메뉴 건너뛰기




Volumn 17, Issue 4, 2002, Pages 307-315

Analysis and Prediction of Absorption Behavior for Theophylline Orally Administered as Powders Based on Gastrointestinal-transit-Absorption (Gita) Model

Author keywords

biopharmaceutics classi cation system class I; gastrointestinal transit absorption (GITA) model; oral absorption; powder; prediction; theophylline

Indexed keywords


EID: 84982814204     PISSN: 13474367     EISSN: 18800920     Source Type: Journal    
DOI: 10.2133/dmpk.17.307     Document Type: Article
Times cited : (17)

References (30)
  • 2
    • 0031680610 scopus 로고    scopus 로고
    • Absorption behavior of orally administered drugs in rats treated with propantheline
    • Haruta, S., Iwasaki, N., Ogawara, K., Higaki, K. and Kimura, T.: Absorption behavior of orally administered drugs in rats treated with propantheline. J. Pharm. Sci., 87: 1081-1085 (1998).
    • (1998) J. Pharm. Sci. , vol.87 , pp. 1081-1085
    • Haruta, S.1    Iwasaki, N.2    Ogawara, K.3    Higaki, K.4    Kimura, T.5
  • 3
    • 0022639241 scopus 로고
    • Allopurinol absorption from diŝerent sites of the rat gastrointestinal tract
    • Patel, V. S. and Kramer, W. G.: Allopurinol absorption from diŝerent sites of the rat gastrointestinal tract. J. Pharm. Sci., 75: 275-277 (1986).
    • (1986) J. Pharm. Sci. , vol.75 , pp. 275-277
    • Patel, V.S.1    Kramer, W.G.2
  • 5
    • 0013826475 scopus 로고
    • Intestinal absorption of riboflavin by man.
    • Stripp, B.: Intestinal absorption of riboflavin by man. Acta Pharmacol. Toxicol., 22: 353-362 (1965).
    • (1965) Acta Pharmacol. Toxicol. , vol.22 , pp. 353-362
    • Stripp, B.1
  • 6
    • 0028143513 scopus 로고
    • Griseofulvin absorption from diŝerent sites in the human small intestine
    • Gramatte, T.: Griseofulvin absorption from diŝerent sites in the human small intestine. Biopharm. Drug Dispos., 15: 747-759 (1994).
    • (1994) Biopharm. Drug Dispos. , vol.15 , pp. 747-759
    • Gramatte, T.1
  • 7
    • 0036481691 scopus 로고    scopus 로고
    • Gastrointestinal transit and drug absorption
    • Kimura, T. and Higaki, K.: Gastrointestinal transit and drug absorption. Biol. Pharm. Bull., 25: 149-164 (2002).
    • (2002) Biol. Pharm. Bull. , vol.25 , pp. 149-164
    • Kimura, T.1    Higaki, K.2
  • 8
    • 85024461788 scopus 로고    scopus 로고
    • In G. S. Banker and C. T. Rhodes (ed.) Modern Pharmaceutics, 3rd ed., Marcel Dekker, New York
    • Mayerson, M.: Principles of drug absorption, In G. S. Banker and C. T. Rhodes (ed.), Modern Pharmaceutics, 3rd ed., Marcel Dekker, New York, 1996, pp. 21-71.
    • (1996) Principles of drug absorption , pp. 21-71
    • Mayerson, M.1
  • 9
    • 0030581087 scopus 로고    scopus 로고
    • Active secretion and enterocytic drug metabolism barriers to drug absorption
    • Wacher, V. J., Salphati, L. and Benet, L. Z.: Active secretion and enterocytic drug metabolism barriers to drug absorption. Adv. Drug Deliv. Rev., 20: 157-180 (1996).
    • (1996) Adv. Drug Deliv. Rev. , vol.20 , pp. 157-180
    • Wacher, V.J.1    Salphati, L.2    Benet, L.Z.3
  • 10
    • 0030928205 scopus 로고    scopus 로고
    • Prediction of the plasma concentration prô-les of orally administered drugs in rats on the basis of gastrointestinal transit kinetics and absorbability
    • Sawamoto, T., Haruta, S., Kurosaki, Y., Higaki, K. and Kimura, T.: Prediction of the plasma concentration prô-les of orally administered drugs in rats on the basis of gastrointestinal transit kinetics and absorbability. J. Pharm. Pharmacol., 49: 450-457 (1997).
    • (1997) J. Pharm. Pharmacol. , vol.49 , pp. 450-457
    • Sawamoto, T.1    Haruta, S.2    Kurosaki, Y.3    Higaki, K.4    Kimura, T.5
  • 11
    • 0034009449 scopus 로고    scopus 로고
    • Analysis and prediction of absorption prôle including hepatiĉrst-pass metabolism of N-methyltyramine, a potent stimulant of gastrin release present in beer, afer oral ingestion in rats by gastrointestinal-transit-absorption model
    • Kimura, T., Iwasaki, N., Yokoe, J., Haruta, S., Yokoo, Y., Ogawara, K. and Higaki, K.: Analysis and prediction of absorption prôle including hepatiĉrst-pass metabolism of N-methyltyramine, a potent stimulant of gastrin release present in beer, afer oral ingestion in rats by gastrointestinal-transit-absorption model. Drug Metab. Dispos., 28: 577-581 (2000).
    • (2000) Drug Metab. Dispos. , vol.28 , pp. 577-581
    • Kimura, T.1    Iwasaki, N.2    Yokoe, J.3    Haruta, S.4    Yokoo, Y.5    Ogawara, K.6    Higaki, K.7
  • 12
    • 0035070539 scopus 로고    scopus 로고
    • Evaluation of absorption kinetics of orally administered theophylline in rats based on gastrointestinal transit monitoring by gamma scintigraphy
    • Haruta, S., Kawai, K., Jinnouchi, S., Ogawara, K., Higaki, K., Tamura, S., Arimori, K. and Kimura, T.: Evaluation of absorption kinetics of orally administered theophylline in rats based on gastrointestinal transit monitoring by gamma scintigraphy. J. Pharm. Sci., 90: 464-473 (2001).
    • (2001) J. Pharm. Sci. , vol.90 , pp. 464-473
    • Haruta, S.1    Kawai, K.2    Jinnouchi, S.3    Ogawara, K.4    Higaki, K.5    Tamura, S.6    Arimori, K.7    Kimura, T.8
  • 13
    • 0037148655 scopus 로고    scopus 로고
    • Prediction of plasma concentration-time curve of orally administered theophylline based on a scintigraphic monitoring of gastrointestinal transit in human volunteers
    • Haruta, S., Kawai, K., Nishii, R., Jinnouchi, S., Ogawara, K., Higaki, K., Tamura, S., Arimori, K. and Kimura, T.: Prediction of plasma concentration-time curve of orally administered theophylline based on a scintigraphic monitoring of gastrointestinal transit in human volunteers. Int. J. Pharm., 233: 179-190 (2002).
    • (2002) Int. J. Pharm. , vol.233 , pp. 179-190
    • Haruta, S.1    Kawai, K.2    Nishii, R.3    Jinnouchi, S.4    Ogawara, K.5    Higaki, K.6    Tamura, S.7    Arimori, K.8    Kimura, T.9
  • 15
    • 0028948839 scopus 로고
    • A theoretical basis for a biopharmaceutic drug classîcation: The correlation of in vitro drug product dissolution and in vivo bioavailability
    • Amidon, G. L., Lennernas, H., Shah, V. P. and Crison, J. R.: A theoretical basis for a biopharmaceutic drug classîcation: The correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm. Res., 12: 413-420 (1995).
    • (1995) Pharm. Res. , vol.12 , pp. 413-420
    • Amidon, G.L.1    Lennernas, H.2    Shah, V.P.3    Crison, J.R.4
  • 16
    • 0024642303 scopus 로고
    • A nonlinear least squares program. MULTI (FILT), based on fast inverse Laplace transform for microcomputer
    • Yano, Y., Yamaoka, K. and Tanaka, H.: A nonlinear least squares program. MULTI (FILT), based on fast inverse Laplace transform for microcomputer. Chem. Pharm. Bull., 37: 1035-1038 (1989).
    • (1989) Chem. Pharm. Bull. , vol.37 , pp. 1035-1038
    • Yano, Y.1    Yamaoka, K.2    Tanaka, H.3
  • 18
    • 0017698381 scopus 로고
    • Canine gastric emptying of solids and liquids.
    • Hinder, R. A. and Kelly, K. A.: Canine gastric emptying of solids and liquids. Am. J. Physiol., 233: E335-E340 (1977).
    • (1977) Am. J. Physiol. , vol.233 , pp. E335-E340
    • Hinder, R.A.1    Kelly, K.A.2
  • 19
    • 0022149368 scopus 로고
    • Relation between antral motility and gastric emptying of solids and liquids in humans
    • Camilleri, M., Malagelada, J. R., Brown, M. L. and Becker, G.: Relation between antral motility and gastric emptying of solids and liquids in humans. Am. J. Physiol., 249: G580-G585 (1985).
    • (1985) Am. J. Physiol. , vol.249 , pp. G580-G585
    • Camilleri, M.1    Malagelada, J.R.2    Brown, M.L.3    Becker, G.4
  • 21
    • 0025042445 scopus 로고
    • The influence of density on the gastrointestinal transit of pellets
    • Devereux, J. E., Newton, J. M. Short, M. B.: The influence of density on the gastrointestinal transit of pellets. J. Pharm. Pharmacol., 42: 500-501 (1990).
    • (1990) J. Pharm. Pharmacol. , vol.42 , pp. 500-501
    • Devereux, J.E.1    Newton, J.M.2    Short, M.B.3
  • 22
    • 0033034920 scopus 로고    scopus 로고
    • Gastrointestinal transit of pellets in rats: eŝect of size and density
    • Tuleu, C., Andrieux, C., Boy, P. and Chaumeil, J. C.: Gastrointestinal transit of pellets in rats: eŝect of size and density. Int. J. Pharm., 180: 123-131 (1999).
    • (1999) Int. J. Pharm. , vol.180 , pp. 123-131
    • Tuleu, C.1    Andrieux, C.2    Boy, P.3    Chaumeil, J.C.4
  • 23
    • 0001155833 scopus 로고
    • Micromeritics
    • Baltimore, Williams & Wilkins
    • Martin, A. Micromeritics. In Physical Pharmacy. Baltimore, Williams & Wilkins, 1993, pp. 423-452.
    • (1993) In Physical Pharmacy , pp. 423-452
    • Martin, A.1
  • 24
    • 0022538998 scopus 로고
    • Transit of pharmaceutical dosage forms through the small intestine
    • Davis, S. S., Hardy, J. G. and Fara, J. W.: Transit of pharmaceutical dosage forms through the small intestine. Gut, 27: 886-892 (1986).
    • (1986) Gut , vol.27 , pp. 886-892
    • Davis, S.S.1    Hardy, J.G.2    Fara, J.W.3
  • 26
    • 0030576552 scopus 로고    scopus 로고
    • Indirect gastrointestinal transit monitoring and absorption of theophylline.
    • Peh, K. K. and Yuen, K. H.: Indirect gastrointestinal transit monitoring and absorption of theophylline. Int. J. Pharm., 139: 95-103 (1996).
    • (1996) Int. J. Pharm. , vol.139 , pp. 95-103
    • Peh, K.K.1    Yuen, K.H.2
  • 27
    • 85008065764 scopus 로고
    • New method for the evaluation of in vitro dissolution time and disintegration time
    • Tanigawara, Y., Yamaoka, K., Nakagawa, T. and Uno, T.: New method for the evaluation of in vitro dissolution time and disintegration time. Chem. Pharm. Bull., 30: 1088-1090 (1982).
    • (1982) Chem. Pharm. Bull. , vol.30 , pp. 1088-1090
    • Tanigawara, Y.1    Yamaoka, K.2    Nakagawa, T.3    Uno, T.4
  • 28
    • 0019981366 scopus 로고
    • Correlation between in vivo mean dissolution time and in vitro mean dissolution time of ampicillin products
    • Tanigawara, Y., Yamaoka, K., Nakagawa, T. and Uno, T.: Correlation between in vivo mean dissolution time and in vitro mean dissolution time of ampicillin products. J. Pharmacobio-Dyn., 5: 370-372 (1982).
    • (1982) J. Pharmacobio-Dyn. , vol.5 , pp. 370-372
    • Tanigawara, Y.1    Yamaoka, K.2    Nakagawa, T.3    Uno, T.4
  • 29
    • 0000919395 scopus 로고
    • Development of in vitro dissolution tests which correlate quantitatively with dissolution rate-limited drug absorption in man.
    • Levy, G., Leeonards, J. R. and Prockual, J. A.: Development of in vitro dissolution tests which correlate quantitatively with dissolution rate-limited drug absorption in man. J. Pharm. Sci., 54: 1719-1722 (1965).
    • (1965) J. Pharm. Sci. , vol.54 , pp. 1719-1722
    • Levy, G.1    Leeonards, J.R.2    Prockual, J.A.3
  • 30
    • 0014138173 scopus 로고
    • Establishment of sink conditions in dissolution rate determinations: Theoretical considerations and application to nondisintegrating dosage forms
    • Gibaldi, M. and Feldman, S.: Establishment of sink conditions in dissolution rate determinations: Theoretical considerations and application to nondisintegrating dosage forms. J. Pharm. Sci., 56: 1238-1242 (1967).
    • (1967) J. Pharm. Sci. , vol.56 , pp. 1238-1242
    • Gibaldi, M.1    Feldman, S.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.