메뉴 건너뛰기




Volumn 1, Issue 3, 2010, Pages 139-146

Effect of toremifene and ospemifene, compared to acolbifene, on estrogen-sensitive parameters in rat and human uterine tissues

Author keywords

acolbifene; Ishikawa cells; ospemifene; rat uterus; toremifene

Indexed keywords

ACOLBIFENE; ALKALINE PHOSPHATASE; ESTRADIOL; ESTROGEN; OSPEMIFENE; TOREMIFENE;

EID: 84987844143     PISSN: 18681883     EISSN: 18681891     Source Type: Journal    
DOI: 10.1515/HMBCI.2010.016     Document Type: Article
Times cited : (5)

References (38)
  • 1
    • 0037435046 scopus 로고    scopus 로고
    • Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions
    • Jordan VC. Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions. J Med Chem 2003;46:883-908.
    • (2003) J Med Chem , vol.46 , pp. 883-908
    • Jordan, V.1
  • 2
    • 0037468902 scopus 로고    scopus 로고
    • Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 2. Clinical considerations and new agents
    • Jordan VC. Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 2. Clinical considerations and new agents. J Med Chem 2003;46:1081-111.
    • (2003) J Med Chem , vol.46 , pp. 1081-1111
    • Jordan, V.1
  • 5
    • 0033649898 scopus 로고    scopus 로고
    • Selective estrogen receptor modulators (SERMs) in clinical practice
    • Plouffe L. Jr. Selective estrogen receptor modulators (SERMs) in clinical practice. J Soc Gynecol Investig 2000;7(Suppl 1): S38-S46.
    • (2000) J Soc Gynecol Investig , vol.7 , pp. S38-S46
    • Plouffe, L.1
  • 6
    • 0346618937 scopus 로고
    • Crossed coupling of functionalised ketones by low valent titanium (the McMurry reaction): a new stereo-selective synthesis of tamoxifen
    • Coe PL., Scriven CE. Crossed coupling of functionalised ketones by low valent titanium (the McMurry reaction): a new stereo-selective synthesis of tamoxifen. J Chem Soc Perkin Trans 1986;1:475.
    • (1986) J Chem Soc Perkin Trans , vol.1 , pp. 475
    • Coe, P.1    Scriven, C.2
  • 7
    • 0034837530 scopus 로고    scopus 로고
    • Catalytic asymmetric solid-phase cyclopropanation
    • Nagashima T., Davies HM. Catalytic asymmetric solid-phase cyclopropanation. J Am Chem Soc 2001;123:2695-6.
    • (2001) J Am Chem Soc , vol.123 , pp. 2695-2696
    • Nagashima, T.1    Davies, H.2
  • 8
    • 0029893855 scopus 로고    scopus 로고
    • New highly stereoselective synthesis of (Z)-4-hydroxytamoxifen and (Z)-4-hydroxytoremifene via McMurry reaction
    • Gauthier S., Mailhot J., Labrie F. New highly stereoselective synthesis of (Z)-4-hydroxytamoxifen and (Z)-4-hydroxytoremifene via McMurry reaction. J Org Chem 1996;61:3890-3.
    • (1996) J Org Chem , vol.61 , pp. 3890-3893
    • Gauthier, S.1    Mailhot, J.2    Labrie, F.3
  • 10
    • 0030860885 scopus 로고    scopus 로고
    • Blockade of the stimulatory effect of estrogens., OH-tamoxifen., OH-toremifene., droloxifene and raloxifene on alkaline phosphatase activity by the antiestro-gen EM-800 in human endometrial adenocarcinoma Ishikawa cells
    • Simard J., Sanchez R., Poirier D., Gauthier S., Singh SM., Merand Y., Bélanger A., Labrie C., Labrie F. Blockade of the stimulatory effect of estrogens., OH-tamoxifen., OH-toremifene., droloxifene and raloxifene on alkaline phosphatase activity by the antiestro-gen EM-800 in human endometrial adenocarcinoma Ishikawa cells. Cancer Res 1997;57:3494-7.
    • (1997) Cancer Res , vol.57 , pp. 3494-3497
    • Simard, J.1    Sanchez, R.2    Poirier, D.3    Gauthier, S.4    Singh, S.5    Merand, Y.6    Bélanger, A.7    Labrie, C.8    Labrie, F.9
  • 11
    • 0025605629 scopus 로고
    • A simple and sensitive microtiter plate estrogen bio-assay based on stimulation of alkaline phosphatase in Ishikawa cells: estrogenic action of Δ5 adrenal steroids
    • Littlefield BA., Gurpide E., Markiewicz L., McKinley B., Hoch-berg RB. A simple and sensitive microtiter plate estrogen bio-assay based on stimulation of alkaline phosphatase in Ishikawa cells: estrogenic action of Δ5 adrenal steroids. Endocrinology 1990;127:2757-62.
    • (1990) Endocrinology , vol.127 , pp. 2757-2762
    • Littlefield, B.1    Gurpide, E.2    Markiewicz, L.3    McKinley, B.4    Hoch-berg, R.5
  • 12
    • 0016231072 scopus 로고
    • Apparent positive cooperative effect in cyclic AMP and corticosterone production by isolated adrenal cells in response to ACTH analogues
    • Rodbard D. Apparent positive cooperative effect in cyclic AMP and corticosterone production by isolated adrenal cells in response to ACTH analogues. Endocrinology 1974;94:1427-37.
    • (1974) Endocrinology , vol.94 , pp. 1427-1437
    • Rodbard, D.1
  • 13
    • 0000882795 scopus 로고
    • Extension of multiple range tests to group means with unique numbers of replications
    • Kramer CY. Extension of multiple range tests to group means with unique numbers of replications. Biometrics 1956;12: 307-10.
    • (1956) Biometrics , vol.12 , pp. 307-310
    • Kramer, C.1
  • 16
    • 17744368482 scopus 로고    scopus 로고
    • Selective estrogenic effects of a novel triphenylethylene compound., FC1271a., on bone., cholesterol level., and reproductive tissues in intact and ovariectomized rats
    • Qu Q., Zheng H., Dahllund J., Laine A., Cockcroft N., Peng Z., Koskinen M., Hemminki K., Kangas L., Vaananen K., Harkonen P. Selective estrogenic effects of a novel triphenylethylene compound., FC1271a., on bone., cholesterol level., and reproductive tissues in intact and ovariectomized rats. Endocrinology 2000; 141:809-20.
    • (2000) Endocrinology , vol.141 , pp. 809-820
    • Qu, Q.1    Zheng, H.2    Dahllund, J.3    Laine, A.4    Cockcroft, N.5    Peng, Z.6    Koskinen, M.7    Hemminki, K.8    Kangas, L.9    Vaananen, K.10    Harkonen, P.11
  • 19
    • 0037052731 scopus 로고    scopus 로고
    • Comparison of the effects of EM-652 (SCH 57068), Tamoxifen., toremifene., droloxifene., idoxifene., GW-5638 and raloxifene on the growth of human ZR-75-1 breast tumors in nude mice
    • Gutman M., Couillard S., Roy J., Labrie F., Candas B., Labrie C. Comparison of the effects of EM-652 (SCH 57068), Tamoxifen., toremifene., droloxifene., idoxifene., GW-5638 and raloxifene on the growth of human ZR-75-1 breast tumors in nude mice. Int J Cancer 2002;99:273-8.
    • (2002) Int J Cancer , vol.99 , pp. 273-278
    • Gutman, M.1    Couillard, S.2    Roy, J.3    Labrie, F.4    Candas, B.5    Labrie, C.6
  • 21
    • 0029994748 scopus 로고    scopus 로고
    • Raloxifene., tamoxifen., nafoxi-dine., or estrogen effects on reproductive and nonreproductive tissues in ovariectomized rats
    • Sato M., Rippy MK., Bryant HU. Raloxifene., tamoxifen., nafoxi-dine., or estrogen effects on reproductive and nonreproductive tissues in ovariectomized rats. FASEB J 1996;10:905-12.
    • (1996) FASEB J , vol.10 , pp. 905-912
    • Sato, M.1    Rippy, M.2    Bryant, H.3
  • 22
    • 0031171316 scopus 로고    scopus 로고
    • Activity of raloxifene in immature and ovariectomized rat uterotrophic assays
    • Ashby J., Odum J., Foster JR. Activity of raloxifene in immature and ovariectomized rat uterotrophic assays. Regul Toxicol Pharmacol 1997;25:226-31.
    • (1997) Regul Toxicol Pharmacol , vol.25 , pp. 226-231
    • Ashby, J.1    Odum, J.2    Foster, J.3
  • 25
    • 0642367765 scopus 로고    scopus 로고
    • Effects of ospemifene., a novel SERM., on hormones., genital tract., climacteric symptoms., and quality of life in postmenopausal women: a double-blind., randomized trial
    • Rutanen EM., Heikkinen J., Halonen K., Komi J., Lammintausta R., Ylikorkala O. Effects of ospemifene., a novel SERM., on hormones., genital tract., climacteric symptoms., and quality of life in postmenopausal women: a double-blind., randomized trial. Menopause 2003;10:433-9.
    • (2003) Menopause , vol.10 , pp. 433-439
    • Rutanen, E.1    Heikkinen, J.2    Halonen, K.3    Komi, J.4    Lammintausta, R.5    Ylikorkala, O.6
  • 27
    • 0027201832 scopus 로고
    • Synthetic anti-estrogens modulate induction of pS2 and cathepsin-D messenger ribonucleic acid by growth factors and adenosine 3', 5'-mono-phosphate in MCF7 cells
    • Chalbos D., Philips A., Galtier F., Rochefort H. Synthetic anti-estrogens modulate induction of pS2 and cathepsin-D messenger ribonucleic acid by growth factors and adenosine 3',5'-mono-phosphate in MCF7 cells. Endocrinology 1993;133:571-6.
    • (1993) Endocrinology , vol.133 , pp. 571-576
    • Chalbos, D.1    Philips, A.2    Galtier, F.3    Rochefort, H.4
  • 28
    • 0023915865 scopus 로고
    • Contrasting actions of tamoxifen on endometrial and breast tumor growth in the athymic mouse
    • Gottardis MM., Robinson SP., Satyaswaroop PG., Jordan VC. Contrasting actions of tamoxifen on endometrial and breast tumor growth in the athymic mouse. Cancer Res 1988; 48:812-5.
    • (1988) Cancer Res , vol.48 , pp. 812-815
    • Gottardis, M.1    Robinson, S.2    Satyaswaroop, P.3    Jordan, V.4
  • 30
    • 0024396042 scopus 로고
    • Down-regulation of estrogen receptors by androgens in the ZR-75-1 human breast cancer cell line
    • Poulin R., Simard J., Labrie C., Petitclerc L., Dumont M., Lagace L., Labrie F. Down-regulation of estrogen receptors by androgens in the ZR-75-1 human breast cancer cell line. Endocrinology 1989;125:392-9.
    • (1989) Endocrinology , vol.125 , pp. 392-399
    • Poulin, R.1    Simard, J.2    Labrie, C.3    Petitclerc, L.4    Dumont, M.5    Lagace, L.6    Labrie, F.7
  • 31
    • 0024847508 scopus 로고
    • Comparative studies on the effects of steroidal and nonsteroidal oestrogen antagonists on the proliferation of human breast cancer cells
    • Wakeling AE. Comparative studies on the effects of steroidal and nonsteroidal oestrogen antagonists on the proliferation of human breast cancer cells. J Steroid Biochem 1989;34:183-8.
    • (1989) J Steroid Biochem , vol.34 , pp. 183-188
    • Wakeling, A.1
  • 32
    • 0028287647 scopus 로고
    • Effects of tamoxifen on uterus and ovaries of postmenopausal women in a randomized breast cancer prevention trial
    • Kedar RP., Bourne TH., Powles TJ., Collins WP., Ashley SE., Cos-grove DO., Campbell S. Effects of tamoxifen on uterus and ovaries of postmenopausal women in a randomized breast cancer prevention trial. Lancet 1994;343:1318-21.
    • (1994) Lancet , vol.343 , pp. 1318-1321
    • Kedar, R.1    Bourne, T.2    Powles, T.3    Collins, W.4    Ashley, S.5    Cos-grove, D.6    Campbell, S.7
  • 33
    • 0028793795 scopus 로고
    • A retrospective study of tamoxifen and endometrial cancer in breast cancer patients
    • Robinson DC., Bloss JD., Schiano MA. A retrospective study of tamoxifen and endometrial cancer in breast cancer patients. Gynecol Oncol 1995;59:186-90.
    • (1995) Gynecol Oncol , vol.59 , pp. 186-190
    • Robinson, D.1    Bloss, J.2    Schiano, M.3
  • 34
    • 0035815248 scopus 로고    scopus 로고
    • Prospective study on gynaecological effects of two antioestrogens tamoxifen and toremifene in postmenopausal women
    • Marttunen MB., Cacciatore B., Hietanen P., Pyrhonen S., Tiitinen A., Wahlstrom T., Ylikorkala O. Prospective study on gynaecological effects of two antioestrogens tamoxifen and toremifene in postmenopausal women. Br J Cancer 2001;84:897-902.
    • (2001) Br J Cancer , vol.84 , pp. 897-902
    • Marttunen, M.1    Cacciatore, B.2    Hietanen, P.3    Pyrhonen, S.4    Tiitinen, A.5    Wahlstrom, T.6    Ylikorkala, O.7
  • 36
    • 0027412216 scopus 로고
    • High-grade endometrial carcinoma in tamoxifen-treated breast cancer patients
    • Magriples U., Naftolin F., Schwartz PE., Carcangiu ML. High-grade endometrial carcinoma in tamoxifen-treated breast cancer patients. J Clin Oncol 1993;11:485-90.
    • (1993) J Clin Oncol , vol.11 , pp. 485-490
    • Magriples, U.1    Naftolin, F.2    Schwartz, P.3    Carcangiu, M.4
  • 37
    • 0025239673 scopus 로고
    • Tamoxifen for breast cancer: associated endometrial cancer
    • Gusberg SB. Tamoxifen for breast cancer: associated endometrial cancer. Cancer 1990;65:1463-4.
    • (1990) Cancer , vol.65 , pp. 1463-1464
    • Gusberg, S.1
  • 38
    • 23244446876 scopus 로고    scopus 로고
    • Effects of dehydro-epiandrosterone., Premarin and Acolbifene on histomorphology and sex steroid receptors in the rat vagina
    • Berger L., El-Alfy M., Martel C., Labrie F. Effects of dehydro-epiandrosterone., Premarin and Acolbifene on histomorphology and sex steroid receptors in the rat vagina. J Steroid Biochem Mol Biol 2005;96:201-15.
    • (2005) J Steroid Biochem Mol Biol , vol.96 , pp. 201-215
    • Berger, L.1    El-Alfy, M.2    Martel, C.3    Labrie, F.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.