a novel inverse agonist for GPR12

Biochemical and Biophysical Research Communications

Volumn 493, Issue 1, 2017, Pages 451-454

  Brown, Kevin J ^a   Laun, Alyssa S ^a   Song, Zhao Hui ^a  

^a University of Louisville School of Medicine   (United States)

Author keywords

Cannabidiol; GPR12; Inverse agonist; Orphan receptor

Indexed keywords

CANNABIDIOL; CHOLERA TOXIN; CYCLIC AMP; G PROTEIN COUPLED RECEPTOR; G PROTEIN COUPLED RECEPTOR 12; HYDROXYL GROUP; INHIBITORY GUANINE NUCLEOTIDE BINDING PROTEIN; PERTUSSIS TOXIN; STIMULATORY GUANINE NUCLEOTIDE BINDING PROTEIN; UNCLASSIFIED DRUG; GPR12 PROTEIN, HUMAN;

ARTICLE; CAMP ASSAY; CONTROLLED STUDY; DRUG TARGETING; HUMAN; HUMAN CELL; METASTASIS INHIBITION; METASTATIC CELL LINE; PRIORITY JOURNAL; PROTEIN EXPRESSION; RECEPTOR UPREGULATION; STRUCTURE ACTIVITY RELATION; VISCOELASTICITY; AGONISTS; DOSE RESPONSE; HEK293 CELL LINE; METABOLISM;

CANNABIDIOL; CYCLIC AMP; DOSE-RESPONSE RELATIONSHIP, DRUG; HEK293 CELLS; HUMANS; RECEPTORS, G-PROTEIN-COUPLED;

EID: 85029511577     PISSN: 0006291X     EISSN: 10902104     Source Type: Journal    
DOI: 10.1016/j.bbrc.2017.09.001     Document Type: Article

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